Drug Gene Type Source nalmefene OPRK1 Text_Mining(affects(binding)) CTD nalmefene OPRK1 Text_Mining(decreases(activity)) CTD nalmefene OPRM1 Text_Mining(affects(binding)) CTD nalmefene OPRM1 Text_Mining(decreases(activity)) CTD nalmefene OPRM1 Text_Mining(increases(expression)) CTD nalmefene PRL Text_Mining(decreases(reaction)) CTD nalmefene PRL Text_Mining(increases(expression)) CTD nalmefene ESR1 Potency-Replicate_1=29.8493(uM) D4 PubChem nalmefene OPRK1 IC50=0.5(uM) D4 PubChem nalmefene OPRK1 IC50=0.779(uM) D4 PubChem nalmefene OPRK1 IC50=500.0(nM) D4 ChEMBL nalmefene OPRK1 IC50=779.0(nM) D4 ChEMBL