Drug Gene Type Source TPEN AARS Text_Mining(decreases(expression)) CTD TPEN ABCC10 Text_Mining(decreases(expression)) CTD TPEN ABCC9 Text_Mining(increases(expression)) CTD TPEN ABL1 Text_Mining(decreases(expression)) CTD TPEN ACADL Text_Mining(decreases(expression)) CTD TPEN ACADL Text_Mining(decreases(reaction)) CTD TPEN AIFM1 Text_Mining(affects(cotreatment)) CTD TPEN AIFM1 Text_Mining(affects(localization)) CTD TPEN AIFM1 Text_Mining(decreases(reaction)) CTD TPEN AP2B1 Text_Mining(increases(expression)) CTD TPEN APC2 Text_Mining(increases(expression)) CTD TPEN APOB Text_Mining(decreases(expression)) CTD TPEN APOB Text_Mining(decreases(reaction)) CTD TPEN ARHGEF18 Text_Mining(decreases(expression)) CTD TPEN AZIN1 Text_Mining(increases(expression)) CTD TPEN BAX Text_Mining(decreases(reaction)) CTD TPEN BAX Text_Mining(increases(expression)) CTD TPEN BBC3 Text_Mining(decreases(expression)) CTD TPEN BBS9 Text_Mining(increases(expression)) CTD TPEN BCL2 Text_Mining(decreases(expression)) CTD TPEN BCL2 Text_Mining(decreases(reaction)) CTD TPEN BCL2L1 Text_Mining(decreases(expression)) CTD TPEN BCL2L1 Text_Mining(decreases(reaction)) CTD TPEN BRD1 Text_Mining(decreases(expression)) CTD TPEN BRD3 Text_Mining(decreases(expression)) CTD TPEN BRD8 Text_Mining(decreases(expression)) CTD TPEN C10ORF54 Text_Mining(increases(expression)) CTD TPEN C11ORF95 Text_Mining(decreases(expression)) CTD TPEN C1ORF50 Text_Mining(decreases(expression)) CTD TPEN CAMSAP1 Text_Mining(decreases(expression)) CTD TPEN CASP1 Text_Mining(increases(expression)) CTD TPEN CASP3 Text_Mining(affects(cotreatment)) CTD TPEN CASP3 Text_Mining(increases(activity)) CTD TPEN CASP3 Text_Mining(affects(reaction)) CTD TPEN CASP3 Text_Mining(decreases(reaction)) CTD TPEN CASP3 Text_Mining(increases(cleavage)) CTD TPEN CASP3 Text_Mining(decreases(expression)) CTD TPEN CASP3 Text_Mining(increases(expression)) CTD TPEN CASP8 Text_Mining(increases(activity)) CTD TPEN CASP9 Text_Mining(increases(activity)) CTD TPEN CCDC130 Text_Mining(decreases(expression)) CTD TPEN CCL2 Text_Mining(increases(expression)) CTD TPEN CCL22 Text_Mining(increases(expression)) CTD TPEN CCL3 Text_Mining(increases(expression)) CTD TPEN CCND1 Text_Mining(increases(expression)) CTD TPEN CCR1 Text_Mining(increases(expression)) CTD TPEN CCR2 Text_Mining(decreases(expression)) CTD TPEN CCR2 Text_Mining(increases(expression)) CTD TPEN CD14 Text_Mining(increases(expression)) CTD TPEN CD14 Text_Mining(increases(reaction)) CTD TPEN CD14 Text_Mining(affects(cotreatment)) CTD TPEN CD14 Text_Mining(decreases(reaction)) CTD TPEN CD58 Text_Mining(decreases(expression)) CTD TPEN CDH1 Text_Mining(affects(cotreatment)) CTD TPEN CDH1 Text_Mining(increases(cleavage)) CTD TPEN CDH1 Text_Mining(decreases(reaction)) CTD TPEN CEBPD Text_Mining(decreases(expression)) CTD TPEN CFP Text_Mining(increases(expression)) CTD TPEN