Drug Gene Type Source Ici 118551 ACTA2 Text_Mining(decreases(expression)) CTD Ici 118551 ACTA2 Text_Mining(decreases(reaction)) CTD Ici 118551 ADRB1 Text_Mining(affects(binding)) CTD Ici 118551 ADRB1 Text_Mining(decreases(activity)) CTD Ici 118551 ADRB1 Text_Mining(decreases(abundance)) CTD Ici 118551 ADRB1 Text_Mining(decreases(reaction)) CTD Ici 118551 ADRB2 Text_Mining(affects(binding)) CTD Ici 118551 ADRB2 Text_Mining(decreases(abundance)) CTD Ici 118551 ADRB2 Text_Mining(decreases(activity)) CTD Ici 118551 ADRB2 Text_Mining(decreases(reaction)) CTD Ici 118551 ADRB2 Text_Mining(increases(abundance)) CTD Ici 118551 ADRB2 Text_Mining(increases(expression)) CTD Ici 118551 ADRB2 Text_Mining(increases(phosphorylation)) CTD Ici 118551 ADRB2 Text_Mining(decreases(response to substance)) CTD Ici 118551 ADRB2 Text_Mining(affects(cotreatment)) CTD Ici 118551 ADRB2 Text_Mining(increases(activity)) CTD Ici 118551 ADRB2 Text_Mining(increases(reaction)) CTD Ici 118551 ADRB3 Text_Mining(affects(binding)) CTD Ici 118551 ADRB3 Text_Mining(decreases(activity)) CTD Ici 118551 ADRB3 Text_Mining(decreases(abundance)) CTD Ici 118551 ADRB3 Text_Mining(increases(activity)) CTD Ici 118551 ADRB3 Text_Mining(decreases(reaction)) CTD Ici 118551 ADRBK1 Text_Mining(affects(cotreatment)) CTD Ici 118551 ADRBK1 Text_Mining(increases(expression)) CTD Ici 118551 ALPP Text_Mining(decreases(reaction)) CTD Ici 118551 ALPP Text_Mining(increases(expression)) CTD Ici 118551 ARRB2 Text_Mining(affects(binding)) CTD Ici 118551 ARRB2 Text_Mining(decreases(reaction)) CTD Ici 118551 ARRB2 Text_Mining(increases(reaction)) CTD Ici 118551 BAX Text_Mining(affects(cotreatment)) CTD Ici 118551 BAX Text_Mining(increases(expression)) CTD Ici 118551 BCL2 Text_Mining(affects(cotreatment)) CTD Ici 118551 BCL2 Text_Mining(decreases(expression)) CTD Ici 118551 CYP1B1 Text_Mining(decreases(reaction)) CTD Ici 118551 CYP1B1 Text_Mining(increases(expression)) CTD Ici 118551 EDN1 Text_Mining(decreases(expression)) CTD Ici 118551 EDN1 Text_Mining(decreases(reaction)) CTD Ici 118551 GNAS Text_Mining(affects(cotreatment)) CTD Ici 118551 GNAS Text_Mining(increases(expression)) CTD Ici 118551 IL5 Text_Mining(decreases(reaction)) CTD Ici 118551 IL5 Text_Mining(increases(abundance)) CTD Ici 118551 KCNH2 Text_Mining(decreases(activity)) CTD Ici 118551 KCNH2 Text_Mining(affects(binding)) CTD Ici 118551 MAPK1 Text_Mining(affects(binding)) CTD Ici 118551 MAPK1 Text_Mining(decreases(activity)) CTD Ici 118551 MAPK1 Text_Mining(decreases(reaction)) CTD Ici 118551 MAPK1 Text_Mining(increases(phosphorylation)) CTD Ici 118551 MAPK1 Text_Mining(increases(expression)) CTD Ici 118551 MAPK3 Text_Mining(affects(binding)) CTD Ici 118551 MAPK3 Text_Mining(decreases(activity)) CTD Ici 118551 MAPK3 Text_Mining(decreases(reaction)) CTD Ici 118551 MAPK3 Text_Mining(increases(phosphorylation)) CTD Ici 118551 MAPK3 Text_Mining(increases(expression)) CTD Ici 118551 MMP2 Text_Mining(decreases(expression)) CTD Ici 118551 MMP2 Text_Mining(decreases(secretion)) CTD Ici 118551 MMP9 Text_Mining(decreases(expression)) CTD Ici 118551 MMP9 Text_Mining(decreases(secretion)) CTD Ici 118551 PTGS2 Text_Mining(affects(binding)) CTD Ici 118551 PTGS2 Text_Mining(decreases(activity)) CTD Ici 118551 PTGS2 Text_Mining(decreases(reaction)) CTD Ici 118551 PTGS2 Text_Mining(increases(expression)) CTD Ici 118551 PTGS2 Text_Mining(decreases(expression)) CTD Ici 118551 RB1 Text_Mining(decreases(expression)) CTD Ici 118551 RB1 Text_Mining(decreases(reaction)) CTD Ici 118551 REN Text_Mining(decreases(reaction)) CTD Ici 118551 REN Text_Mining(increases(activity)) CTD Ici 118551 TNF Text_Mining(decreases(reaction)) CTD Ici 118551 TNF Text_Mining(increases(expression)) CTD Ici 118551 VEGFA Text_Mining(decreases(expression)) CTD Ici 118551 CYP1A2 None=None(uM) D4 PubChem Ici 118551 CYP1A2 AC50=1584.89(nM) D4 ChEMBL Ici 118551 CYP1A2 AC50=398.11(nM) D4 ChEMBL Ici 118551 CYP2D6 Potency=15.8489(uM) D4 PubChem Ici 118551 CYP2D6 None=None(uM) D4 PubChem Ici 118551 CYP2D6 AC50=15848.9(nM) D4 ChEMBL Ici 118551 CYP2D6 Potency=15848.9(nM) D4 ChEMBL Ici 118551 TDP1 Potency=3.3498(uM) D4 PubChem Ici 118551 TDP1 Potency=11.8856(uM) D4 PubChem Ici 118551 TSHR Potency=39.8107(uM) D4 PubChem Ici 118551 TSHR Potency=39810.7(nM) D4 ChEMBL