Drug Gene Type Source AT 877 SLC12A2 Text_Mining(increases(expression)) CTD AT 877 ATAD5 Potency=10.3225(uM) D4 PubChem AT 877 ATAD5 Potency=10322.5(nM) D4 ChEMBL AT 877 CFTR None=None(uM) D4 PubChem AT 877 CFTR IC50_CF-PAF_Mean=None(uM) D4 PubChem AT 877 CYP19A1 Potency-Replicate_1=13.3332(uM) D4 PubChem AT 877 CYP19A1 None=None(uM) D4 PubChem AT 877 CYP2D6 Potency=0.1995(uM) D4 PubChem AT 877 CYP2D6 None=None(uM) D4 PubChem AT 877 CYP2D6 AC50=199.53(nM) D4 ChEMBL AT 877 CYP2D6 Potency=199.5(nM) D4 ChEMBL AT 877 CYP3A4 Potency=12.5893(uM) D4 PubChem AT 877 CYP3A4 None=None(uM) D4 PubChem AT 877 CYP3A4 AC50=12589.2(nM) D4 ChEMBL AT 877 CYP3A4 Potency=12589.3(nM) D4 ChEMBL AT 877 ESR1 Potency-Replicate_1=6.6824(uM) D4 PubChem AT 877 ESR1 ER Potency (uM)=8.41267(uM) D4 PubChem AT 877 HTT Potency=12.5893(uM) D4 PubChem AT 877 HTT Potency=12589.3(nM) D4 ChEMBL AT 877 KDM4A Potency=89125.1(nM) D4 ChEMBL AT 877 MDM2 None=None(uM) D4 PubChem AT 877 MDM4 None=None(uM) D4 PubChem AT 877 PRKACA AC50_uM=0.837(uM) D4 PubChem AT 877 PRKACA AC50_uM=1.558(uM) D4 PubChem AT 877 PRKACA AC50=1558.0(nM) D4 ChEMBL AT 877 PRKACA None=None(uM) D4 PubChem AT 877 PRKACB Inhibition=None(Unspecified) D4 ChEMBL AT 877 PRKD1 None=None(uM) D4 PubChem AT 877 PRKX Inhibition=None(Unspecified) D4 ChEMBL AT 877 ROCK2 Inhibition=None(Unspecified) D4 ChEMBL AT 877 ROCK2 None=None(uM) D4 PubChem AT 877 STK33 AC50_uM=5.98(uM) D4 PubChem AT 877 STK33 AC50_uM=9.44(uM) D4 PubChem AT 877 STK33 AC50_uM=12.6(uM) D4 PubChem AT 877 STK33 EC50_uM=9.583(uM) D4 PubChem AT 877 STK33 None=None(uM) D4 PubChem