CLCN7 Text_Mining(decreases(expression)) CTD TPEN CLCNKB Text_Mining(increases(expression)) CTD TPEN CREBBP Text_Mining(affects(binding)) CTD TPEN CREBBP Text_Mining(decreases(reaction)) CTD TPEN CRYZ Text_Mining(decreases(expression)) CTD TPEN CTDP1 Text_Mining(decreases(expression)) CTD TPEN CTDSP2 Text_Mining(decreases(expression)) CTD TPEN CTNNB1 Text_Mining(affects(cotreatment)) CTD TPEN CTNNB1 Text_Mining(increases(cleavage)) CTD TPEN CTNNB1 Text_Mining(decreases(reaction)) CTD TPEN CTSK Text_Mining(increases(expression)) CTD TPEN CX3CR1 Text_Mining(increases(expression)) CTD TPEN CXCL2 Text_Mining(increases(expression)) CTD TPEN CXCL8 Text_Mining(increases(secretion)) CTD TPEN CYTH4 Text_Mining(decreases(expression)) CTD TPEN DAD1 Text_Mining(decreases(expression)) CTD TPEN DDX23 Text_Mining(decreases(expression)) CTD TPEN DGCR14 Text_Mining(decreases(expression)) CTD TPEN DGCR2 Text_Mining(decreases(expression)) CTD TPEN DGKZ Text_Mining(decreases(expression)) CTD TPEN DHX58 Text_Mining(increases(expression)) CTD TPEN DICER1 Text_Mining(decreases(expression)) CTD TPEN DSTN Text_Mining(increases(expression)) CTD TPEN DYNC1LI2 Text_Mining(decreases(expression)) CTD TPEN EGFL7 Text_Mining(increases(expression)) CTD TPEN EGLN1 Text_Mining(increases(activity)) CTD TPEN EGLN1 Text_Mining(decreases(reaction)) CTD TPEN EHD1 Text_Mining(decreases(expression)) CTD TPEN ELF4 Text_Mining(decreases(expression)) CTD TPEN FADD Text_Mining(decreases(expression)) CTD TPEN FAM13A Text_Mining(increases(expression)) CTD TPEN FEZ1 Text_Mining(increases(expression)) CTD TPEN FOXO3 Text_Mining(decreases(expression)) CTD TPEN FRAT2 Text_Mining(decreases(expression)) CTD TPEN FZR1 Text_Mining(decreases(expression)) CTD TPEN G6PD Text_Mining(decreases(expression)) CTD TPEN GGA2 Text_Mining(decreases(expression)) CTD TPEN GMIP Text_Mining(decreases(expression)) CTD TPEN GOLPH3L Text_Mining(decreases(expression)) CTD TPEN GORASP2 Text_Mining(decreases(expression)) CTD TPEN GSTA1 Text_Mining(decreases(expression)) CTD TPEN HAX1 Text_Mining(increases(expression)) CTD TPEN HIC2 Text_Mining(decreases(expression)) CTD TPEN HIF1A Text_Mining(affects(binding)) CTD TPEN HIF1A Text_Mining(decreases(reaction)) CTD TPEN HIF1A Text_Mining(decreases(ubiquitination)) CTD TPEN HIF1A Text_Mining(increases(expression)) CTD TPEN HIF1A Text_Mining(increases(stability)) CTD TPEN HIST1H1C Text_Mining(increases(expression)) CTD TPEN HIST1H1D Text_Mining(increases(expression)) CTD TPEN HIST1H2BD Text_Mining(increases(expression)) CTD TPEN HIST1H2BE Text_Mining(increases(expression)) CTD TPEN HIST1H2BH Text_Mining(increases(expression)) CTD TPEN HIST1H2BK Text_Mining(increases(expression)) CTD TPEN HIST1H2BM Text_Mining(increases(expression)) CTD TPEN HIST1H3I Text_Mining(increases(expression)) CTD TPEN HIST1H4L Text_Mining(increases(expression)) CTD TPEN HIST2H2AA3 