Drug Gene Type Source Fulvestrant ESR1 Text_Mining(PMID21729658,PMID22286314,PMID22795960,PMID24335365,PMID21847409,PMID21075433,PMID20494961,PMID20926342,PMID23881388,PMID21319872,PMID20151846,PMID23500091,PMID21839641,PMID21477578,PMID21699443,PMID21378333,PMID22616615,PMID23278394,PMID23798616,PMID22050013,PMID21906312,PMID24505287,PMID21533195,PMID19966214,PMID20164664,PMID22982765,PMID23179494,PMID22119979,PMID22826433,PMID21566246,PMID21464335,PMID22646768,PMID21816233,PMID23299092,PMID20739074,PMID21473877,PMID20579400,PMID20807822,PMID20306159,PMID22999294,PMID23764179,PMID21480391,PMID23399957,PMID25028367,PMID20305694,PMID20393009,PMID23936773,PMID21345137,PMID22759564,PMID20842631,PMID24589524,PMID23936234,PMID20332324,PMID22521773,PMID23714446,PMID24227889,PMID22319644,PMID21856997,PMID23592396,PMID20061804,PMID20512796,PMID20669046,PMID21642474,PMID23649836,PMID21916582,PMID22961055,PMID21966546,PMID22319200,PMID21362200,PMID21726350,PMID20596666,PMID21144907,PMID20876285,PMID20034504,PMID20700755,PMID23609470,PMID23569364,PMID23077249,PMID22859269,PMID22538444,PMID22234368,PMID23857583,PMID23462505,PMID24448819,PMID23526212,PMID22869106,PMID24874954,PMID23236424,PMID23523357,PMID21292820,PMID22427208,PMID24407733,PMID20981412,PMID19609946,PMID23801303,PMID23845572,PMID23087146,PMID23911795,PMID21057537,PMID24643679,PMID23419388,PMID23615023,PMID21170268,PMID22535971,PMID22418699,PMID24747123,PMID20215421,PMID23466753,PMID23593342,PMID22015101,PMID23085002,PMID22041887,PMID21595894,PMID21792889,PMID20654613,PMID21792626,PMID22560634,PMID22383111,PMID22896656,PMID21863258,PMID21339261,PMID22276069,PMID24440569,PMID24724101,PMID23626803,PMID24819550,PMID20160663,PMID19931544,PMID20549698,PMID22123186,PMID23033157,PMID21205741,PMID22049316,PMID21737572,PMID21284537,PMID24916694,PMID21801281,PMID21908557,PMID23649927,PMID22056872,PMID23052036,PMID23605692,PMID21299862,PMID21127968,PMID23362266,PMID24379833,PMID24758408,PMID23216744,PMID24298433,PMID23844554,PMID20164203,PMID24037977) BOSS Fulvestrant EREG Text_Mining(PMID20938664,PMID22549111,PMID24505287,PMID20104523,PMID20104523,PMID22826433,PMID20103631,PMID24374015,PMID24374015,PMID24007820,PMID20156170,PMID21276249,PMID20208560,PMID20208560,PMID20061804,PMID22319200,PMID20596666,PMID20034504,PMID20034504,PMID22840697,PMID22396492,PMID22892083,PMID24723976,PMID24874954,PMID21224239,PMID20405008,PMID23911795,PMID20874728,PMID20375134,PMID21248290,PMID24785473,PMID24457069,PMID19697122,PMID19697122,PMID20215511,PMID20215511,PMID20215511,PMID19626437,PMID19626437,PMID19815064,PMID20215421,PMID20826728,PMID21396094,PMID20068169,PMID20068169,PMID22173127,PMID22173127,PMID22613849,PMID22613849,PMID21246834,PMID24782439,PMID24782439,PMID23686416,PMID23772748,PMID24169358,PMID23758675) BOSS Fulvestrant EGFR Text_Mining(PMID23881388,PMID22317766,PMID21639949,PMID24924416,PMID23399957,PMID20332324,PMID24335372,PMID21642474,PMID21966546,PMID23609470,PMID22418699,PMID24268810,PMID19697122,PMID21396094,PMID21595894,PMID21792626,PMID22560634,PMID22560634,PMID21339261,PMID24819550,PMID24819550,PMID20549698,PMID19238537,PMID24394127,PMID23686416,PMID22258476,PMID24379833,PMID24758408,PMID24758408) BOSS Fulvestrant PGR Text_Mining(PMID22286314,PMID21075433,PMID23881388,PMID23500091,PMID21473877,PMID21276249,PMID23592396,PMID21642474,PMID22961055,PMID22396492,PMID22892083,PMID23845572,PMID21248290,PMID21248290,PMID22669982,PMID23902874,PMID21339261,PMID24724101,PMID23605692) BOSS Fulvestrant ERBB2 Text_Mining(PMID19875750,PMID20306159,PMID24513268,PMID21966546,PMID20876285,PMID22840697,PMID21922395,PMID23845572,PMID24554387,PMID21863258,PMID22276069,PMID24724101,PMID20549698,PMID22123186,PMID19238537,PMID24394127,PMID23686416) BOSS Fulvestrant DDR2 Text_Mining(PMID24924416,PMID24513268,PMID21642474,PMID23857583,PMID24448819,PMID24448819,PMID19815064,PMID23593342,PMID23593342,PMID23593342,PMID21792889,PMID21792889,PMID22560634,PMID22258476,PMID23758675,PMID23844554) BOSS