Drug Gene Type Source cyclobenzaprine SLC22A2 Text_Mining(decreases(reaction)) CTD cyclobenzaprine SLC22A2 Text_Mining(increases(uptake)) CTD cyclobenzaprine CYP1A2 None=None(uM) D4 PubChem cyclobenzaprine CYP2D6 Potency=6.3096(uM) D4 PubChem cyclobenzaprine CYP2D6 None=None(uM) D4 PubChem cyclobenzaprine CYP2D6 AC50=6309.57(nM) D4 ChEMBL cyclobenzaprine CYP2D6 Potency=6309.6(nM) D4 ChEMBL cyclobenzaprine DRD1 Potency=1.0(uM) D4 PubChem cyclobenzaprine DRD1 Potency=1000.0(nM) D4 ChEMBL