Drug Gene Type Source rotenone ATP8A2 Text_Mining(PMID22697124,PMID21268709,PMID20209153,PMID22510598,PMID21033441,PMID22930474,PMID19695309,PMID20151456,PMID21415535,PMID22814253,PMID21814580,PMID20484937,PMID23802648,PMID20374433,PMID20443048,PMID19693701,PMID21958946,PMID21643997,PMID24228605,PMID23769741,PMID23281261,PMID23971408,PMID23245650,PMID24349535,PMID23259041,PMID23874855,PMID21445095,PMID24596095,PMID20224768,PMID19995567,PMID20005986,PMID20207656,PMID23911619,PMID24570045,PMID20971059,PMID22123175,PMID22606219,PMID19923925,PMID21484098,PMID20883473,PMID24122005,PMID20942856,PMID24002177,PMID21780161,PMID21875114,PMID22865232,PMID20962050,PMID21514419,PMID24150756,PMID23605682,PMID24434522,PMID24508187,PMID21339825,PMID19781600,PMID22414808,PMID22214982,PMID21889400,PMID22288477,PMID21542899,PMID20445170,PMID20035277,PMID20107899,PMID20349346,PMID21659507,PMID22086148,PMID23912160,PMID24948319,PMID24948273,PMID23010494,PMID20632939,PMID21350246,PMID22906069,PMID23499835,PMID20937116,PMID24205431,PMID20655985,PMID21398508,PMID23738008,PMID21159641,PMID24558474,PMID24493626,PMID21352099,PMID23508964,PMID22801494,PMID24948305) BOSS rotenone CASP3 Text_Mining(PMID23189969,PMID23098804,PMID22846965,PMID21799745,PMID22985856,PMID24315037,PMID24122264,PMID22942730,PMID24228605,PMID22974977,PMID24337984,PMID21723922,PMID22970265,PMID21899552,PMID21216964,PMID21091473,PMID24440618,PMID21044082,PMID20811676,PMID24830863,PMID24852355,PMID20962050,PMID21963892,PMID24549762,PMID19857556,PMID24330357,PMID23605682,PMID21061154,PMID23963993,PMID23900721,PMID20056314,PMID19781773,PMID22350517,PMID22210314,PMID22710069,PMID19874289,PMID22659498,PMID22401854,PMID22483284,PMID20417273,PMID24948319,PMID24948319,PMID20226830,PMID22002081,PMID22623043,PMID20875851,PMID19850127,PMID22526376,PMID24949116,PMID23291720,PMID24882730,PMID22264378,PMID24382325,PMID24142350,PMID24142350,PMID23508964,PMID23725013,PMID23997112) BOSS rotenone NDUFA5 Text_Mining(PMID21893155,PMID22158713,PMID22387164,PMID22387164,PMID22484275,PMID20300811,PMID22324553,PMID21484267,PMID23957165,PMID23816754,PMID24497186,PMID24104397,PMID21890492,PMID23238793,PMID24596095,PMID20207656,PMID20074573,PMID23118969,PMID22945465,PMID20117074,PMID20628600,PMID21749117,PMID22854968,PMID24355434,PMID21827296,PMID22239987,PMID21864496,PMID22190282,PMID23669099,PMID24365956,PMID21454572,PMID21339825,PMID21212096,PMID21505151,PMID22214982,PMID21424245,PMID23548633,PMID22430089,PMID22661471,PMID21659507,PMID22305999,PMID22086148,PMID20226830,PMID24560713,PMID22750028,PMID21398508,PMID23671162,PMID23010495,PMID21352099,PMID20724705) BOSS rotenone GCH1 Text_Mining(PMID21212524,PMID20169778,PMID23098804,PMID21798348,PMID22521663,PMID21277943,PMID23281940,PMID24006664,PMID20807515,PMID22316420,PMID23819239,PMID23073839,PMID21742033,PMID19644772,PMID22985856,PMID21953489,PMID22483308,PMID23639798,PMID23714208,PMID22942730,PMID24195216,PMID24613722,PMID23441691,PMID22895566,PMID21899552,PMID22342763,PMID25069193,PMID20374418,PMID20823569,PMID19626387,PMID22546249,PMID24175569,PMID21061154,PMID23446007,PMID23121049,PMID24381808,PMID22710069,PMID23159314,PMID20854799,PMID24070629,PMID24296154,PMID23353925,PMID22483311) BOSS