Drug Gene Type Source 5-(N-Methyl-N-isobutyl)amiloride CCL2 Text_Mining(decreases(reaction)) CTD 5-(N-Methyl-N-isobutyl)amiloride CCL2 Text_Mining(increases(expression)) CTD 5-(N-Methyl-N-isobutyl)amiloride CXCL8 Text_Mining(decreases(reaction)) CTD 5-(N-Methyl-N-isobutyl)amiloride CXCL8 Text_Mining(increases(secretion)) CTD 5-(N-Methyl-N-isobutyl)amiloride CXCL8 Text_Mining(increases(expression)) CTD 5-(N-Methyl-N-isobutyl)amiloride IL1B Text_Mining(decreases(reaction)) CTD 5-(N-Methyl-N-isobutyl)amiloride IL1B Text_Mining(increases(secretion)) CTD 5-(N-Methyl-N-isobutyl)amiloride NFKB1 Text_Mining(affects(localization)) CTD 5-(N-Methyl-N-isobutyl)amiloride NFKB1 Text_Mining(decreases(reaction)) CTD 5-(N-Methyl-N-isobutyl)amiloride NFKB1 Text_Mining(increases(activity)) CTD 5-(N-Methyl-N-isobutyl)amiloride RELA Text_Mining(affects(localization)) CTD 5-(N-Methyl-N-isobutyl)amiloride RELA Text_Mining(decreases(reaction)) CTD 5-(N-Methyl-N-isobutyl)amiloride RELA Text_Mining(increases(activity)) CTD 5-(N-Methyl-N-isobutyl)amiloride CYP1A2 None=None(uM) D4 PubChem 5-(N-Methyl-N-isobutyl)amiloride CYP1A2 AC50=794.33(nM) D4 ChEMBL 5-(N-Methyl-N-isobutyl)amiloride CYP2D6 Potency=39.8107(uM) D4 PubChem 5-(N-Methyl-N-isobutyl)amiloride CYP2D6 None=None(uM) D4 PubChem 5-(N-Methyl-N-isobutyl)amiloride CYP2D6 AC50=39810.7(nM) D4 ChEMBL 5-(N-Methyl-N-isobutyl)amiloride CYP2D6 Potency=39810.7(nM) D4 ChEMBL 5-(N-Methyl-N-isobutyl)amiloride KCNH2 Potency=1.9953(uM) D4 PubChem 5-(N-Methyl-N-isobutyl)amiloride MPHOSPH8 Potency=44.6684(uM) D4 PubChem 5-(N-Methyl-N-isobutyl)amiloride MPHOSPH8 Potency=44668.4(nM) D4 ChEMBL