Drug Gene Type Source ellipticine BAX Text_Mining(increases(expression)) CTD ellipticine BCL2 Text_Mining(decreases(expression)) CTD ellipticine BID Text_Mining(decreases(expression)) CTD ellipticine BID Text_Mining(increases(cleavage)) CTD ellipticine CASP3 Text_Mining(decreases(reaction)) CTD ellipticine CASP3 Text_Mining(increases(activity)) CTD ellipticine CASP3 Text_Mining(increases(cleavage)) CTD ellipticine CASP7 Text_Mining(decreases(reaction)) CTD ellipticine CASP7 Text_Mining(increases(activity)) CTD ellipticine CASP7 Text_Mining(increases(cleavage)) CTD ellipticine CASP8 Text_Mining(increases(activity)) CTD ellipticine CASP8 Text_Mining(increases(cleavage)) CTD ellipticine CASP9 Text_Mining(increases(activity)) CTD ellipticine CASP9 Text_Mining(increases(cleavage)) CTD ellipticine CCNB1 Text_Mining(decreases(expression)) CTD ellipticine CCNB1 Text_Mining(increases(expression)) CTD ellipticine CCND1 Text_Mining(decreases(expression)) CTD ellipticine CDC25C Text_Mining(decreases(expression)) CTD ellipticine CDK1 Text_Mining(decreases(expression)) CTD ellipticine CDK1 Text_Mining(increases(phosphorylation)) CTD ellipticine CDKN1B Text_Mining(decreases(expression)) CTD ellipticine CYP1A1 Text_Mining(increases(metabolic processing)) CTD ellipticine CYP1A1 Text_Mining(decreases(reaction)) CTD ellipticine CYP1A1 Text_Mining(increases(activity)) CTD ellipticine CYP1A2 Text_Mining(increases(metabolic processing)) CTD ellipticine CYP1A2 Text_Mining(decreases(reaction)) CTD ellipticine CYP1A2 Text_Mining(increases(activity)) CTD ellipticine CYP1B1 Text_Mining(increases(metabolic processing)) CTD ellipticine CYP2C19 Text_Mining(increases(metabolic processing)) CTD ellipticine CYP2C9 Text_Mining(increases(metabolic processing)) CTD ellipticine CYP2D6 Text_Mining(increases(metabolic processing)) CTD ellipticine CYP2E1 Text_Mining(increases(metabolic processing)) CTD ellipticine CYP3A4 Text_Mining(affects(cotreatment)) CTD ellipticine CYP3A4 Text_Mining(increases(oxidation)) CTD ellipticine CYP3A4 Text_Mining(increases(metabolic processing)) CTD ellipticine MAPK1 Text_Mining(decreases(reaction)) CTD ellipticine MAPK1 Text_Mining(increases(phosphorylation)) CTD ellipticine MAPK3 Text_Mining(decreases(reaction)) CTD ellipticine MAPK3 Text_Mining(increases(phosphorylation)) CTD ellipticine MDM2 Text_Mining(decreases(response to substance)) CTD ellipticine PARP1 Text_Mining(increases(cleavage)) CTD ellipticine POR Text_Mining(affects(cotreatment)) CTD ellipticine POR Text_Mining(increases(oxidation)) CTD ellipticine TOP2B Text_Mining(decreases(response to substance)) CTD ellipticine TOP2B Text_Mining(increases(response to substance)) CTD ellipticine XIAP Text_Mining(decreases(expression)) CTD ellipticine ABCB1 None=None(uM) D4 PubChem