Drug Gene Type Source Dasatinib DDR2 Text_Mining(PMID23932362,PMID23277333,PMID21523723,PMID20685895,PMID20557276,PMID22469781,PMID22469781,PMID22992064,PMID20959018,PMID22328973,PMID22586301,PMID24296828,PMID20406949,PMID23942795,PMID21792346,PMID21792346,PMID20811002,PMID21937681,PMID23127174,PMID24804581,PMID24804581,PMID21156787,PMID22227013,PMID24718698,PMID21751967,PMID21423210,PMID24819299,PMID24128713,PMID24733895,PMID20860375,PMID24569990,PMID23572291,PMID23192268,PMID20515951,PMID21262832,PMID22262776,PMID20473900,PMID22592211,PMID23896410,PMID23896410,PMID22539950,PMID20736294,PMID23010482,PMID20628031,PMID23020072,PMID23972547,PMID23066441,PMID23899511,PMID23721490,PMID23721490,PMID24069415,PMID24069538,PMID22362357,PMID21523734,PMID23918525,PMID24072218,PMID23872305,PMID22673542,PMID23729178,PMID20565769,PMID24756783,PMID20955590,PMID24501773,PMID21670084) BOSS Dasatinib KIT Text_Mining(PMID24211243,PMID22687981,PMID22127285,PMID23754592,PMID20156689,PMID22936666,PMID23127495,PMID20304669,PMID20304669,PMID20387067,PMID20113198,PMID20406945,PMID23127174,PMID23127174,PMID21153679,PMID21362052,PMID21680801,PMID24718698,PMID20570632,PMID19996579,PMID19996579,PMID20844972,PMID20844972,PMID20591500,PMID20591500,PMID20591500,PMID20662899,PMID23840364,PMID21226671,PMID20145167,PMID21262832,PMID23149070,PMID22410759,PMID21689725,PMID20685771,PMID22246246,PMID20072833,PMID23896410,PMID22539950,PMID23539538,PMID24756784,PMID21419931,PMID21263099,PMID22555087,PMID22652566,PMID21442641,PMID24369222,PMID21523734,PMID24072218,PMID24281418,PMID23582185,PMID23582185,PMID23720340,PMID21463117,PMID24756783,PMID24052572,PMID21670084,PMID24404189) BOSS Dasatinib SRC Text_Mining(PMID20689754,PMID22282699,PMID20226597,PMID20087228,PMID20015594,PMID23516140,PMID20068106,PMID24994118,PMID21528941,PMID20001232,PMID20947248,PMID21976132,PMID22548338,PMID20387067,PMID20190765,PMID21902298,PMID21406471,PMID21153679,PMID21208651,PMID22130962,PMID22233429,PMID22392508,PMID22710723,PMID21282564,PMID21282564,PMID23049365,PMID24420842,PMID24407585,PMID24210599,PMID24676703,PMID22538170,PMID23466625,PMID23112129,PMID22089930,PMID22246246,PMID23580575,PMID23896410,PMID23560534,PMID23319332,PMID21623279,PMID24756784,PMID21286377,PMID23652277,PMID21263099,PMID21781226,PMID24918603,PMID21642769,PMID23318429,PMID23872305,PMID19890374,PMID23696637,PMID21670084) BOSS Dasatinib TPM3 Text_Mining(PMID24062017,PMID21299457,PMID21908430,PMID23569389,PMID24297450,PMID20028401,PMID23913852,PMID23433665,PMID22956142,PMID23836561,PMID22548338,PMID23576564,PMID20387067,PMID20529804,PMID20222756,PMID21792346,PMID21902298,PMID21454413,PMID20537386,PMID22392508,PMID21098337,PMID20460883,PMID22871019,PMID23049365,PMID24779033,PMID24130846,PMID20369050,PMID24297701,PMID24807266,PMID24652384,PMID21278787,PMID23044928,PMID21888027,PMID22262776,PMID23187745,PMID22985168,PMID23825585,PMID24586514,PMID24756784,PMID24756786,PMID24258348,PMID22555087,PMID24350829,PMID23233201,PMID23815902,PMID21463117,PMID21505103,PMID24666486,PMID23729178,PMID19890374,PMID21670084,PMID24404189) BOSS Dasatinib EGFR