Drug Gene Type Source raloxifene ESR1 Text_Mining(PMID19819155,PMID20145354,PMID23664736,PMID20190360,PMID20190369,PMID21741883,PMID21966167,PMID23103222,PMID20171784,PMID22453607,PMID23546819,PMID23955099,PMID23157045,PMID21505049,PMID22170716,PMID22061801,PMID23988275,PMID21953363,PMID24036624,PMID20958960,PMID22622807,PMID24418098,PMID23772059,PMID23842642,PMID21335463,PMID20926342,PMID24757949,PMID20399327,PMID24228255,PMID20513233,PMID21228613,PMID20083158,PMID20190364,PMID19828145,PMID24108389,PMID23165656,PMID22398780,PMID22290018,PMID21693498,PMID22223434,PMID22679310,PMID21774370,PMID22619254,PMID24136418,PMID25012765,PMID22164341,PMID24389818,PMID20816507,PMID22534326,PMID21467260,PMID21880792,PMID23621618,PMID22453024,PMID21088662,PMID20452495,PMID20169039,PMID20551107,PMID20927038,PMID22403109,PMID21719986,PMID21871812,PMID22139492,PMID23076912,PMID23737033,PMID22543247,PMID20661164,PMID21601973,PMID22161827,PMID21903021,PMID22476901,PMID20674746,PMID23170835,PMID20386345,PMID21513812,PMID21397017,PMID20207825,PMID20429824,PMID23036732,PMID23227210,PMID24061412,PMID23344476,PMID23246169,PMID21937736,PMID24495098,PMID24999330,PMID20518194,PMID21654612,PMID20569451,PMID25054138,PMID24347426,PMID23727128,PMID24833917,PMID21072271,PMID21072279,PMID22739699,PMID22035517,PMID23635953,PMID23613312,PMID24775644,PMID21595855,PMID20102385,PMID21315285,PMID20945400,PMID20092935,PMID21294695,PMID20480545,PMID20544555,PMID22319035,PMID23942473,PMID22533838,PMID23201442,PMID22285935,PMID21753870,PMID22005391,PMID21493749,PMID22635014,PMID21689408,PMID20596666,PMID21666713,PMID20609538,PMID22405286,PMID23630443,PMID19745773,PMID20017619,PMID23810002,PMID22480687,PMID22105178,PMID22311517,PMID23462505,PMID22212320,PMID24410282,PMID24722370,PMID24595623,PMID22889955,PMID22853318,PMID19996623,PMID21964465,PMID21742056,PMID20603714,PMID20185791,PMID19914376,PMID23835710,PMID24342775,PMID21290426,PMID20446043,PMID23665515,PMID22647137,PMID24689036,PMID20843951,PMID22925430,PMID24526372,PMID24810565,PMID24205315,PMID23471663,PMID21159208,PMID20613670,PMID21376723,PMID23173704,PMID22684228,PMID23764426,PMID20938747,PMID23225083,PMID24311443,PMID24618912,PMID24770313,PMID24109197,PMID19798460,PMID20107426,PMID23276611,PMID21993078,PMID22429462,PMID22841776,PMID22140478,PMID21600284,PMID20686605,PMID21536054,PMID20664987,PMID23062036,PMID22683727,PMID21158712,PMID20888885,PMID24406683,PMID24373794,PMID24782323,PMID20073985,PMID21175240,PMID21185374,PMID20473319,PMID21920358,PMID19533603,PMID21395502,PMID21737572,PMID24516352,PMID24964310,PMID24367182,PMID22845341,PMID22466336,PMID20688441,PMID24080207,PMID23171676,PMID23777900,PMID24431404,PMID21982237,PMID24481452,PMID24598415,PMID21420980,PMID23682072,PMID24069582,PMID25035541,PMID23786776,PMID24518153,PMID22716221,PMID21253797,PMID24346250,PMID24037977,PMID20372779,PMID24615483) BOSS raloxifene EREG Text_Mining(PMID24697167,PMID20447057,PMID20083158,PMID20083158,PMID23639488,PMID20419096,PMID20419096,PMID20814901,PMID23170835,PMID22819149,PMID20659801,PMID21184272,PMID21253796,PMID25054138,PMID25048912,PMID20387803,PMID20387803,PMID20544555,PMID20596666,PMID21501150,PMID20609538,PMID20609538,PMID23323567,PMID24880111,PMID21671899,PMID20824855,PMID21624057,PMID22077482,PMID24015958,PMID24785473,PMID21564348,PMID20686605,PMID20555430,PMID23634843,PMID20073985,PMID21420980,PMID20372779,PMID20372779) BOSS raloxifene PTH