ellipticine AHR None=None(uM) D4 PubChem ellipticine APAF1 None=None(uM) D4 PubChem ellipticine APEX1 Potency=3162.3(nM) D4 ChEMBL ellipticine APOBEC3F Potency=10.0(uM) D4 PubChem ellipticine APOBEC3G Potency=14.581(uM) D4 PubChem ellipticine APP None=None(uM) D4 PubChem ellipticine ATAD5 Potency=16.3535(uM) D4 PubChem ellipticine ATAD5 Potency=16353.5(nM) D4 ChEMBL ellipticine BAZ2B Potency=56.2341(uM) D4 PubChem ellipticine BAZ2B Potency=56234.1(nM) D4 ChEMBL ellipticine BCL2L1 None=None(uM) D4 PubChem ellipticine CACNA1H EC50_1=3.99(uM) D4 PubChem ellipticine CACNA1H None=None(uM) D4 PubChem ellipticine CACNA1H EC50=3990.0(nM) D4 ChEMBL ellipticine CBX1 Potency=50.1187(uM) D4 PubChem ellipticine CBX1 Potency=50118.7(nM) D4 ChEMBL ellipticine CFTR None=None(uM) D4 PubChem ellipticine CLK3 None=None(uM) D4 PubChem ellipticine CRHBP None=None(uM) D4 PubChem ellipticine CRHR2 None=None(uM) D4 PubChem ellipticine CYP1A2 None=None(uM) D4 PubChem ellipticine CYP1A2 AC50=19.95(nM) D4 ChEMBL ellipticine CYP2C19 Potency=3.1623(uM) D4 PubChem ellipticine CYP2C19 Potency=6.3096(uM) D4 PubChem ellipticine CYP2C19 None=None(uM) D4 PubChem ellipticine CYP2C19 Potency=3162.3(nM) D4 ChEMBL ellipticine CYP2C19 AC50=3162.28(nM) D4 ChEMBL ellipticine CYP2C19 Potency=6309.6(nM) D4 ChEMBL ellipticine CYP2D6 Potency=6.3096(uM) D4 PubChem ellipticine CYP2D6 Potency=31.6228(uM) D4 PubChem ellipticine CYP2D6 None=None(uM) D4 PubChem ellipticine CYP2D6 AC50=6309.57(nM) D4 ChEMBL ellipticine CYP2D6 Potency=31622.8(nM) D4 ChEMBL ellipticine CYP2D6 Potency=6309.6(nM) D4 ChEMBL ellipticine CYP3A4 Potency=0.1585(uM) D4 PubChem ellipticine CYP3A4 Potency=0.3981(uM) D4 PubChem ellipticine CYP3A4 None=None(uM) D4 PubChem ellipticine CYP3A4 AC50=158.49(nM) D4 ChEMBL ellipticine CYP3A4 Potency=158.5(nM) D4 ChEMBL ellipticine CYP3A4 Potency=398.1(nM) D4 ChEMBL ellipticine DRD1 Potency=10.0(uM) D4 PubChem ellipticine DRD1 None=None(uM) D4 PubChem ellipticine DRD1 Potency=10000.0(nM) D4 ChEMBL ellipticine EHMT2 Potency=21.1923(uM) D4 PubChem ellipticine EHMT2 Potency=21192.3(nM) D4 ChEMBL ellipticine FEN1 Potency=10.6213(uM) D4 PubChem ellipticine FEN1 Potency=11.9173(uM) D4 PubChem ellipticine FEN1 Potency=10621.3(nM) D4 ChEMBL ellipticine GAA Potency=35.4813(uM) D4 PubChem ellipticine GAA Potency=35481.3(nM) D4 ChEMBL ellipticine GAPDH None=None(uM) D4 PubChem ellipticine GMNN Potency=5.8048(uM) D4 PubChem ellipticine GMNN Potency=7.0795(uM) D4 PubChem ellipticine GMNN Potency=7.3078(uM) D4 PubChem ellipticine GMNN Potency=7079.5(nM) D4 ChEMBL ellipticine GNAO1 None=None(uM) D4 PubChem ellipticine GPR35 IC50=None(uM) D4 PubChem ellipticine HBB Potency=12.5893(uM) D4 PubChem ellipticine HBB Potency=31.6228(uM) D4 PubChem ellipticine HBB Potency=12589.3(nM) D4 ChEMBL