rotenone DECR1 Text_Mining(PMID23722112,PMID24374334,PMID23148249,PMID21295135,PMID23241345,PMID20041858,PMID22094225,PMID22252868,PMID22945465,PMID21248133,PMID20722506,PMID23349115,PMID24226522,PMID23956071,PMID20231142,PMID21368743,PMID21524703,PMID21505151,PMID21792922,PMID22387155,PMID22549734,PMID23524287,PMID22430089,PMID22442197,PMID23958265,PMID22002081,PMID21138635,PMID20444986,PMID20736017,PMID24191234,PMID21798540,PMID24188932,PMID23232926,PMID21597236,PMID24053613,PMID22946344,PMID24355174,PMID21575165,PMID23349663,PMID20727219) BOSS rotenone ROS1 Text_Mining(PMID21238542,PMID22301167,PMID22510598,PMID22160863,PMID22387164,PMID22985602,PMID20300811,PMID23328116,PMID20117172,PMID22616995,PMID22895566,PMID22521218,PMID22366220,PMID23914057,PMID21190861,PMID20018182,PMID24002177,PMID24959670,PMID24226522,PMID24027419,PMID24736663,PMID23900721,PMID21524703,PMID23643711,PMID19874289,PMID24948319,PMID23010494,PMID20875851,PMID23499835,PMID23619395,PMID23738008,PMID24142350,PMID24755484,PMID22683349) BOSS rotenone MRPL23 Text_Mining(PMID21067569,PMID21419806,PMID20596942,PMID21085094,PMID20098733,PMID18639366,PMID23281940,PMID21799745,PMID22392151,PMID24618574,PMID24195216,PMID23623990,PMID20117172,PMID22056602,PMID22536024,PMID21091473,PMID24440618,PMID20464527,PMID20374418,PMID19681169,PMID21152247,PMID19626387,PMID24002177,PMID24175569,PMID23244436,PMID23984410,PMID19857556,PMID22198804,PMID19850127,PMID24407237,PMID22483311) BOSS rotenone BCL2 Text_Mining(PMID21664962,PMID22985856,PMID24228605,PMID23769741,PMID21723922,PMID21807080,PMID21899552,PMID22300030,PMID24625983,PMID19777565,PMID24214023,PMID24549762,PMID21061154,PMID23963993,PMID23900721,PMID22560595,PMID22288477,PMID22210314,PMID22483284,PMID22623043,PMID24205431,PMID24882730,PMID22264378,PMID24382325,PMID24755484,PMID23251750,PMID21403387) BOSS rotenone CYCS Text_Mining(PMID23189969,PMID22936601,PMID21799745,PMID21484267,PMID22942730,PMID22464971,PMID22015496,PMID23077897,PMID21216964,PMID25089873,PMID21044082,PMID22239987,PMID24214023,PMID23952718,PMID21454572,PMID23900721,PMID22661471,PMID20663895,PMID24205431,PMID23619395,PMID24382325,PMID23725013,PMID22946344) BOSS rotenone SLC7A1 Text_Mining(PMID23227042,PMID23639798,PMID22378894,PMID21445095,PMID24780191,PMID24175569,PMID23963993,PMID23643711,PMID22210314,PMID22064362,PMID20417273,PMID23994302,PMID20226830,PMID20688078,PMID24205431,PMID23738008,PMID24493626,PMID21199725,PMID23205777,PMID23353925,PMID21575165) BOSS rotenone CASP9 Text_Mining(PMID22974977,PMID21216964,PMID20018182,PMID25089873,PMID20811676,PMID24830863,PMID24852355,PMID20962050,PMID24214023,PMID24549762,PMID23605682,PMID21061154,PMID22710069,PMID22401854,PMID20226830,PMID19850127,PMID23291720,PMID23725013) BOSS rotenone TP53 Text_Mining(PMID21893155,PMID22289634,PMID22289634,PMID21223980,PMID21223980,PMID23899557,PMID23899557,PMID23714208,PMID21780161,PMID23774475,PMID23963993,PMID19874289,PMID22905163,PMID24949116,PMID24382325,PMID23664925) BOSS