Fulvestrant BCL2 Text_Mining(PMID20305694,PMID21172805,PMID20876285,PMID23609470,PMID22961366,PMID20457620,PMID22015101,PMID20654613,PMID20062536,PMID22162424,PMID19931544,PMID22123186,PMID21801281,PMID21127968) BOSS Fulvestrant ERBB2 Text_Mining(PMID19875750,PMID23390495,PMID23443928,PMID20332324,PMID20876285,PMID21922395,PMID19697122,PMID21396094,PMID21595894,PMID21339261,PMID24724101,PMID22123186,PMID21299862,PMID24169358) BOSS Fulvestrant AKR1B1 Text_Mining(PMID20164664,PMID22017761,PMID22234368,PMID22535971,PMID22535971,PMID22613849,PMID24916694,PMID24782439,PMID24782439,PMID23052036,PMID23686416) BOSS Fulvestrant ESR2 Text_Mining(PMID20061804,PMID20034504,PMID20034504,PMID20405008,PMID20874728,PMID21248290,PMID20826728,PMID20433925,PMID20433925,PMID22162424,PMID21246834) BOSS Fulvestrant MERTK Text_Mining(PMID24793639,PMID20034504,PMID20034504,PMID20651347,PMID20826728,PMID24440569,PMID24782439,PMID24379833,PMID24379833,PMID24169358) BOSS Fulvestrant TP53 Text_Mining(PMID22549111,PMID23077249,PMID24747123,PMID22041887,PMID20549698,PMID20549698,PMID19238537,PMID24916694,PMID23216744) BOSS Fulvestrant IGFBP1 Text_Mining(PMID21464335,PMID22444722,PMID23649836,PMID23649836,PMID22427208,PMID22427208,PMID21595894,PMID21908557,PMID23844554) BOSS Fulvestrant VEGFA Text_Mining(PMID22548798,PMID24924416,PMID23088607,PMID23801303,PMID22015101,PMID22162424,PMID22258476,PMID22258476) BOSS Fulvestrant PRL Text_Mining(PMID21464335,PMID22017761,PMID21276249,PMID20700755,PMID23523357,PMID24407733,PMID24643679,PMID22015101) BOSS Fulvestrant EGF Text_Mining(PMID22646768,PMID23609470,PMID23153318,PMID22560634,PMID20068169,PMID23605692,PMID23686416,PMID24758408) BOSS Fulvestrant ERBB3 Text_Mining(PMID21639949,PMID23999432,PMID23609470,PMID21396094,PMID24819550,PMID22123186,PMID23686416) BOSS Fulvestrant NR4A1 Text_Mining(PMID23542955,PMID23443928,PMID20306159,PMID25028579,PMID20156170,PMID23153318,PMID22418699) BOSS Fulvestrant MAPK3 Text_Mining(PMID20874728,PMID22673740,PMID24440569,PMID23686416,PMID23772748,PMID24758408,PMID23216744) BOSS Fulvestrant TSC1 Text_Mining(PMID24837491,PMID23159849,PMID22538444,PMID24643679,PMID20457620,PMID22383111,PMID20549698) BOSS Fulvestrant MTOR Text_Mining(PMID23299092,PMID23714446,PMID21362200,PMID21339261,PMID22149876,PMID23605692) BOSS Fulvestrant EPHB2 Text_Mining(PMID23466753,PMID22383111,PMID23686416,PMID23772748,PMID23362266,PMID24379833) BOSS Fulvestrant CDT1 Text_Mining(PMID24462822,PMID24747123,PMID21801281,PMID23064032,PMID23064032,PMID24298433) BOSS Fulvestrant ABCA1 Text_Mining(PMID21966546,PMID23247057,PMID20874728,PMID21595894,PMID21792889) BOSS Fulvestrant MYC Text_Mining(PMID22396492,PMID22892083,PMID20525379,PMID22896656,PMID21863258) BOSS Fulvestrant PCNA Text_Mining(PMID20525379,PMID22383111,PMID22896656,PMID21284537,PMID20145171,PMID) BOSS Fulvestrant AR Ratio Potency (uM)=7.18374(uM) D4 PubChem Fulvestrant CYP19A1 Potency-Replicate_1=0.0153(uM) D4 PubChem Fulvestrant CYP19A1 Potency-Replicate_1=0.0596(uM) D4 PubChem Fulvestrant CYP19A1 None=None(uM) D4 PubChem Fulvestrant EPHX2 Inhibition=None(Unspecified) D4 ChEMBL Fulvestrant ESR1 ER Potency (uM)=0.00685199(uM) D4 PubChem Fulvestrant ESR1 Potency-Replicate_1=0.0086(uM) D4 PubChem Fulvestrant ESR1 ER Potency (uM)=0.0219584(uM) D4 PubChem Fulvestrant ESR1 Ratio Potency (uM)=0.0254889(uM) D4 PubChem Fulvestrant ESR1 Potency-Replicate_1=0.0298(uM) D4 PubChem Fulvestrant ESR1 Ratio Potency (uM)=0.111001(uM) D4 PubChem Fulvestrant ESR1 Potency-Replicate_1=0.6007(uM) D4 PubChem Fulvestrant ESR1 Potency-Replicate_1=3.4648(uM) D4 PubChem Fulvestrant ESR1 Activity=None(Unspecified) D4 ChEMBL Fulvestrant ESR2 Activity=None(Unspecified) D4 ChEMBL Fulvestrant ESRRA Activity=None(Unspecified) D4 ChEMBL Fulvestrant NFE2L2 Ratio Potency (uM)=17.2114(uM) D4 PubChem Fulvestrant NR1H4 None=None(uM) D4 PubChem Fulvestrant NR3C1 Potency-Replicate_1=1.2294(uM) D4 PubChem Fulvestrant NR3C1 None=None(uM) D4 PubChem