Drug Gene Type Source astemizole LYZ Text_Mining(PMID21807463,PMID21130885,PMID21782952,PMID22580022,PMID21752343,PMID20816809,PMID21824474,PMID22579550,PMID22626564,PMID20883799,PMID22155010,PMID22475776,PMID22032903,PMID22551979,PMID21300159,PMID21983421) BOSS astemizole CYP2C8 Text_Mining(PMID24788058,PMID22328583,PMID22328583,PMID22328583,PMID22328583,PMID22328583,PMID19923256,PMID24021950,PMID24021950,PMID24021950,PMID24021950,PMID20926621,PMID20926621,PMID20926621,PMID20926621,PMID20926621) BOSS astemizole KCNH1 Text_Mining(PMID21443504,PMID21508374,PMID22495877,PMID19932096,PMID24819656,PMID22930803,PMID22984610,PMID22357737,PMID22357737,PMID21315112,PMID23881642,PMID23881642) BOSS astemizole MPO Text_Mining(PMID21782952,PMID20816809,PMID21824474,PMID22626564,PMID22155010,PMID22475776,PMID21300159,PMID23926395,PMID) BOSS astemizole ABCB1 None=None(uM) D4 PubChem astemizole APAF1 None=None(uM) D4 PubChem astemizole APLNR None=None(uM) D4 PubChem astemizole AR Potency-Replicate_1=12.464(uM) D4 PubChem astemizole AR Potency-Replicate_1=18.9959(uM) D4 PubChem astemizole AVPR1A None=None(uM) D4 PubChem astemizole CACNA1H None=None(uM) D4 PubChem astemizole CYP19A1 Potency-Replicate_1=6.2468(uM) D4 PubChem astemizole CYP19A1 Potency-Replicate_1=21.1317(uM) D4 PubChem astemizole CYP2D6 Potency=7.9433(uM) D4 PubChem astemizole CYP2D6 None=None(uM) D4 PubChem astemizole CYP2D6 AC50=7943.28(nM) D4 ChEMBL astemizole CYP2D6 Potency=7943.3(nM) D4 ChEMBL astemizole DRD1 None=None(uM) D4 PubChem astemizole GMNN Potency=3.6626(uM) D4 PubChem astemizole GMNN Potency=4.6109(uM) D4 PubChem astemizole GMNN Potency=23.715(uM) D4 PubChem astemizole GNA15 None=None(uM) D4 PubChem astemizole HPSE Activity=None(Unspecified) D4 ChEMBL astemizole IDH1 Potency=14.581(uM) D4 PubChem astemizole IL1B None=None(uM) D4 PubChem astemizole ITGA4 None=None(uM) D4 PubChem astemizole JAK2 None=None(uM) D4 PubChem astemizole MAP4K2 None=None(uM) D4 PubChem astemizole MDM2 None=None(uM) D4 PubChem astemizole MDM4 None=None(uM) D4 PubChem astemizole MITF None=None(uM) D4 PubChem astemizole MMP14 EC50=None(uM) D4 PubChem astemizole OXTR None=None(uM) D4 PubChem astemizole PAX8 None=None(uM) D4 PubChem astemizole PPARD Potency-Replicate_1=29.847(uM) D4 PubChem astemizole PPARG Potency-Replicate_1=29.847(uM) D4 PubChem astemizole STK33 None=None(uM) D4 PubChem astemizole TAAR1 None=None(uM) D4 PubChem astemizole TDP1 Potency=2.6609(uM) D4 PubChem astemizole TDP1 Potency=3.7586(uM) D4 PubChem astemizole TDP1 Potency=7.3078(uM) D4 PubChem astemizole TDP1 Potency=10.3225(uM) D4 PubChem astemizole TDP1 Potency=14.581(uM) D4 PubChem astemizole TDP1 Potency=16.3601(uM) D4 PubChem astemizole TP53 Potency=12.5893(uM) D4 PubChem astemizole TP53 Potency=12589.3(nM) D4 ChEMBL astemizole UBE2N None=None(uM) D4 PubChem