Text_Mining(increases(expression)) CTD TPEN HIST2H2BE Text_Mining(increases(expression)) CTD TPEN HLA-DPB1 Text_Mining(increases(expression)) CTD TPEN HLX Text_Mining(decreases(expression)) CTD TPEN HMOX2 Text_Mining(decreases(expression)) CTD TPEN HNF4A Text_Mining(decreases(activity)) CTD TPEN HNF4A Text_Mining(decreases(reaction)) CTD TPEN HNMT Text_Mining(increases(expression)) CTD TPEN IFI27 Text_Mining(increases(expression)) CTD TPEN IFI6 Text_Mining(increases(expression)) CTD TPEN IFNG Text_Mining(affects(cotreatment)) CTD TPEN IFNG Text_Mining(increases(activity)) CTD TPEN IFNG Text_Mining(increases(cleavage)) CTD TPEN IFNG Text_Mining(decreases(reaction)) CTD TPEN IFNG Text_Mining(increases(secretion)) CTD TPEN IFNGR1 Text_Mining(increases(expression)) CTD TPEN IFNGR2 Text_Mining(decreases(expression)) CTD TPEN IL10 Text_Mining(decreases(reaction)) CTD TPEN IL10 Text_Mining(decreases(secretion)) CTD TPEN IL10 Text_Mining(decreases(expression)) CTD TPEN IL10RA Text_Mining(increases(expression)) CTD TPEN IL10RB Text_Mining(increases(expression)) CTD TPEN IL13RA1 Text_Mining(increases(expression)) CTD TPEN IL1B Text_Mining(increases(expression)) CTD TPEN IL4 Text_Mining(decreases(expression)) CTD TPEN IL4R Text_Mining(decreases(expression)) CTD TPEN IL4R Text_Mining(increases(expression)) CTD TPEN IL6 Text_Mining(increases(secretion)) CTD TPEN IL6R Text_Mining(increases(expression)) CTD TPEN INTS6 Text_Mining(decreases(expression)) CTD TPEN IQGAP2 Text_Mining(increases(expression)) CTD TPEN IRF1 Text_Mining(decreases(expression)) CTD TPEN ISG15 Text_Mining(increases(expression)) CTD TPEN ITGAM Text_Mining(increases(expression)) CTD TPEN ITGAM Text_Mining(increases(reaction)) CTD TPEN ITGAM Text_Mining(affects(cotreatment)) CTD TPEN ITGAM Text_Mining(decreases(reaction)) CTD TPEN ITSN2 Text_Mining(decreases(expression)) CTD TPEN JUN Text_Mining(decreases(reaction)) CTD TPEN JUN Text_Mining(increases(activity)) CTD TPEN KAT6A Text_Mining(decreases(expression)) CTD TPEN KAZN Text_Mining(decreases(expression)) CTD TPEN KIF23 Text_Mining(decreases(expression)) CTD TPEN KRT8 Text_Mining(increases(expression)) CTD TPEN KRT8 Text_Mining(decreases(reaction)) CTD TPEN LAMP2 Text_Mining(decreases(expression)) CTD TPEN LATS2 Text_Mining(decreases(expression)) CTD TPEN LATS2 Text_Mining(decreases(reaction)) CTD TPEN LILRA5 Text_Mining(increases(expression)) CTD TPEN LTA Text_Mining(increases(expression)) CTD TPEN MAD2L1BP Text_Mining(decreases(expression)) CTD TPEN MAP2K5 Text_Mining(decreases(expression)) CTD TPEN MAPKBP1 Text_Mining(decreases(expression)) CTD TPEN MBNL2 Text_Mining(increases(expression)) CTD TPEN METTL10 Text_Mining(decreases(expression)) CTD TPEN MMP10 Text_Mining(increases(expression)) CTD TPEN MMP9 Text_Mining(affects(binding)) CTD TPEN MMP9 Text_Mining(decreases(reaction)) CTD TPEN MRPL12 Text_Mining(decreases(expression)) CTD