rotenone WDTC1 Text_Mining(PMID21033441,PMID22037189,PMID23957165,PMID20443048,PMID23077897,PMID22192354,PMID21059655,PMID21542899,PMID20035277,PMID23912160,PMID20632939,PMID22906069,PMID20937116,PMID21159641,PMID21352099,PMID24948305) BOSS rotenone LDHA Text_Mining(PMID20169778,PMID20634262,PMID21081703,PMID21356207,PMID21899552,PMID20026743,PMID24998649,PMID22560595,PMID23121049,PMID21542899,PMID20445170,PMID20417273,PMID20656495,PMID20226830,PMID20536682) BOSS rotenone PARK7 Text_Mining(PMID20940149,PMID23065353,PMID21907265,PMID21907265,PMID21455296,PMID22898350,PMID20464527,PMID21219333,PMID20823569,PMID22710069,PMID24949116,PMID24158912,PMID24070629) BOSS rotenone MAPK3 Text_Mining(PMID24641423,PMID24226522,PMID20056314,PMID20231142,PMID23579275,PMID22264378,PMID22778212,PMID23738008,PMID24755484,PMID21300668,PMID22946344,PMID23349663) BOSS rotenone INS Text_Mining(PMID21401303,PMID20022987,PMID19781600,PMID21505151,PMID23643711,PMID22210314,PMID23524287,PMID23958265,PMID21350246,PMID23499835) BOSS rotenone HSD17B6 Text_Mining(PMID22158713,PMID23722112,PMID23874855,PMID20074573,PMID20117074,PMID20628600,PMID21339825,PMID21505151,PMID23354121,PMID23912160) BOSS rotenone ABCA1 Text_Mining(PMID20418776,PMID20418776,PMID23916614,PMID22366220,PMID20056314,PMID19900598,PMID20162567,PMID21077940,PMID22350517,PMID22087877) BOSS rotenone SLC25A20 Text_Mining(PMID23770533,PMID19889626,PMID22863937,PMID20374433,PMID24108391,PMID24122005,PMID22586224,PMID23291720,PMID21403387) BOSS rotenone EPHB2 Text_Mining(PMID23916614,PMID22898350,PMID19900598,PMID22560595,PMID23579275,PMID22659498,PMID23232926,PMID23251750,PMID21403387) BOSS rotenone MPP6 Text_Mining(PMID24351065,PMID23238634,PMID22265821,PMID23121049,PMID20854799,PMID23319378,PMID21352099,PMID24341912,PMID23997112) BOSS rotenone ACHE Text_Mining(PMID23868340,PMID23676090,PMID24831121,PMID21715067,PMID22521218,PMID23092410,PMID20656495,PMID20575555,PMID20536682) BOSS rotenone HMOX1 Text_Mining(PMID21219333,PMID24451142,PMID24451142,PMID22864061,PMID20875851,PMID20875851,PMID20536682,PMID22683349,PMID22683349) BOSS rotenone RHO Text_Mining(PMID21388687,PMID24473093,PMID21742033,PMID23593279,PMID20628600,PMID24150756,PMID23028832,PMID22661471) BOSS rotenone SOD1 Text_Mining(PMID24167416,PMID21484267,PMID22447502,PMID22579008,PMID24141050,PMID23619395,PMID24188932,PMID21368742) BOSS rotenone SETD2 Text_Mining(PMID20637638,PMID23916614,PMID20546814,PMID21875114,PMID24858344,PMID24188932,PMID24586439,PMID22087877) BOSS rotenone IL6 Text_Mining(PMID22261544,PMID22330755,PMID20701773,PMID24830863,PMID22932892,PMID22932892,PMID23159314,PMID22685265) BOSS rotenone GPX1 Text_Mining(PMID21748272,PMID23148249,PMID25069193,PMID24175569,PMID21884756,PMID24205431,PMID23660306,PMID22946344) BOSS rotenone TRAPPC9 Text_Mining(PMID22807129,PMID22807129,PMID22807129,PMID23899557,PMID22616995,PMID20107899,PMID22483311) BOSS rotenone BDNF-AS