Drug Gene Type Source orlistat ABHD12 Text_Mining(decreases(activity)) CTD orlistat ABHD16A Text_Mining(decreases(activity)) CTD orlistat ATF4 Text_Mining(increases(expression)) CTD orlistat CASP3 Text_Mining(increases(activity)) CTD orlistat CASP3 Text_Mining(increases(cleavage)) CTD orlistat CASP8 Text_Mining(increases(activity)) CTD orlistat CASP8 Text_Mining(increases(cleavage)) CTD orlistat CCK Text_Mining(decreases(reaction)) CTD orlistat CCK Text_Mining(increases(secretion)) CTD orlistat CCK Text_Mining(decreases(abundance)) CTD orlistat CCK Text_Mining(decreases(secretion)) CTD orlistat CDKN1B Text_Mining(increases(expression)) CTD orlistat CEL Text_Mining(decreases(activity)) CTD orlistat CLPS Text_Mining(affects(cotreatment)) CTD orlistat CLPS Text_Mining(decreases(reaction)) CTD orlistat CLPS Text_Mining(increases(hydrolysis)) CTD orlistat CPB2 Text_Mining(decreases(expression)) CTD orlistat CXCL8 Text_Mining(decreases(reaction)) CTD orlistat CXCL8 Text_Mining(increases(expression)) CTD orlistat CYP3A4 Text_Mining(increases(expression)) CTD orlistat DAGLA Text_Mining(decreases(activity)) CTD orlistat DDIT3 Text_Mining(increases(expression)) CTD orlistat DDIT4 Text_Mining(increases(expression)) CTD orlistat EIF2A Text_Mining(decreases(reaction)) CTD orlistat EIF2A Text_Mining(increases(phosphorylation)) CTD orlistat EIF4E Text_Mining(increases(phosphorylation)) CTD orlistat ERBB2 Text_Mining(affects(response to substance)) CTD orlistat ERBB2 Text_Mining(affects(localization)) CTD orlistat ERBB2 Text_Mining(decreases(expression)) CTD orlistat ERN1 Text_Mining(affects(reaction)) CTD orlistat ERN1 Text_Mining(affects(splicing)) CTD orlistat ETV4 Text_Mining(increases(expression)) CTD orlistat FASN Text_Mining(affects(response to substance)) CTD orlistat FASN Text_Mining(affects(binding)) CTD orlistat FASN Text_Mining(decreases(activity)) CTD orlistat FASN Text_Mining(decreases(reaction)) CTD orlistat FASN Text_Mining(decreases(response to substance)) CTD orlistat FASN Text_Mining(decreases(abundance)) CTD orlistat FASN Text_Mining(decreases(chemical synthesis)) CTD orlistat FASN Text_Mining(decreases(expression)) CTD orlistat GCG Text_Mining(decreases(reaction)) CTD orlistat GCG Text_Mining(increases(secretion)) CTD orlistat GCG Text_Mining(decreases(expression)) CTD orlistat GCG Text_Mining(decreases(secretion)) CTD orlistat GHRL Text_Mining(decreases(expression)) CTD orlistat GHRL Text_Mining(decreases(reaction)) CTD orlistat GHRL Text_Mining(decreases(secretion)) CTD orlistat GIP Text_Mining(decreases(expression)) CTD orlistat GPX8 Text_Mining(increases(expression)) CTD orlistat HBA1 Text_Mining(decreases(expression)) CTD orlistat HSPA5 Text_Mining(increases(expression)) CTD orlistat IL6 Text_Mining(decreases(reaction)) CTD orlistat IL6 Text_Mining(increases(expression)) CTD orlistat INS Text_Mining(affects(expression)) CTD orlistat INS Text_Mining(decreases(expression)) CTD orlistat INS Text_Mining(increases(expression)) CTD orlistat KDELR3 Text_Mining(increases(expression)) CTD orlistat KDR Text_Mining(decreases(expression)) CTD orlistat KRT81 Text_Mining(increases(expression)) CTD orlistat LIPF Text_Mining(decreases(activity)) CTD orlistat LPL Text_Mining(decreases(activity)) CTD orlistat LPL Text_Mining(decreases(reaction)) CTD orlistat LPL Text_Mining(increases(hydrolysis)) CTD orlistat LPL Text_Mining(increases(uptake)) CTD orlistat LPL Text_Mining(increases(activity)) CTD orlistat NPY Text_Mining(increases(expression)) CTD orlistat NR1I2 Text_Mining(increases(activity)) CTD orlistat NTS Text_Mining(decreases(reaction)) CTD orlistat NTS Text_Mining(increases(secretion)) CTD orlistat PARP1 Text_Mining(affects(cotreatment)) CTD orlistat PARP1 Text_Mining(increases(cleavage)) CTD orlistat PLA2G7 Text_Mining(affects(cotreatment)) CTD orlistat PLA2G7 Text_Mining(decreases(activity)) CTD orlistat PNLIP Text_Mining(affects(folding)) CTD orlistat PNLIP Text_Mining(affects(cotreatment)) CTD orlistat PNLIP Text_Mining(decreases(reaction)) CTD orlistat PNLIP Text_Mining(increases(hydrolysis)) CTD orlistat PNLIP Text_Mining(decreases(abundance)) CTD orlistat PNLIP Text_Mining(decreases(secretion)) CTD orlistat PNLIP Text_Mining(decreases(activity)) CTD orlistat PNLIPRP2 Text_Mining(decreases(activity)) CTD orlistat PON1 Text_Mining(increases(activity)) CTD orlistat PPY Text_Mining(decreases(reaction)) CTD orlistat PPY Text_Mining(increases(secretion)) CTD orlistat PYY Text_Mining(decreases(reaction)) CTD orlistat PYY Text_Mining(increases(expression)) CTD orlistat PYY Text_Mining(increases(secretion)) CTD orlistat PYY Text_Mining(decreases(secretion)) CTD orlistat RB1 Text_Mining(decreases(phosphorylation)) CTD orlistat SEC24D Text_Mining(increases(expression)) CTD orlistat SKP2 Text_Mining(decreases(activity)) CTD orlistat SKP2 Text_Mining(decreases(expression)) CTD orlistat SLC22A2 Text_Mining(decreases(reaction)) CTD orlistat SLC22A2 Text_Mining(increases(uptake)) CTD orlistat TNF Text_Mining(decreases(activity)) CTD orlistat TNF Text_Mining(decreases(reaction)) CTD orlistat TNFSF10 Text_Mining(increases(response to substance)) CTD orlistat XBP1 Text_Mining(affects(reaction)) CTD orlistat XBP1 Text_Mining(affects(splicing)) CTD orlistat DAGLA Activity=None(Unspecified) D4 ChEMBL orlistat DAGLB None=None(uM) D4 PubChem orlistat DAGLB Activity=None(Unspecified) D4 ChEMBL orlistat FASN None=None(uM) D4 PubChem orlistat PAFAH2 None=None(uM) D4 PubChem orlistat PLA2G7 None=None(uM) D4 PubChem orlistat PNLIP Activity=None(Unspecified) D4 ChEMBL orlistat TDP1 Potency=18.3564(uM) D4 PubChem orlistat TNNC1 None=None(uM) D4 PubChem orlistat TNNI3 None=None(uM) D4 PubChem orlistat TNNT2 None=None(uM) D4 PubChem