Text_Mining(PMID21204748,PMID24080257,PMID20685895,PMID23049743,PMID20667610,PMID23594190,PMID20190765,PMID22407177,PMID23800712,PMID21423210,PMID21664897,PMID22761868,PMID20855820,PMID21903773,PMID23242808,PMID24457597,PMID23908684,PMID21881918,PMID20142592,PMID20515951,PMID19804422,PMID19804422,PMID21955398,PMID20473900,PMID21510831,PMID23590835,PMID24216225,PMID21623279,PMID21623279,PMID23010482,PMID23066441,PMID20956938,PMID21266529,PMID23899511,PMID23721490,PMID24919575,PMID22973964,PMID23816254,PMID22787428,PMID20955590,PMID24501773) BOSS Dasatinib AURKB Text_Mining(PMID20807497,PMID20036005,PMID20156689,PMID21842698,PMID22469781,PMID22469781,PMID21883956,PMID21883956,PMID24486585,PMID20190765,PMID22425385,PMID22649091,PMID20684746,PMID22242683,PMID20860375,PMID20425399,PMID22846973,PMID24676703,PMID20145167,PMID23826126,PMID23826126,PMID22721004,PMID22519766,PMID23748749,PMID24260357,PMID21463117,PMID19890374,PMID24713129) BOSS Dasatinib BCR Text_Mining(PMID20597967,PMID21717440,PMID24297450,PMID23180974,PMID20028401,PMID24215620,PMID22956142,PMID19758698,PMID20040619,PMID20222756,PMID22612329,PMID20460883,PMID23090888,PMID23553655,PMID24305542,PMID20310049,PMID23044928,PMID22985168,PMID23825585,PMID24396109,PMID24729196,PMID20143399,PMID24350829,PMID23233201,PMID23815902,PMID24666486,PMID24404189) BOSS Dasatinib TRAF3 Text_Mining(PMID22645182,PMID23630094,PMID20388735,PMID22689211,PMID23598197,PMID20597967,PMID23836556,PMID23676643,PMID21528941,PMID24215620,PMID20659155,PMID20875554,PMID20040619,PMID21792346,PMID21863287,PMID21454413,PMID21376587,PMID20111071,PMID21381013,PMID24333704,PMID21663515,PMID24305542,PMID22721004,PMID24691568,PMID21813412,PMID23872305,PMID24404189) BOSS Dasatinib EPHB2 Text_Mining(PMID24296828,PMID23133664,PMID22649091,PMID24117380,PMID22169110,PMID22306341,PMID21955398,PMID22858987,PMID23325840,PMID23825585,PMID23826126,PMID23560534,PMID22797920,PMID23824064,PMID21286377,PMID21266529,PMID20143399,PMID23721490,PMID24918603,PMID22285507,PMID20955590) BOSS Dasatinib CDT1 Text_Mining(PMID23843632,PMID23843632,PMID20685895,PMID22891038,PMID24107928,PMID22815843,PMID21106726,PMID24133973,PMID21718141,PMID21663515,PMID23065516,PMID24239173,PMID24239173,PMID20423956,PMID20423956,PMID20699436,PMID23374617,PMID24019750,PMID22285507,PMID24480804) BOSS Dasatinib CASP3 Text_Mining(PMID23049975,PMID23588374,PMID24994118,PMID20406949,PMID20863376,PMID23149070,PMID22538170,PMID21455605,PMID23404469,PMID24976045,PMID24586514,PMID24126464,PMID24918603,PMID23233201,PMID20699436,PMID22362357,PMID23918525,PMID24407160,PMID24155950) BOSS Dasatinib IL3 Text_Mining(PMID20304669,PMID20387067,PMID20387067,PMID21220747,PMID20591500,PMID20591500,PMID21299849,PMID22089930,PMID23560534,PMID23539538,PMID21286377,PMID21286377,PMID21286377,PMID20585448,PMID20585448,PMID24407160,PMID24155950,PMID24404189) BOSS Dasatinib STAT3 Text_Mining(PMID24211243,PMID20953816,PMID22130962,PMID20808823,PMID20682659,PMID22246246,PMID23580575,PMID22516066,PMID22797920,PMID21286377,PMID21266529,PMID23721490,PMID20955590,PMID24155950) BOSS Dasatinib ABCA1 Text_Mining(PMID23422267,PMID21423210,PMID20515943,PMID22182854,PMID20682659,PMID23826126,PMID20736294,PMID23066441,PMID20956938,PMID21266529,PMID23899511,PMID21352196,PMID22285507,PMID24155950) BOSS