Text_Mining(PMID24780767,PMID21061154,PMID22560595,PMID22288477,PMID22288477,PMID20854799,PMID20854799) BOSS rotenone PPARG Text_Mining(PMID19693701,PMID20064719,PMID22928487,PMID21875114,PMID24374061,PMID20162567,PMID22745725) BOSS rotenone PLAU Text_Mining(PMID23703371,PMID23073839,PMID23238634,PMID24418467,PMID24418467,PMID21061154,PMID22288477) BOSS rotenone AGT Text_Mining(PMID23788763,PMID23774475,PMID20231142,PMID20444986,PMID24191234,PMID24053613,PMID23349663) BOSS rotenone CYBB Text_Mining(PMID23050834,PMID23349115,PMID22549734,PMID22685265,PMID24053613,PMID24053613,PMID23349663) BOSS rotenone POLD4 Text_Mining(PMID19777565,PMID23977201,PMID24214023,PMID24226522,PMID19900598,PMID22659498,PMID21199725) BOSS rotenone PRRT2 Text_Mining(PMID22414808,PMID21792922,PMID23900672,PMID22087877,PMID20536682,PMID24053613,PMID22683349) BOSS rotenone CDT1 Text_Mining(PMID24747077,PMID24747077,PMID23198691,PMID20645919,PMID20645919,PMID20645919,PMID20645919) BOSS rotenone MPO Text_Mining(PMID21704008,PMID23593274,PMID23056359,PMID23650208,PMID20655985,PMID24273204) BOSS rotenone ALOX5 Text_Mining(PMID21488210,PMID21488210,PMID24858057,PMID24858057,PMID24998649,PMID24998649) BOSS rotenone EDN1 Text_Mining(PMID22928487,PMID20231142,PMID20444986,PMID20444986,PMID21575165,PMID21575165) BOSS rotenone SPARC Text_Mining(PMID21723922,PMID22385295,PMID24122005,PMID24508187,PMID23508964,PMID24341912) BOSS rotenone AATF Text_Mining(PMID23868340,PMID23676090,PMID21715067,PMID20656495,PMID20656495,PMID20575555) BOSS rotenone SLC6A3 Text_Mining(PMID22342763,PMID24749734,PMID19681169,PMID23710172,PMID24381808,PMID22659498) BOSS rotenone GJA1 Text_Mining(PMID23456878,PMID23456878,PMID23783886,PMID23783886,PMID20824494,PMID20824494) BOSS rotenone SLC26A1 Text_Mining(PMID24552419,PMID22268123,PMID22268123,PMID23874855,PMID21505151,PMID22086148) BOSS rotenone ISYNA1 Text_Mining(PMID24315037,PMID22928487,PMID22252868,PMID23159314,PMID23353925,PMID23353925) BOSS rotenone PINK1 Text_Mining(PMID20940149,PMID24967965,PMID22536024,PMID22319455,PMID24374061,PMID24158912) BOSS rotenone STAT3 Text_Mining(PMID20224768,PMID19781773,PMID22932892,PMID22847181,PMID23251750,PMID21403387) BOSS rotenone DHFR Text_Mining(PMID24135141,PMID22192354,PMID22549734,PMID21059655,PMID22064362) BOSS rotenone ROCK1 Text_Mining(PMID23670202,PMID23130145,PMID24948271,PMID20360439,PMID23738008) BOSS rotenone XDH Text_Mining(PMID25069193,PMID21570952,PMID22141451,PMID21597236,PMID20727219) BOSS rotenone TNF Text_Mining(PMID23939409,PMID20041858,PMID20026743,PMID23645222,PMID22685265) BOSS rotenone MEOX2 Text_Mining(PMID21295135,PMID20722506,PMID22549734,PMID22685265,PMID24053613) BOSS rotenone VEGFA Text_Mining(PMID23922721,PMID23788766,PMID20811676,PMID22745725,PMID22483311) BOSS rotenone REEP5 Text_Mining(PMID21699019,PMID22945465,PMID22387155,PMID20226830,PMID20688078) BOSS rotenone IDE Text_Mining(PMID21472727,PMID22659498,PMID21159641,PMID21159641,PMID22683349) BOSS rotenone JAK2 Text_Mining(PMID20224768,PMID22932892,PMID20875851,PMID23251750,PMID21403387) BOSS rotenone LRRK2 