Drug Gene Type Source trifluoperazine KRIT1 Text_Mining(PMID24316213,PMID20392081,PMID21656570,PMID20544963,PMID22331049,PMID21787279,PMID22242837,PMID20939762,PMID21554771,PMID21067198,PMID20599654,PMID20127670,PMID20670642,PMID22836907,PMID24834716,PMID22532474,PMID21495717,PMID22727910,PMID20823341,PMID22423588,PMID24661599,PMID23495675,PMID22773043,PMID21613217,PMID20172594,PMID22265637,PMID24420770,PMID24069359,PMID23722687,PMID24304694,PMID22325880,PMID22952939,PMID22307798,PMID22964480,PMID21544200,PMID23523950,PMID22683910,PMID22988760,PMID22323633,PMID22343183,PMID21869564,PMID24266766,PMID24459849,PMID22510452,PMID24211787,PMID23142130,PMID22974423) BOSS trifluoperazine GYPE Text_Mining(PMID24631340,PMID21098645,PMID21632963,PMID21632963,PMID21632963,PMID24601226,PMID24601226,PMID24601226,PMID24601226,PMID21673130,PMID21673130,PMID21673130,PMID21673130,PMID22579593,PMID22579593,PMID22579593,PMID22579593,PMID22579593,PMID22579593,PMID22252501,PMID20375181,PMID20375181,PMID23704698,PMID23704698,PMID23704698,PMID23611809,PMID23611809) BOSS trifluoperazine TNFRSF13C Text_Mining(PMID20851282,PMID24241722,PMID21348624,PMID22817951,PMID21983455,PMID22678547,PMID20382888,PMID24132550,PMID23724438,PMID22974423) BOSS trifluoperazine SLC25A20 Text_Mining(PMID22423588,PMID22234896,PMID23954492,PMID23203067,PMID22988760,PMID22323633,PMID21869564,PMID24266766) BOSS trifluoperazine AURKB Text_Mining(PMID20823341,PMID24266766,PMID22510452,PMID22252501,PMID24211787,PMID22974423) BOSS trifluoperazine ATP1B1 Text_Mining(PMID22796571,PMID22796571,PMID22234896,PMID22234896,PMID23523950) BOSS trifluoperazine TFP1 Text_Mining(PMID20544963,PMID23831300,PMID22952939,PMID20112292,PMID22683910,PMID) BOSS trifluoperazine ABCB1 None=None(uM) D4 PubChem trifluoperazine APAF1 None=None(uM) D4 PubChem trifluoperazine ATXN2 Potency=19.9526(uM) D4 PubChem trifluoperazine ATXN2 Potency=25.1189(uM) D4 PubChem trifluoperazine BAZ2B Potency=35.4813(uM) D4 PubChem trifluoperazine BAZ2B Potency=35481.3(nM) D4 ChEMBL trifluoperazine CBX1 Potency=31.6228(uM) D4 PubChem trifluoperazine CBX1 Potency=31622.8(nM) D4 ChEMBL trifluoperazine CHRM4 None=None(uM) D4 PubChem trifluoperazine CYP19A1 Potency-Replicate_1=26.6032(uM) D4 PubChem trifluoperazine CYP1A2 None=None(uM) D4 PubChem trifluoperazine CYP1A2 AC50=630.96(nM) D4 ChEMBL trifluoperazine CYP1A2 AC50=1000.0(nM) D4 ChEMBL trifluoperazine CYP2C19 Potency=1.9953(uM) D4 PubChem trifluoperazine CYP2C19 Potency=12.5893(uM) D4 PubChem trifluoperazine CYP2C19 None=None(uM) D4 PubChem trifluoperazine CYP2C19 Potency=12589.3(nM) D4 ChEMBL trifluoperazine CYP2C19 AC50=12589.2(nM) D4 ChEMBL trifluoperazine CYP2C19 Potency=1995.3(nM) D4 ChEMBL trifluoperazine CYP2D6 Potency=0.3162(uM) D4 PubChem trifluoperazine CYP2D6 Potency=1.0(uM) D4 PubChem trifluoperazine CYP2D6 