Drug Gene Type Source celastrol AHSA1 Text_Mining(increases(expression)) CTD celastrol AKR1C1 Text_Mining(increases(expression)) CTD celastrol AKR1C2 Text_Mining(increases(expression)) CTD celastrol AKT1 Text_Mining(decreases(phosphorylation)) CTD celastrol AR Text_Mining(decreases(reaction)) CTD celastrol AR Text_Mining(increases(degradation)) CTD celastrol AR Text_Mining(decreases(expression)) CTD celastrol ARID5B Text_Mining(decreases(expression)) CTD celastrol ATF3 Text_Mining(increases(expression)) CTD celastrol BAG3 Text_Mining(increases(expression)) CTD celastrol BAX Text_Mining(increases(expression)) CTD celastrol BCL2 Text_Mining(decreases(expression)) CTD celastrol BIRC5 Text_Mining(decreases(expression)) CTD celastrol BTG1 Text_Mining(decreases(expression)) CTD celastrol C21ORF33 Text_Mining(decreases(expression)) CTD celastrol CACYBP Text_Mining(increases(expression)) CTD celastrol CASP3 Text_Mining(affects(cotreatment)) CTD celastrol CASP3 Text_Mining(increases(cleavage)) CTD celastrol CASP8 Text_Mining(increases(cleavage)) CTD celastrol CASP9 Text_Mining(increases(cleavage)) CTD celastrol CAST Text_Mining(decreases(reaction)) CTD celastrol CAST Text_Mining(increases(degradation)) CTD celastrol CBR3 Text_Mining(increases(expression)) CTD celastrol CDC7 Text_Mining(decreases(expression)) CTD celastrol CDK2 Text_Mining(decreases(expression)) CTD celastrol CHORDC1 Text_Mining(increases(expression)) CTD celastrol CITED2 Text_Mining(decreases(expression)) CTD celastrol CYP1A1 Text_Mining(decreases(expression)) CTD celastrol DDIT3 Text_Mining(increases(expression)) CTD celastrol DDIT4 Text_Mining(increases(expression)) CTD celastrol DNAJA1 Text_Mining(increases(expression)) CTD celastrol DNAJB4 Text_Mining(increases(expression)) CTD celastrol EFNB2 Text_Mining(decreases(expression)) CTD celastrol EGFR Text_Mining(affects(cotreatment)) CTD celastrol EGFR Text_Mining(affects(expression)) CTD celastrol EGFR Text_Mining(decreases(expression)) CTD celastrol FAS Text_Mining(increases(expression)) CTD celastrol FASLG Text_Mining(increases(expression)) CTD celastrol FICD Text_Mining(increases(expression)) CTD celastrol FLT3 Text_Mining(decreases(expression)) CTD celastrol GCLM Text_Mining(increases(expression)) CTD celastrol GDF15 Text_Mining(increases(expression)) CTD celastrol GTPBP2 Text_Mining(increases(expression)) CTD celastrol HILPDA Text_Mining(decreases(expression)) CTD celastrol HMGCS1 Text_Mining(increases(expression)) CTD celastrol HMOX1 Text_Mining(increases(expression)) CTD celastrol HSP90AA1 Text_Mining(decreases(activity)) CTD celastrol HSPA1A Text_Mining(increases(expression)) CTD celastrol HSPA1B Text_Mining(increases(expression)) CTD celastrol HSPA5 Text_Mining(increases(expression)) CTD celastrol HSPH1 Text_Mining(increases(expression)) CTD celastrol ICAM1 Text_Mining(decreases(reaction)) CTD celastrol ICAM1 Text_Mining(increases(expression)) CTD celastrol IFNG Text_Mining(decreases(reaction)) CTD celastrol IFNG Text_Mining(increases(expression)) CTD celastrol IL1B Text_Mining(decreases(reaction)) CTD celastrol IL1B Text_Mining(increases(expression)) CTD celastrol IL1RN Text_Mining(decreases(expression)) CTD celastrol INSIG1 Text_Mining(increases(expression)) CTD celastrol JAG1 Text_Mining(decreases(expression)) CTD celastrol KCNN2 Text_Mining(decreases(expression)) CTD celastrol LDLR Text_Mining(increases(expression)) CTD celastrol LPIN1 Text_Mining(increases(expression)) CTD celastrol LTN1 Text_Mining(decreases(expression)) CTD celastrol MAFB Text_Mining(decreases(expression)) CTD celastrol MDH2 Text_Mining(decreases(expression)) CTD celastrol ME1 