ellipticine HBB Potency=31622.8(nM) D4 ChEMBL ellipticine HIF1A Potency=5.0119(uM) D4 PubChem ellipticine HIF1A Potency=5011.9(nM) D4 ChEMBL ellipticine IDH1 Potency=10.3225(uM) D4 PubChem ellipticine IL1B None=None(uM) D4 PubChem ellipticine INS None=None(uM) D4 PubChem ellipticine JAK2 None=None(uM) D4 PubChem ellipticine KCNH2 Potency=19.9526(uM) D4 PubChem ellipticine KDM4E Potency=12589.3(nM) D4 ChEMBL ellipticine MAP1LC3A None=None(uM) D4 PubChem ellipticine MAP3K3 None=None(uM) D4 PubChem ellipticine MAP3K5 None=None(uM) D4 PubChem ellipticine MAP4K2 None=None(uM) D4 PubChem ellipticine MAPT Potency=10.0(uM) D4 PubChem ellipticine MAPT Potency=11.2202(uM) D4 PubChem ellipticine MAPT Potency=10000.0(nM) D4 ChEMBL ellipticine MAPT Potency=11220.2(nM) D4 ChEMBL ellipticine MCL1 None=None(uM) D4 PubChem ellipticine MDM2 None=None(uM) D4 PubChem ellipticine MDM4 None=None(uM) D4 PubChem ellipticine MITF None=None(uM) D4 PubChem ellipticine NCF1 None=None(uM) D4 PubChem ellipticine NCOA1 None=None(uM) D4 PubChem ellipticine NFE2L2 Potency=7.3078(uM) D4 PubChem ellipticine NFE2L2 Potency=7307.8(nM) D4 ChEMBL ellipticine NLRP1 None=None(uM) D4 PubChem ellipticine NLRP3 None=None(uM) D4 PubChem ellipticine NR5A1 None=None(uM) D4 PubChem ellipticine PIM1 None=None(uM) D4 PubChem ellipticine PIM2 None=None(uM) D4 PubChem ellipticine POLB Potency=3.9811(uM) D4 PubChem ellipticine POLB Potency=15.8489(uM) D4 PubChem ellipticine POLB Potency=15848.9(nM) D4 ChEMBL ellipticine POLB Potency=3981.1(nM) D4 ChEMBL ellipticine POLI Potency=14.1254(uM) D4 PubChem ellipticine PPARG None=None(uM) D4 PubChem ellipticine PPP1CA None=None(uM) D4 PubChem ellipticine PRKACA None=None(uM) D4 PubChem ellipticine PRKD1 None=None(uM) D4 PubChem ellipticine PTBP1 Potency=31.6228(uM) D4 PubChem ellipticine PTBP1 None=None(uM) D4 PubChem ellipticine PTBP1 Potency=31622.8(nM) D4 ChEMBL ellipticine RAD54L None=None(uM) D4 PubChem ellipticine RECQL Potency=10000.0(nM) D4 ChEMBL ellipticine RECQL Potency=4466.8(nM) D4 ChEMBL ellipticine RGS4 None=None(uM) D4 PubChem ellipticine ROCK2 None=None(uM) D4 PubChem ellipticine STAT6 Potency=15.8489(uM) D4 PubChem ellipticine STAT6 Potency=15848.9(nM) D4 ChEMBL ellipticine STK33 None=None(uM) D4 PubChem ellipticine TDP1 Potency=1.4581(uM) D4 PubChem ellipticine TDP1 Potency=2.3109(uM) D4 PubChem ellipticine TDP1 Potency=50118.7(nM) D4 ChEMBL ellipticine THPO Potency=10.0(uM) D4 PubChem ellipticine THPO Potency=10000.0(nM) D4 ChEMBL ellipticine TOP2A Inhibition=None(Unspecified) D4 ChEMBL ellipticine TOP2A Activity=None(Unspecified) D4 ChEMBL ellipticine TP53 Potency=10.0(uM) D4 PubChem ellipticine TP53 Potency=12.5893(uM) D4 PubChem ellipticine TP53 Potency=10000.0(nM) D4 ChEMBL ellipticine TP53 Potency=12589.3(nM) D4 ChEMBL