Text_Mining(PMID20034599,PMID21069410,PMID20621892,PMID22572963,PMID20189664,PMID24722767,PMID24722767,PMID20839286,PMID20839286,PMID20839286,PMID20190367,PMID22130786,PMID21072279,PMID21321169,PMID23843805,PMID21595855,PMID20228675,PMID20428990,PMID23078546,PMID22311517,PMID21046091,PMID20449570,PMID20446043,PMID22925430,PMID24795812,PMID24100598,PMID24100401,PMID19957165,PMID21175240,PMID24964310,PMID21542947,PMID22716221) BOSS raloxifene TCP1 Text_Mining(PMID20532481,PMID24515577,PMID19757416,PMID21753740,PMID24081731,PMID22099387,PMID22265062,PMID23831360,PMID22256806,PMID21542002,PMID21667891,PMID21901476,PMID23828276,PMID19898839,PMID23263929,PMID20228675,PMID23121774,PMID22635014,PMID21824859,PMID20428990,PMID22715862,PMID20446043,PMID22925430,PMID20843165,PMID21075980,PMID24641458,PMID24606074,PMID21542947,PMID22716221) BOSS raloxifene CYP2C8 Text_Mining(PMID21880792,PMID20459297,PMID21493749,PMID22859722,PMID22859722,PMID22859722,PMID22859722,PMID22859722,PMID22515117,PMID22515117,PMID21600284,PMID21600284,PMID21870861,PMID21870861,PMID23786776) BOSS raloxifene HLP Text_Mining(PMID21997754,PMID22112384,PMID21767526,PMID20405834,PMID20405834,PMID22421793,PMID22942318,PMID20812728,PMID20812728,PMID21859377,PMID21859377,PMID22375838,PMID22859722) BOSS raloxifene BTF3P11 Text_Mining(PMID21536255,PMID20963556,PMID23873632,PMID19948337,PMID21050847,PMID21519319,PMID21519319,PMID22067277,PMID20938747,PMID24964310,PMID24615483,PMID24615483) BOSS raloxifene CEACAM1 Text_Mining(PMID20036346,PMID25037077,PMID21660558,PMID23632659,PMID21617993,PMID22762129,PMID21187295,PMID20428990,PMID22311517,PMID21970822,PMID19798460,PMID24641458) BOSS raloxifene BEST1 Text_Mining(PMID21774365,PMID20687153,PMID20601292,PMID23281041,PMID21774355,PMID23092698,PMID24791357,PMID21595855,PMID23035625,PMID24942322,PMID22338309) BOSS raloxifene IGFBP1 Text_Mining(PMID22170716,PMID21285152,PMID19048282,PMID20207825,PMID22319035,PMID20843951,PMID22669332,PMID22669332,PMID23786776) BOSS raloxifene PGR Text_Mining(PMID21473058,PMID21184272,PMID23665515,PMID21185374,PMID23171676,PMID24481452,PMID24069582,PMID23786776,PMID20372779) BOSS raloxifene CYP2B6 Text_Mining(PMID21997754,PMID21767526,PMID21303923,PMID22909231,PMID22909231,PMID22942318,PMID20812728,PMID22859722,PMID21870861) BOSS raloxifene MAPK3 Text_Mining(PMID22480687,PMID22480687,PMID20686605,PMID21536054,PMID21536054,PMID22683727,PMID24726471,PMID20372779) BOSS raloxifene GYPE Text_Mining(PMID21937736,PMID22661630,PMID22661630,PMID24399855,PMID24399855,PMID24399855,PMID24399855,PMID23682072) BOSS raloxifene CYGB Text_Mining(PMID22112384,PMID21303923,PMID22421793,PMID22909231,PMID22942318,PMID20812728,PMID22859722,PMID21870861) BOSS raloxifene AOX1 Text_Mining(PMID23918666,PMID23918666,PMID22996261,PMID24824603,PMID24156774,PMID24406683,PMID22404107) BOSS raloxifene EGFR Text_Mining(PMID23842642,PMID21666713,PMID24689036,PMID24015958,PMID20664987,PMID24782323,PMID21253797) BOSS raloxifene UGT1A10 Text_Mining(PMID21859377,PMID21859377,PMID21859377,PMID23499758,PMID23499758,PMID23499758,PMID23682072) BOSS raloxifene TNFSF11 Text_Mining(PMID21536255,PMID19948337,PMID21050847,PMID24942322,PMID20938747,PMID24964310,PMID24615483) BOSS raloxifene XDH Text_Mining(PMID21939274,PMID24824603,PMID24824603,PMID20888885,PMID24406683,PMID22404107) BOSS raloxifene CCNL2 Text_Mining(PMID20564133,PMID24253314,PMID23588749,PMID20956826,PMID21666713,PMID21395502) BOSS raloxifene BCL2 Text_Mining(PMID20447057,PMID21573987,PMID20945400,PMID22260523,PMID24516352,PMID24726471) BOSS raloxifene MERTK Text_Mining(PMID22453024,PMID22212320,PMID21742056,PMID24782323,PMID24726471,PMID20372779) BOSS raloxifene CASP3 