TPEN MT1A Text_Mining(affects(cotreatment)) CTD TPEN MT1A Text_Mining(increases(expression)) CTD TPEN MT1A Text_Mining(decreases(reaction)) CTD TPEN MT1B Text_Mining(affects(cotreatment)) CTD TPEN MT1B Text_Mining(increases(expression)) CTD TPEN MT1E Text_Mining(decreases(reaction)) CTD TPEN MT1E Text_Mining(increases(expression)) CTD TPEN MT1G Text_Mining(decreases(expression)) CTD TPEN MT1H Text_Mining(decreases(expression)) CTD TPEN MT1L Text_Mining(decreases(expression)) CTD TPEN MT1X Text_Mining(decreases(reaction)) CTD TPEN MT1X Text_Mining(increases(expression)) CTD TPEN MT1X Text_Mining(decreases(expression)) CTD TPEN MT2A Text_Mining(affects(cotreatment)) CTD TPEN MT2A Text_Mining(increases(expression)) CTD TPEN MT2A Text_Mining(decreases(reaction)) CTD TPEN MTF1 Text_Mining(decreases(reaction)) CTD TPEN MTF1 Text_Mining(increases(expression)) CTD TPEN MTTP Text_Mining(decreases(expression)) CTD TPEN MTTP Text_Mining(decreases(reaction)) CTD TPEN MX2 Text_Mining(increases(expression)) CTD TPEN MYC Text_Mining(decreases(expression)) CTD TPEN MYD88 Text_Mining(increases(expression)) CTD TPEN NAB2 Text_Mining(decreases(expression)) CTD TPEN NCBP2 Text_Mining(increases(expression)) CTD TPEN NCLN Text_Mining(decreases(expression)) CTD TPEN NFKB1 Text_Mining(affects(localization)) CTD TPEN NFKB1 Text_Mining(decreases(reaction)) CTD TPEN NFKBIA Text_Mining(decreases(reaction)) CTD TPEN NFKBIA Text_Mining(increases(degradation)) CTD TPEN NFKBIA Text_Mining(decreases(expression)) CTD TPEN NKX3-2 Text_Mining(decreases(expression)) CTD TPEN NLGN1 Text_Mining(increases(expression)) CTD TPEN NLRX1 Text_Mining(decreases(expression)) CTD TPEN NSMCE4A Text_Mining(decreases(expression)) CTD TPEN NUP50 Text_Mining(increases(expression)) CTD TPEN OGT Text_Mining(decreases(expression)) CTD TPEN PARP1 Text_Mining(affects(reaction)) CTD TPEN PARP1 Text_Mining(increases(cleavage)) CTD TPEN PIK3C3 Text_Mining(decreases(expression)) CTD TPEN PLSCR1 Text_Mining(increases(expression)) CTD TPEN POLR2A Text_Mining(decreases(expression)) CTD TPEN POLR2D Text_Mining(decreases(expression)) CTD TPEN PON2 Text_Mining(decreases(expression)) CTD TPEN POU4F2 Text_Mining(increases(expression)) CTD TPEN PPARA Text_Mining(decreases(activity)) CTD TPEN PPARA Text_Mining(decreases(reaction)) CTD TPEN PPP2R2D Text_Mining(decreases(expression)) CTD TPEN PSMB2 Text_Mining(increases(expression)) CTD TPEN PTCRA Text_Mining(increases(expression)) CTD TPEN PTP4A1 Text_Mining(increases(expression)) CTD TPEN PTPRN Text_Mining(increases(expression)) CTD TPEN PUS1 Text_Mining(decreases(expression)) CTD TPEN QRICH1 Text_Mining(decreases(expression)) CTD TPEN RAD51 Text_Mining(increases(expression)) CTD TPEN RAD51C Text_Mining(increases(expression)) CTD TPEN RB1 Text_Mining(increases(expression)) CTD TPEN RB1 Text_Mining(decreases(reaction)) CTD TPEN RELA