Drug Gene Type Source CL 218872 GABRA1 Text_Mining(affects(binding)) CTD CL 218872 GABRA1 Text_Mining(increases(activity)) CTD CL 218872 GABRB3 Text_Mining(affects(binding)) CTD CL 218872 GABRB3 Text_Mining(increases(activity)) CTD CL 218872 GABRG2 Text_Mining(affects(binding)) CTD CL 218872 GABRG2 Text_Mining(increases(activity)) CTD CL 218872 CYP1A2 None=None(uM) D4 PubChem CL 218872 CYP1A2 AC50=79.43(nM) D4 ChEMBL CL 218872 HSD17B10 Potency=19952.6(nM) D4 ChEMBL CL 218872 ITGA4 None=None(uM) D4 PubChem