Text_Mining(PMID23055790,PMID22536024,PMID24158912,PMID24407237,PMID22483311) BOSS rotenone HSPA4 Text_Mining(PMID20705047,PMID22447502,PMID22710069,PMID23900672,PMID24296154,PMID) BOSS rotenone ABCB1 None=None(uM) D4 PubChem rotenone AR Potency-Replicate_1=0.0097(uM) D4 PubChem rotenone AR Potency-Replicate_1=0.0247(uM) D4 PubChem rotenone AR Potency-Replicate_1=0.1883(uM) D4 PubChem rotenone AR Potency-Replicate_1=0.2791(uM) D4 PubChem rotenone AR Potency-Replicate_1=0.7562(uM) D4 PubChem rotenone CBX1 Potency=35.4813(uM) D4 PubChem rotenone CBX1 Potency=35481.3(nM) D4 ChEMBL rotenone CDK1 Activity=None(Unspecified) D4 ChEMBL rotenone CFL1 Activity=None(Unspecified) D4 ChEMBL rotenone CYP19A1 Potency-Replicate_1=14.9601(uM) D4 PubChem rotenone CYP19A1 Potency-Replicate_1=34.3762(uM) D4 PubChem rotenone CYP19A1 Potency-Replicate_1=34.8312(uM) D4 PubChem rotenone CYP1A2 None=None(uM) D4 PubChem rotenone CYP2C19 Potency=1.0(uM) D4 PubChem rotenone CYP2C19 Potency=1000.0(nM) D4 ChEMBL rotenone CYP3A4 Potency=15.8489(uM) D4 PubChem rotenone CYP3A4 Potency=15848.9(nM) D4 ChEMBL rotenone ESR1 Potency-Replicate_1=0.0154(uM) D4 PubChem rotenone ESR1 ER Potency (uM)=0.0306379(uM) D4 PubChem rotenone ESR1 ER Potency (uM)=0.0310433(uM) D4 PubChem rotenone ESR1 Potency-Replicate_1=0.0391(uM) D4 PubChem rotenone ESR1 ER Potency (uM)=0.143968(uM) D4 PubChem rotenone ESR1 Potency-Replicate_1=0.1496(uM) D4 PubChem rotenone ESR1 Ratio Potency (uM)=40.4169(uM) D4 PubChem rotenone ESR1 Potency-Replicate_1=48.9662(uM) D4 PubChem rotenone GLS Potency=11.2202(uM) D4 PubChem rotenone GMNN Potency=0.7546(uM) D4 PubChem rotenone GMNN Potency=0.92(uM) D4 PubChem rotenone GMNN Potency=1.0659(uM) D4 PubChem rotenone GMNN Potency=1.4125(uM) D4 PubChem rotenone GMNN Potency=3.9327(uM) D4 PubChem rotenone GMNN Potency=1412.5(nM) D4 ChEMBL rotenone GMNN Potency=1065.9(nM) D4 ChEMBL rotenone GMNN Potency=754.6(nM) D4 ChEMBL rotenone GMNN Potency=920.0(nM) D4 ChEMBL rotenone JUN Activity=None(Unspecified) D4 ChEMBL rotenone MTOR Potency=0.0465(uM) D4 PubChem rotenone MTOR Potency=0.0585(uM) D4 PubChem rotenone MTOR Potency=58.5(nM) D4 ChEMBL rotenone MTOR Inhibition=None(Unspecified) D4 ChEMBL rotenone MTOR Activity=None(Unspecified) D4 ChEMBL rotenone MTOR Potency=46.5(nM) D4 ChEMBL rotenone NFE2L2 Potency-Replicate_1=0.0077(uM) D4 PubChem rotenone NFE2L2 Ratio Potency (uM)=0.017903(uM) D4 PubChem rotenone NFE2L2 Ratio Potency (uM)=0.0203533(uM) D4 PubChem rotenone NFE2L2 Ratio Potency (uM)=0.0455233(uM) D4 PubChem rotenone NR1H4 Potency-Replicate_1=0.7497(uM) D4 PubChem rotenone NR1H4 None=None(uM) D4 PubChem rotenone PPARD Potency-Replicate_1=4.8966(uM) D4 PubChem rotenone PPARG Potency-Replicate_1=13.3322(uM) D4 PubChem rotenone PPARG Potency=44.6684(uM) D4 PubChem rotenone PPARG None=None(uM) D4 PubChem rotenone RXRA Potency=19.9526(uM) D4 PubChem rotenone TDP1 Potency=0.1496(uM) D4 PubChem rotenone TDP1 Potency=0.1884(uM) D4 PubChem rotenone TDP1 Potency=0.2371(uM) D4 PubChem rotenone TP53 Activity=None(Unspecified) D4 ChEMBL