Potency=1.9953(uM) D4 PubChem trifluoperazine CYP2D6 None=None(uM) D4 PubChem trifluoperazine CYP2D6 Potency=1995.3(nM) D4 ChEMBL trifluoperazine CYP2D6 AC50=1000.0(nM) D4 ChEMBL trifluoperazine CYP2D6 AC50=1995.26(nM) D4 ChEMBL trifluoperazine CYP2D6 Potency=316.2(nM) D4 ChEMBL trifluoperazine CYP2D6 Potency=1000.0(nM) D4 ChEMBL trifluoperazine CYP3A4 Potency=15.8489(uM) D4 PubChem trifluoperazine CYP3A4 None=None(uM) D4 PubChem trifluoperazine CYP3A4 AC50=15848.9(nM) D4 ChEMBL trifluoperazine CYP3A4 Potency=15848.9(nM) D4 ChEMBL trifluoperazine DRD1 Potency=0.8913(uM) D4 PubChem trifluoperazine DRD1 Potency=891.3(nM) D4 ChEMBL trifluoperazine DRD1 None=None(uM) D4 PubChem trifluoperazine DRD2 None=None(uM) D4 PubChem trifluoperazine DRD3 None=None(uM) D4 PubChem trifluoperazine EHMT2 Potency=11.2202(uM) D4 PubChem trifluoperazine EHMT2 Potency=15.8489(uM) D4 PubChem trifluoperazine EHMT2 Potency=15848.9(nM) D4 ChEMBL trifluoperazine EHMT2 Potency=11220.2(nM) D4 ChEMBL trifluoperazine GLP1R Potency=8.9125(uM) D4 PubChem trifluoperazine GMNN Potency=23.1093(uM) D4 PubChem trifluoperazine HTR2A None=None(uM) D4 PubChem trifluoperazine HTR2C None=None(uM) D4 PubChem trifluoperazine IDH1 Potency=20.5962(uM) D4 PubChem trifluoperazine KCNH2 None=None(uM) D4 PubChem trifluoperazine KCNH2 Potency=2.8184(uM) D4 PubChem trifluoperazine KCNQ1 None=None(uM) D4 PubChem trifluoperazine MAP4K2 None=None(uM) D4 PubChem trifluoperazine MAPK1 Potency=25.1189(uM) D4 PubChem trifluoperazine MAPK1 Potency=25118.9(nM) D4 ChEMBL trifluoperazine MLLT3 None=None(uM) D4 PubChem trifluoperazine MPHOSPH8 Potency=19.9526(uM) D4 PubChem trifluoperazine MPHOSPH8 Potency=19952.6(nM) D4 ChEMBL trifluoperazine PLA2G7 None=None(uM) D4 PubChem trifluoperazine PTGER2 None=None(uM) D4 PubChem trifluoperazine RAD52 AC50_uM=13.0(uM) D4 PubChem trifluoperazine RAD52 None=None(uM) D4 PubChem trifluoperazine RAD52 None=None(uM) D4 PubChem trifluoperazine RGS4 Potency=18.8876(uM) D4 PubChem trifluoperazine SMAD3 None=None(uM) D4 PubChem trifluoperazine STK33 None=None(uM) D4 PubChem trifluoperazine TDP1 Potency=3.7192(uM) D4 PubChem trifluoperazine TDP1 Potency=4.6109(uM) D4 PubChem trifluoperazine TDP1 Potency=5.1735(uM) D4 PubChem trifluoperazine TDP1 Potency=6.6138(uM) D4 PubChem trifluoperazine TDP1 Potency=16.3601(uM) D4 PubChem trifluoperazine TDP1 Potency=4.2172(uM) D4 PubChem trifluoperazine TDP1 Potency=5.9569(uM) D4 PubChem trifluoperazine THPO Potency=15.8489(uM) D4 PubChem trifluoperazine THPO Potency=15848.9(nM) D4 ChEMBL trifluoperazine TP53 Potency=15.8489(uM) D4 PubChem trifluoperazine TP53 Potency=19.9526(uM) D4 PubChem trifluoperazine TP53 Potency=19952.6(nM) D4 ChEMBL trifluoperazine TP53 Potency=15848.9(nM) D4 ChEMBL trifluoperazine UBE2N None=None(uM) D4 PubChem trifluoperazine USP1 Potency=50.1187(uM) D4 PubChem