Text_Mining(PMID20945400,PMID19745773,PMID22480687,PMID23385821,PMID22965848,PMID21420980) BOSS raloxifene IL6 Text_Mining(PMID21372495,PMID22311517,PMID24456369,PMID21159208,PMID19533603,PMID19533603) BOSS raloxifene INS Text_Mining(PMID23638622,PMID23263929,PMID22077482,PMID24311443,PMID24641458,PMID21185374) BOSS raloxifene VEGFA Text_Mining(PMID22066937,PMID20590611,PMID19828145,PMID20017619,PMID20686605) BOSS raloxifene RALA Text_Mining(PMID23871851,PMID20839286,PMID24939720,PMID21912817,PMID22841776) BOSS raloxifene SOST Text_Mining(PMID21660558,PMID22451221,PMID24964310,PMID22338309,PMID24615483) BOSS raloxifene EPHB2 Text_Mining(PMID20945400,PMID23471663,PMID21536054,PMID24782323,PMID20372779) BOSS raloxifene TNFRSF11A Text_Mining(PMID21824859,PMID24964310,PMID22338309,PMID24615483,PMID24615483) BOSS raloxifene SHBG Text_Mining(PMID20096825,PMID22319035,PMID22077482,PMID20843951,PMID23786776) BOSS raloxifene TNF Text_Mining(PMID21513812,PMID23221506,PMID22067277,PMID22480687,PMID22845341,PMID) BOSS raloxifene ALDH1A1 Potency=0.5012(uM) D4 PubChem raloxifene ALDH1A1 Potency=1.122(uM) D4 PubChem raloxifene ALDH1A1 Potency=2511.9(nM) D4 ChEMBL raloxifene ALDH1A1 Potency=1122.0(nM) D4 ChEMBL raloxifene ALDH1A1 Potency=501.2(nM) D4 ChEMBL raloxifene ATXN2 Potency=28.1838(uM) D4 PubChem raloxifene CBX1 Potency=31.6228(uM) D4 PubChem raloxifene CBX1 Potency=31622.8(nM) D4 ChEMBL raloxifene CYP19A1 Potency-Replicate_1=0.0039(uM) D4 PubChem raloxifene CYP19A1 None=None(uM) D4 PubChem raloxifene CYP1A2 Inhibition=None(Unspecified) D4 ChEMBL raloxifene CYP2C19 Potency=10.0(uM) D4 PubChem raloxifene CYP2C19 None=None(uM) D4 PubChem raloxifene CYP2C19 Potency=10000.0(nM) D4 ChEMBL raloxifene CYP2C19 AC50=10000.0(nM) D4 ChEMBL raloxifene CYP2C19 Inhibition=None(Unspecified) D4 ChEMBL raloxifene CYP2D6 Potency=7.9433(uM) D4 PubChem raloxifene CYP2D6 Potency=25.1189(uM) D4 PubChem raloxifene CYP2D6 None=None(uM) D4 PubChem raloxifene CYP2D6 AC50=25118.9(nM) D4 ChEMBL raloxifene CYP2D6 Inhibition=None(Unspecified) D4 ChEMBL raloxifene CYP2D6 Potency=7943.3(nM) D4 ChEMBL raloxifene CYP2D6 Potency=25118.9(nM) D4 ChEMBL raloxifene CYP2D6 AC50=7943.28(nM) D4 ChEMBL raloxifene CYP3A4 Potency=1.2589(uM) D4 PubChem raloxifene CYP3A4 Potency=2.5119(uM) D4 PubChem raloxifene CYP3A4 None=None(uM) D4 PubChem raloxifene CYP3A4 AC50=1258.93(nM) D4 ChEMBL raloxifene CYP3A4 AC50=2511.89(nM) D4 ChEMBL raloxifene CYP3A4 Inhibition=None(Unspecified) D4 ChEMBL raloxifene CYP3A4 Potency=1258.9(nM) D4 ChEMBL raloxifene CYP3A4 Potency=2511.9(nM) D4 ChEMBL raloxifene ESR1 Ratio Potency (uM)=0.001(uM) D4 PubChem raloxifene ESR1 ER Potency (uM)=0.00331156(uM) D4 PubChem raloxifene ESR1 Potency-Replicate_1=0.0043(uM) D4 PubChem raloxifene ESR1 Potency-Replicate_1=None(uM) D4 PubChem raloxifene ESR1 Activity=None(Unspecified) D4 ChEMBL raloxifene ESR2 Activity=None(Unspecified) D4 ChEMBL raloxifene GLS Potency=2.8184(uM) D4 PubChem raloxifene HSD17B10 Potency=7943.3(nM) D4 ChEMBL raloxifene HSPB1 Ratio Potency (uM)=57.1533(uM) D4 PubChem raloxifene IL6R Inhibition=None(Unspecified) D4 ChEMBL raloxifene IL6ST Inhibition=None(Unspecified) D4 ChEMBL raloxifene IL6ST Activity=None(Unspecified) D4 ChEMBL raloxifene ITGA4 None=None(uM) D4 PubChem raloxifene MAPT Potency=14125.4(nM) D4 ChEMBL raloxifene THPO Potency=15.8489(uM) D4 PubChem raloxifene THPO Potency=15848.9(nM) D4 ChEMBL raloxifene TP53 Potency=19.9526(uM) D4 PubChem raloxifene TP53 Potency=25.1189(uM) D4 PubChem raloxifene TP53 Potency=19952.6(nM) D4 ChEMBL raloxifene TP53 Potency=25118.9(nM) D4 ChEMBL