Dasatinib ATP8A2 Text_Mining(PMID24550330,PMID24692691,PMID20423990,PMID21883956,PMID20152788,PMID23279183,PMID21264348,PMID20860375,PMID24457597,PMID21410427,PMID24334291,PMID24258348,PMID23652925) BOSS Dasatinib BCL2 Text_Mining(PMID22414011,PMID20664932,PMID23404469,PMID21813412,PMID20699436,PMID22362357,PMID20351071,PMID21642769,PMID22787428,PMID20629079,PMID24052572) BOSS Dasatinib MAPK3 Text_Mining(PMID20953816,PMID20387067,PMID21106726,PMID24733895,PMID23908684,PMID21299849,PMID21804606,PMID21642769,PMID24480804,PMID24480804,PMID20955590) BOSS Dasatinib KDR Text_Mining(PMID23526749,PMID21423276,PMID21423276,PMID22846973,PMID23149070,PMID21510831,PMID23403636,PMID21177802,PMID24133586,PMID23114714,PMID23536435) BOSS Dasatinib INS Text_Mining(PMID23037470,PMID23179903,PMID20685771,PMID22797920,PMID22797920,PMID23300537,PMID24686085,PMID20852754,PMID21225019,PMID21069103,PMID20664824) BOSS Dasatinib ABCG2 Text_Mining(PMID23843632,PMID23843632,PMID22891038,PMID24107928,PMID24133973,PMID21663515,PMID23065516,PMID24322003,PMID20423956,PMID20423956) BOSS Dasatinib VEGFA Text_Mining(PMID21632985,PMID23325408,PMID21350557,PMID21510831,PMID23403636,PMID21177802,PMID24188312,PMID23114714,PMID22076388) BOSS Dasatinib PTK2 Text_Mining(PMID22130962,PMID20940402,PMID23580575,PMID22328516,PMID22797920,PMID21266529,PMID23721490,PMID23114714,PMID24130049) BOSS Dasatinib CPP Text_Mining(PMID24486585,PMID21153679,PMID22509030,PMID21955398,PMID21286377,PMID21263099,PMID21523734,PMID24072218,PMID20955590) BOSS Dasatinib LYN Text_Mining(PMID20215510,PMID23422267,PMID24091144,PMID21955398,PMID23325840,PMID23896410,PMID19890374,PMID23696637,PMID21670084) BOSS Dasatinib COG3 Text_Mining(PMID21446845,PMID22127285,PMID24994118,PMID22649091,PMID24128713,PMID23242808,PMID22169110,PMID23729178) BOSS Dasatinib HLP Text_Mining(PMID20108303,PMID20108303,PMID20684746,PMID24133973,PMID24819355,PMID24794907,PMID21827214,PMID24713129) BOSS Dasatinib JAK2 Text_Mining(PMID21446845,PMID24007855,PMID23186157,PMID21220747,PMID24528501,PMID23560534,PMID23696637,PMID24404189) BOSS Dasatinib PDGFRB Text_Mining(PMID20579391,PMID20375898,PMID20406945,PMID24733895,PMID20685771,PMID23947765,PMID23114714,PMID23536435) BOSS Dasatinib CSF2 Text_Mining(PMID20130598,PMID23400592,PMID20869423,PMID22246246,PMID23652277,PMID23696637,PMID23696637,PMID20383346) BOSS Dasatinib ERBB2 Text_Mining(PMID21184269,PMID20811002,PMID23299860,PMID21664897,PMID22761868,PMID21903773,PMID22973964,PMID23816254) BOSS Dasatinib BBS9 Text_Mining(PMID21549035,PMID22857863,PMID22036594,PMID24013127,PMID24113234,PMID24333704,PMID22987603,PMID23138519) BOSS Dasatinib IFNA17 Text_Mining(PMID20224653,PMID20071983,PMID22564553,PMID21062247,PMID22937303,PMID20221270,PMID20640942,PMID21197073) BOSS Dasatinib MTOR Text_Mining(PMID21632985,PMID20942869,PMID22583069,PMID21804606,PMID20956938,PMID24878063,PMID22076388) BOSS Dasatinib TNF Text_Mining(PMID22797388,PMID23573828,PMID22133278,PMID24976045,PMID22797920,PMID22234699,PMID22673542) BOSS Dasatinib TPSD1 Text_Mining(PMID21362052,PMID22410759,PMID22583069,PMID21689725,PMID21442641,PMID24369222,PMID23720340) BOSS Dasatinib