Drug Gene Type Source GBR 12909 dihydrochloride CYP2C19 Text_Mining(decreases(activity)) CTD GBR 12909 dihydrochloride CYP2C19 Text_Mining(decreases(degradation)) CTD GBR 12909 dihydrochloride CYP2C8 Text_Mining(decreases(degradation)) CTD GBR 12909 dihydrochloride CYP2C8 Text_Mining(decreases(activity)) CTD GBR 12909 dihydrochloride CYP2E1 Text_Mining(decreases(activity)) CTD GBR 12909 dihydrochloride CYP2E1 Text_Mining(decreases(degradation)) CTD GBR 12909 dihydrochloride CYP3A4 Text_Mining(decreases(degradation)) CTD GBR 12909 dihydrochloride CYP3A4 Text_Mining(decreases(activity)) CTD GBR 12909 dihydrochloride GDNF Text_Mining(affects(cotreatment)) CTD GBR 12909 dihydrochloride GDNF Text_Mining(decreases(reaction)) CTD GBR 12909 dihydrochloride GDNF Text_Mining(increases(response to substance)) CTD GBR 12909 dihydrochloride KCNH2 Text_Mining(decreases(reaction)) CTD GBR 12909 dihydrochloride KCNH2 Text_Mining(increases(transport)) CTD GBR 12909 dihydrochloride SLC18A2 Text_Mining(affects(binding)) CTD GBR 12909 dihydrochloride SLC6A3 Text_Mining(affects(binding)) CTD GBR 12909 dihydrochloride SLC6A3 Text_Mining(decreases(reaction)) CTD GBR 12909 dihydrochloride SLC6A3 Text_Mining(increases(uptake)) CTD GBR 12909 dihydrochloride SLC6A3 Text_Mining(decreases(activity)) CTD GBR 12909 dihydrochloride SLC6A3 Text_Mining(decreases(response to substance)) CTD GBR 12909 dihydrochloride ABCB1 None=None(uM) D4 PubChem GBR 12909 dihydrochloride AR Potency-Replicate_1=15.089(uM) D4 PubChem GBR 12909 dihydrochloride AR Potency-Replicate_1=16.7855(uM) D4 PubChem GBR 12909 dihydrochloride CYP19A1 Potency-Replicate_1=18.8336(uM) D4 PubChem GBR 12909 dihydrochloride GMNN Potency=12.5893(uM) D4 PubChem GBR 12909 dihydrochloride GMNN Potency=21.136(uM) D4 PubChem GBR 12909 dihydrochloride GMNN Potency=12589.3(nM) D4 ChEMBL GBR 12909 dihydrochloride KCNH2 Potency=0.2239(uM) D4 PubChem GBR 12909 dihydrochloride MPHOSPH8 Potency=15.8489(uM) D4 PubChem GBR 12909 dihydrochloride MPHOSPH8 Potency=15848.9(nM) D4 ChEMBL GBR 12909 dihydrochloride PPARD Potency-Replicate_1=29.847(uM) D4 PubChem GBR 12909 dihydrochloride RGS4 Potency=37.6858(uM) D4 PubChem GBR 12909 dihydrochloride TDP1 Potency=0.9441(uM) D4 PubChem GBR 12909 dihydrochloride TDP1 Potency=1.0593(uM) D4 PubChem