Drug Gene Type Source lamotrigine ABCB1 Text_Mining(decreases(activity)) CTD lamotrigine CYP17A1 Text_Mining(decreases(activity)) CTD lamotrigine CYP19A1 Text_Mining(decreases(activity)) CTD lamotrigine CYP2A6 Text_Mining(decreases(reaction)) CTD lamotrigine CYP2A6 Text_Mining(increases(glutathionylation)) CTD lamotrigine CYP2A6 Text_Mining(increases(activity)) CTD lamotrigine CYP2B6 Text_Mining(increases(glutathionylation)) CTD lamotrigine CYP2D6 Text_Mining(increases(glutathionylation)) CTD lamotrigine CYP2E1 Text_Mining(increases(glutathionylation)) CTD lamotrigine CYP2E1 Text_Mining(decreases(reaction)) CTD lamotrigine CYP3A4 Text_Mining(increases(glutathionylation)) CTD lamotrigine DBH Text_Mining(increases(response to substance)) CTD lamotrigine DRD2 Text_Mining(increases(response to substance)) CTD lamotrigine HLA-B Text_Mining(affects(response to substance)) CTD lamotrigine HRH1 Text_Mining(increases(response to substance)) CTD lamotrigine HSD3B2 Text_Mining(decreases(activity)) CTD lamotrigine KCNH2 Text_Mining(decreases(activity)) CTD lamotrigine MC2R Text_Mining(increases(response to substance)) CTD lamotrigine NR3C1 Text_Mining(increases(response to substance)) CTD lamotrigine SCN2A Text_Mining(decreases(activity)) CTD lamotrigine UGT1A3 Text_Mining(increases(glucuronidation)) CTD lamotrigine UGT1A4 Text_Mining(increases(activity)) CTD lamotrigine UGT1A4 Text_Mining(increases(glucuronidation)) CTD lamotrigine AQP4 Activity=None(Unspecified) D4 ChEMBL lamotrigine CYP1A2 Inhibition=None(Unspecified) D4 ChEMBL lamotrigine CYP2C19 Inhibition=None(Unspecified) D4 ChEMBL lamotrigine CYP2C9 Inhibition=None(Unspecified) D4 ChEMBL lamotrigine CYP2D6 Potency=6.3096(uM) D4 PubChem lamotrigine CYP2D6 None=None(uM) D4 PubChem lamotrigine CYP2D6 Inhibition=None(Unspecified) D4 ChEMBL lamotrigine CYP2D6 Potency=6309.6(nM) D4 ChEMBL lamotrigine CYP2D6 AC50=6309.57(nM) D4 ChEMBL lamotrigine CYP3A4 Inhibition=None(Unspecified) D4 ChEMBL