MET Text_Mining(PMID20406949,PMID22621691,PMID19804422,PMID20628031,PMID24919575,PMID23318429,PMID20955590) BOSS Dasatinib ERBB2 Text_Mining(PMID21184269,PMID21357651,PMID20515951,PMID21862872,PMID22306341,PMID23319332,PMID23010482) BOSS Dasatinib TACR2 Text_Mining(PMID24149438,PMID20111071,PMID22889761,PMID22005789,PMID23325840,PMID20585556,PMID20585448) BOSS Dasatinib IGFBP1 Text_Mining(PMID23371521,PMID23371521,PMID23716272,PMID21862872,PMID23187461,PMID23300537,PMID23300537) BOSS Dasatinib PPARG Text_Mining(PMID21423276,PMID22874537,PMID23192268,PMID20142592,PMID23149070,PMID23536435,PMID20419513) BOSS Dasatinib HPD Text_Mining(PMID20137810,PMID21598241,PMID22344285,PMID23180974,PMID22612329,PMID24691568,PMID23872305) BOSS Dasatinib GCK Text_Mining(PMID21976132,PMID21539969,PMID22234699,PMID22234699,PMID23652277,PMID20351071) BOSS Dasatinib PXDN Text_Mining(PMID21810917,PMID22130962,PMID23275294,PMID24407585,PMID20682659,PMID22570868) BOSS Dasatinib MRC1 Text_Mining(PMID21990394,PMID21442637,PMID22461032,PMID23836561,PMID24832371,PMID22065971) BOSS Dasatinib ESR1 Text_Mining(PMID20634194,PMID21184269,PMID22588706,PMID22306341,PMID21860001,PMID22787428) BOSS Dasatinib CD34 Text_Mining(PMID20068223,PMID23328954,PMID24528501,PMID22089930,PMID23409026,PMID24404189) BOSS Dasatinib FLT1 Text_Mining(PMID20634194,PMID22621691,PMID22874537,PMID23325408,PMID23192268,PMID22076388) BOSS Dasatinib YES1 Text_Mining(PMID20072833,PMID24756784,PMID21642769,PMID21523734,PMID23318429,PMID21670084) BOSS Dasatinib EGF Text_Mining(PMID22490227,PMID23242808,PMID23319332,PMID20383201,PMID20419513,PMID24501773) BOSS Dasatinib PRRT2 Text_Mining(PMID25031773,PMID24569990,PMID23826126,PMID24260357,PMID24501773,PMID24504051) BOSS Dasatinib AK5 Text_Mining(PMID21406471,PMID22392508,PMID22837181,PMID24173967,PMID20310049,PMID21263099) BOSS Dasatinib AKR1B1 Text_Mining(PMID24403252,PMID21633166,PMID23236591,PMID22672122,PMID20383201,PMID23748749) BOSS Dasatinib CXCL12 Text_Mining(PMID21385851,PMID23133664,PMID23133664,PMID24149438,PMID22889761,PMID22005789) BOSS Dasatinib IL6 Text_Mining(PMID21647156,PMID21197073,PMID20515943,PMID23826126,PMID20383201,PMID23652277) BOSS Dasatinib BTK Text_Mining(PMID20052711,PMID24080257,PMID21883956,PMID23719297,PMID22612424) BOSS Dasatinib BCL2L1 Text_Mining(PMID22344285,PMID21642769,PMID20585448,PMID20585448,PMID24052572) BOSS Dasatinib LCK Text_Mining(PMID20190765,PMID20072833,PMID24756784,PMID23872305,PMID21670084) BOSS Dasatinib CBX8 Text_Mining(PMID22130962,PMID20515943,PMID23300537,PMID23114714,PMID24245541) BOSS Dasatinib TP53 Text_Mining(PMID21106726,PMID23896410,PMID22721004,PMID22362357,PMID24133586) BOSS Dasatinib CSF1 Text_Mining(PMID22425926,PMID22425926,PMID20156689,PMID21873591,PMID20225261) BOSS Dasatinib CASP8 Text_Mining(PMID24352878,PMID24352878,PMID20515951,PMID23404469,PMID22354875) BOSS Dasatinib PTEN Text_Mining(PMID24486585,PMID24091144,PMID23319332,PMID23721490,PMID22285507) BOSS Dasatinib PTK2B Text_Mining(PMID23908684,PMID21299849,PMID23300537,PMID20629079,PMID20664824) BOSS Dasatinib FAM109A Text_Mining(PMID22183070,PMID20808823,PMID24396109,PMID21286377,PMID22285507) BOSS Dasatinib PAX3 