Text_Mining(increases(expression)) CTD celastrol MNT Text_Mining(increases(expression)) CTD celastrol MRPL18 Text_Mining(increases(expression)) CTD celastrol MSH6 Text_Mining(decreases(expression)) CTD celastrol MSMO1 Text_Mining(increases(expression)) CTD celastrol MYCBP2 Text_Mining(decreases(expression)) CTD celastrol MYNN Text_Mining(decreases(expression)) CTD celastrol NBN Text_Mining(decreases(expression)) CTD celastrol NKX3-1 Text_Mining(decreases(expression)) CTD celastrol NREP Text_Mining(decreases(expression)) CTD celastrol OPRK1 Text_Mining(decreases(expression)) CTD celastrol OSER1 Text_Mining(increases(expression)) CTD celastrol PARP1 Text_Mining(affects(cotreatment)) CTD celastrol PARP1 Text_Mining(increases(cleavage)) CTD celastrol PARP1 Text_Mining(increases(reaction)) CTD celastrol PDE9A Text_Mining(decreases(expression)) CTD celastrol PIK3CD Text_Mining(decreases(expression)) CTD celastrol PIK3R1 Text_Mining(decreases(expression)) CTD celastrol PPIF Text_Mining(decreases(expression)) CTD celastrol PURA Text_Mining(decreases(expression)) CTD celastrol RELA Text_Mining(affects(localization)) CTD celastrol RELA Text_Mining(decreases(reaction)) CTD celastrol RELA Text_Mining(increases(activity)) CTD celastrol RRM2 Text_Mining(decreases(expression)) CTD celastrol SELE Text_Mining(decreases(reaction)) CTD celastrol SELE Text_Mining(increases(expression)) CTD celastrol SERP1 Text_Mining(increases(expression)) CTD celastrol SESN1 Text_Mining(decreases(expression)) CTD celastrol SLC3A2 Text_Mining(increases(expression)) CTD celastrol SLC7A11 Text_Mining(decreases(response to substance)) CTD celastrol SLC7A11 Text_Mining(increases(expression)) CTD celastrol SLTM Text_Mining(decreases(expression)) CTD celastrol SOX4 Text_Mining(decreases(expression)) CTD celastrol HSPA13 Text_Mining(increases(expression)) CTD celastrol STIP1 Text_Mining(increases(expression)) CTD celastrol TAOK3 Text_Mining(decreases(expression)) CTD celastrol TMPRSS2 Text_Mining(decreases(expression)) CTD celastrol TNF Text_Mining(affects(localization)) CTD celastrol TNF Text_Mining(decreases(reaction)) CTD celastrol TNF Text_Mining(increases(activity)) CTD celastrol TNF Text_Mining(increases(expression)) CTD celastrol TNFRSF10A Text_Mining(affects(cotreatment)) CTD celastrol TNFRSF10A Text_Mining(increases(cleavage)) CTD celastrol TNFRSF10A Text_Mining(increases(reaction)) CTD celastrol TNFRSF10A Text_Mining(increases(expression)) CTD celastrol TNFRSF10A Text_Mining(increases(localization)) CTD celastrol TNFRSF10B Text_Mining(affects(cotreatment)) CTD celastrol TNFRSF10B Text_Mining(increases(cleavage)) CTD celastrol TNFRSF10B Text_Mining(increases(reaction)) CTD celastrol TNFRSF10B Text_Mining(increases(expression)) CTD celastrol TNFRSF10B Text_Mining(increases(localization)) CTD celastrol TNFSF10 Text_Mining(affects(cotreatment)) CTD celastrol TNFSF10 Text_Mining(increases(cleavage)) CTD celastrol TNFSF10 Text_Mining(increases(reaction)) CTD celastrol TNFSF10 Text_Mining(increases(response to substance)) CTD celastrol TXNIP Text_Mining(decreases(expression)) CTD celastrol TXNRD1 Text_Mining(increases(expression)) CTD celastrol UBE2B Text_Mining(increases(expression)) CTD celastrol UGDH Text_Mining(increases(expression)) CTD celastrol VCAM1 Text_Mining(decreases(reaction)) CTD celastrol VCAM1 Text_Mining(increases(expression)) CTD celastrol WDR77 Text_Mining(decreases(expression)) CTD celastrol ZBTB43 Text_Mining(decreases(expression)) CTD celastrol ZC3H12A Text_Mining(decreases(expression)) CTD celastrol HSP90AB1 Activity=None(Unspecified) D4 ChEMBL celastrol PTGER2 None=None(uM) D4 PubChem