Text_Mining(decreases(activity)) CTD TPEN RELA Text_Mining(decreases(reaction)) CTD TPEN REPIN1 Text_Mining(decreases(expression)) CTD TPEN RGP1 Text_Mining(decreases(expression)) CTD TPEN RIMS2 Text_Mining(increases(expression)) CTD TPEN RNF187 Text_Mining(decreases(expression)) CTD TPEN ROR1 Text_Mining(increases(expression)) CTD TPEN RPL10 Text_Mining(decreases(expression)) CTD TPEN RPRM Text_Mining(increases(expression)) CTD TPEN RPRM Text_Mining(decreases(reaction)) CTD TPEN RPS2P45 Text_Mining(decreases(expression)) CTD TPEN RPS6KA2 Text_Mining(increases(expression)) CTD TPEN RRH Text_Mining(increases(expression)) CTD TPEN S100A12 Text_Mining(increases(expression)) CTD TPEN S100A4 Text_Mining(increases(expression)) CTD TPEN S100A6 Text_Mining(increases(expression)) CTD TPEN S100A8 Text_Mining(increases(expression)) CTD TPEN S100A9 Text_Mining(increases(expression)) CTD TPEN S100P Text_Mining(decreases(expression)) CTD TPEN SCG3 Text_Mining(increases(expression)) CTD TPEN SEC16A Text_Mining(decreases(expression)) CTD TPEN SESN1 Text_Mining(decreases(expression)) CTD TPEN SFN Text_Mining(increases(expression)) CTD TPEN SFN Text_Mining(decreases(reaction)) CTD TPEN SIDT2 Text_Mining(decreases(expression)) CTD TPEN SLC11A2 Text_Mining(increases(expression)) CTD TPEN SLC25A39 Text_Mining(decreases(expression)) CTD TPEN SLC30A1 Text_Mining(decreases(reaction)) CTD TPEN SLC30A1 Text_Mining(increases(expression)) CTD TPEN SLC30A1 Text_Mining(decreases(expression)) CTD TPEN SLC30A1 Text_Mining(increases(reaction)) CTD TPEN SLC30A1 Text_Mining(affects(cotreatment)) CTD TPEN SLC30A5 Text_Mining(affects(cotreatment)) CTD TPEN SLC30A5 Text_Mining(decreases(expression)) CTD TPEN SLC30A5 Text_Mining(increases(expression)) CTD TPEN SLC30A6 Text_Mining(affects(cotreatment)) CTD TPEN SLC30A6 Text_Mining(decreases(expression)) CTD TPEN SLC30A6 Text_Mining(increases(expression)) CTD TPEN SLC30A7 Text_Mining(affects(cotreatment)) CTD TPEN SLC30A7 Text_Mining(decreases(expression)) CTD TPEN SLC30A7 Text_Mining(increases(expression)) CTD TPEN SLC30A7 Text_Mining(increases(reaction)) CTD TPEN SLC39A1 Text_Mining(increases(expression)) CTD TPEN SLC39A10 Text_Mining(affects(cotreatment)) CTD TPEN SLC39A10 Text_Mining(decreases(expression)) CTD TPEN SLC39A14 Text_Mining(affects(cotreatment)) CTD TPEN SLC39A14 Text_Mining(decreases(expression)) CTD TPEN SLC39A2 Text_Mining(decreases(expression)) CTD TPEN SLC39A2 Text_Mining(increases(expression)) CTD TPEN SLC39A4 Text_Mining(increases(expression)) CTD TPEN SLC39A6 Text_Mining(decreases(expression)) CTD TPEN SLC39A6 Text_Mining(decreases(reaction)) CTD TPEN SLC39A6 Text_Mining(increases(cleavage)) CTD TPEN SLC39A6 Text_Mining(increases(expression)) CTD TPEN SLC39A6 Text_Mining(decreases(response to substance)) CTD TPEN SLC7A1 Text_Mining(decreases(expression)) CTD TPEN SLC9A6 Text_Mining(decreases(expression)) CTD