Text_Mining(PMID23142123,PMID20145167,PMID22262776,PMID22710719,PMID22362357) BOSS Dasatinib MTF1 Text_Mining(PMID24229357,PMID24229357,PMID22770610,PMID22770610,PMID22770610) BOSS Dasatinib RASGRF1 Text_Mining(PMID21423210,PMID24434513,PMID20515943,PMID22328516,PMID20585556) BOSS Dasatinib CAV3 Text_Mining(PMID24486585,PMID22570868,PMID21286377,PMID23114714,PMID23114714,PMID) BOSS Dasatinib ABL1 None=0.53(uM) D4 PubChem Dasatinib ABL1 None=0.72(uM) D4 PubChem Dasatinib ABL1 None=0.96(uM) D4 PubChem Dasatinib ABL1 None=1.1(uM) D4 PubChem Dasatinib ABL1 None=1.2(uM) D4 PubChem Dasatinib ABL1 None=2.1(uM) D4 PubChem Dasatinib ABL2 None=0.17(uM) D4 PubChem Dasatinib AHR Potency-Replicate_1=1.1883(uM) D4 PubChem Dasatinib AR Ratio Potency (uM)=10.6822(uM) D4 PubChem Dasatinib AR Potency-Replicate_1=11.9856(uM) D4 PubChem Dasatinib AR Potency-Replicate_1=26.6032(uM) D4 PubChem Dasatinib BLK None=0.21(uM) D4 PubChem Dasatinib BMX None=1.4(uM) D4 PubChem Dasatinib BTK None=1.4(uM) D4 PubChem Dasatinib BTK Activity=None(Unspecified) D4 ChEMBL Dasatinib CSF1R None=0.58(uM) D4 PubChem Dasatinib CSK None=1.0(uM) D4 PubChem Dasatinib CYP19A1 Potency-Replicate_1=1.3333(uM) D4 PubChem Dasatinib DDR1 None=0.69(uM) D4 PubChem Dasatinib DDR2 None=3.2(uM) D4 PubChem Dasatinib EPHA1 None=4.1(uM) D4 PubChem Dasatinib EPHA2 None=0.85(uM) D4 PubChem Dasatinib EPHA3 None=0.093(uM) D4 PubChem Dasatinib EPHA4 None=1.2(uM) D4 PubChem Dasatinib EPHA5 None=0.24(uM) D4 PubChem Dasatinib EPHA8 None=0.24(uM) D4 PubChem Dasatinib EPHB1 None=0.45(uM) D4 PubChem Dasatinib EPHB2 None=0.39(uM) D4 PubChem Dasatinib EPHB3 None=6.9(uM) D4 PubChem Dasatinib EPHB4 None=0.34(uM) D4 PubChem Dasatinib FGR None=0.5(uM) D4 PubChem Dasatinib FRK None=0.31(uM) D4 PubChem Dasatinib FYN None=0.79(uM) D4 PubChem Dasatinib GAK None=2.6(uM) D4 PubChem Dasatinib GMNN Potency=16.7889(uM) D4 PubChem Dasatinib GMNN Potency=18.8375(uM) D4 PubChem Dasatinib HCK None=0.35(uM) D4 PubChem Dasatinib KIT None=0.62(uM) D4 PubChem Dasatinib KIT None=0.68(uM) D4 PubChem Dasatinib KIT None=2.6(uM) D4 PubChem Dasatinib KIT None=2.7(uM) D4 PubChem Dasatinib LCK None=0.2(uM) D4 PubChem Dasatinib LYN None=0.57(uM) D4 PubChem Dasatinib NR0B1 None=None(uM) D4 PubChem Dasatinib NR2F2 None=None(uM) D4 PubChem Dasatinib NR3C1 None=None(uM) D4 PubChem Dasatinib PDGFRA None=0.47(uM) D4 PubChem Dasatinib PDGFRB None=0.63(uM) D4 PubChem Dasatinib PPARD Potency-Replicate_1=0.473(uM) D4 PubChem Dasatinib PPARG None=None(uM) D4 PubChem Dasatinib PRNP None=None(uM) D4 PubChem Dasatinib PTK6 None=7.8(uM) D4 PubChem Dasatinib SIK1 None=3.9(uM) D4 PubChem Dasatinib SIK2 None=6.4(uM) D4 PubChem Dasatinib SMAD3 Potency=1.2589(uM) D4 PubChem Dasatinib SRC None=0.21(uM) D4 PubChem Dasatinib SRC Activity=None(Unspecified) D4 ChEMBL Dasatinib TDP1 Potency=2.1136(uM) D4 PubChem Dasatinib TDP1 Potency=2.3715(uM) D4 PubChem Dasatinib TDP1 Potency=2.8184(uM) D4 PubChem Dasatinib TDP1 Potency=3.9811(uM) D4 PubChem Dasatinib TEC Activity=None(Unspecified) D4 ChEMBL Dasatinib TNK2 None=5.6(uM) D4 PubChem Dasatinib TXK None=2.1(uM) D4 PubChem Dasatinib YES1 Potency=0.0024(uM) D4 PubChem Dasatinib YES1 None=0.3(uM) D4 PubChem