Drug Gene Type Source Tomelukast CYSLTR1 Text_Mining(affects(binding)) CTD Tomelukast CYSLTR1 Text_Mining(increases(activity)) CTD Tomelukast CYSLTR1 Text_Mining(decreases(reaction)) CTD Tomelukast PPARA Text_Mining(affects(binding)) CTD Tomelukast PPARA Text_Mining(increases(activity)) CTD Tomelukast CYP3A4 Potency=2.5119(uM) D4 PubChem Tomelukast CYP3A4 Potency=2511.9(nM) D4 ChEMBL Tomelukast NR3C1 Potency-Replicate_1=23.9145(uM) D4 PubChem Tomelukast NR3C1 None=None(uM) D4 PubChem Tomelukast PPARG Ratio Potency (uM)=0.989298(uM) D4 PubChem Tomelukast PPARG Potency-Replicate_1=2.1872(uM) D4 PubChem Tomelukast PPARG Ratio Potency (uM)=3.33603(uM) D4 PubChem Tomelukast PPARG Potency-Replicate_1=8.7076(uM) D4 PubChem Tomelukast PPARG None=None(uM) D4 PubChem Tomelukast TDP1 Potency=21.136(uM) D4 PubChem Tomelukast TDP1 Potency=23.715(uM) D4 PubChem Tomelukast VDR Potency=44.6684(uM) D4 PubChem