TPEN SLCO1C1 Text_Mining(decreases(expression)) CTD TPEN SMIM7 Text_Mining(decreases(expression)) CTD TPEN SOD1 Text_Mining(increases(expression)) CTD TPEN SPEN Text_Mining(decreases(expression)) CTD TPEN SRC Text_Mining(decreases(reaction)) CTD TPEN SRC Text_Mining(increases(phosphorylation)) CTD TPEN SRSF5 Text_Mining(increases(expression)) CTD TPEN STAT1 Text_Mining(increases(expression)) CTD TPEN STAT3 Text_Mining(decreases(expression)) CTD TPEN STAT3 Text_Mining(decreases(reaction)) CTD TPEN STEAP4 Text_Mining(increases(expression)) CTD TPEN STK10 Text_Mining(decreases(expression)) CTD TPEN SYNRG Text_Mining(decreases(expression)) CTD TPEN TBC1D8 Text_Mining(decreases(expression)) CTD TPEN TGFBR2 Text_Mining(decreases(expression)) CTD TPEN THOP1 Text_Mining(decreases(expression)) CTD TPEN TIMP3 Text_Mining(increases(expression)) CTD TPEN TIMP3 Text_Mining(decreases(reaction)) CTD TPEN TLE1 Text_Mining(decreases(expression)) CTD TPEN TMEM184C Text_Mining(increases(expression)) CTD TPEN TNF Text_Mining(affects(cotreatment)) CTD TPEN TNF Text_Mining(increases(activity)) CTD TPEN TNF Text_Mining(increases(cleavage)) CTD TPEN TNF Text_Mining(increases(reaction)) CTD TPEN TNF Text_Mining(increases(secretion)) CTD TPEN TNF Text_Mining(decreases(reaction)) CTD TPEN TNFAIP8 Text_Mining(decreases(expression)) CTD TPEN TNS3 Text_Mining(decreases(expression)) CTD TPEN TP53 Text_Mining(affects(cotreatment)) CTD TPEN TP53 Text_Mining(decreases(expression)) CTD TPEN TP53 Text_Mining(decreases(reaction)) CTD TPEN TP53 Text_Mining(affects(localization)) CTD TPEN TP53 Text_Mining(increases(expression)) CTD TPEN TP73 Text_Mining(increases(expression)) CTD TPEN TP73 Text_Mining(decreases(reaction)) CTD TPEN TRAK1 Text_Mining(decreases(expression)) CTD TPEN TST Text_Mining(decreases(expression)) CTD TPEN TXNIP Text_Mining(increases(expression)) CTD TPEN TYMS Text_Mining(increases(expression)) CTD TPEN UGCG Text_Mining(decreases(expression)) CTD TPEN UNG Text_Mining(increases(expression)) CTD TPEN USP24 Text_Mining(decreases(expression)) CTD TPEN UVRAG Text_Mining(increases(expression)) CTD TPEN VEGFA Text_Mining(decreases(expression)) CTD TPEN VEGFA Text_Mining(increases(secretion)) CTD TPEN VPS33B Text_Mining(decreases(expression)) CTD TPEN WIPF2 Text_Mining(decreases(expression)) CTD TPEN YWHAZ Text_Mining(increases(expression)) CTD TPEN YWHAZ Text_Mining(decreases(reaction)) CTD TPEN ZCCHC8 Text_Mining(decreases(expression)) CTD TPEN ZFP36 Text_Mining(decreases(expression)) CTD TPEN ZFP64 Text_Mining(decreases(expression)) CTD TPEN ZNF512B Text_Mining(decreases(expression)) CTD TPEN ZNF764 Text_Mining(decreases(expression)) CTD TPEN ZNF816 Text_Mining(decreases(expression)) CTD TPEN MITF None=None(uM) D4 PubChem TPEN STK33 None=None(uM) D4 PubChem TPEN TDP1 Potency=5.6027(uM) D4 PubChem TPEN TDP1 Potency=9.9631(uM) D4 PubChem