GSK429286A http://dsigdb.tanlab.org/DSigDBv1.0/displayDrug.py?db=d2_lincs&id=771 PRKACA ROCK2 NUAK2 ROCK1 PRKAA1 LATS2 PRKG1 RET BLK PRKACB JAK2 PRKX STK38L BTK JAK3 BS-181 http://dsigdb.tanlab.org/DSigDBv1.0/displayDrug.py?db=d2_lincs&id=813 CSNK1A1L CSNK1A1 CDK7 TTK CSNK1E CSNK1D STK33 HIPK4 DYRK1A CLK1 CLK2 DYRK1B CLK4 PHKG2 Barasertib http://dsigdb.tanlab.org/DSigDBv1.0/displayDrug.py?db=d2_lincs&id=632 MUSK PDGFRB PDGFRA MAP4K5 MKNK2 RPS6KB1 STK10 EGFR PLK4 RET MAP2K5 HIPK4 ABL1 FLT3 AXL FLT1 TEK PIK3CA CSF1R NTRK1 NTRK2 DSTYK AURKA AURKB KDR ERBB2 EPHB6 ERBB4 CDK11A CDK11B BLK ANKK1 EIF2AK1 DDR1 KIT CDK7 TIE1 LCK BTK WH-4-025 http://dsigdb.tanlab.org/DSigDBv1.0/displayDrug.py?db=d2_lincs&id=402 STK10 PTK2B ROS1 FGR NTRK3 LYN ERBB4 FGFR3 RET FGFR4 FGFR2 TESK1 FGFR1 ZAK SYK KIT PAK3 EPHB4 SRMS JAK2 JAK3 BMX EPHB2 EPHB3 EPHB1 CSK CDK11A CDK11B BLK HCK TNK2 TNK1 DDR1 STK36 TIE1 LCK BTK PDGFRB PDGFRA EPHA8 EPHA7 EPHA6 EPHA5 EPHA4 EPHA3 EPHA2 EPHA1 MAPK14 TNIK MAPK11 ABL1 FLT4 ABL2 FLT1 TEK SIK1 SIK2 TEC CSF1R MAPK7 KDR SRC FRK FER FES MERTK LTK TNNI3K ALK MAP4K1 PTK2 MAP4K5 MAP4K4 PTK6 LIMK2 LIMK1 EGFR PRKAA2 PRKAA1 RIPK2 CIT YES1 TXK FYN SLK BRAF AS601245 http://dsigdb.tanlab.org/DSigDBv1.0/displayDrug.py?db=d2_lincs&id=774 MAPK12 MKNK2 PLK3 EGFR HIPK3 HIPK2 HIPK1 DYRK2 MAPK10 RIPK4 MAP2K5 MAP2K4 TYK2 BMP2K SRMS GAK JAK3 JAK1 DYRK1A MAPK8 IRAK1 PIP4K2C ERBB2 ULK3 EPHB6 PIM3 PIM1 STK16 AAK1 PIK3C2G ANKK1 CSNK2A2 CSNK2A1 RIOK2 RPS6KA3 CSNK1A1 PIP5K1C MAPK9 SNRK GSK3A MAP2K1 GSK3B BRAF MAP3K19 CLK2 GSK1059615 http://dsigdb.tanlab.org/DSigDBv1.0/displayDrug.py?db=d2_lincs&id=724 TSSK1B STK10 STK11 STK16 HIPK3 HIPK2 HIPK1 HIPK4 AXL GRK7 PIK3CB PIK3CD PIK3CG CSNK1D CSNK1E DMPK DYRK1A IRAK3 IRAK1 PIP4K2C PIP4K2B CAMK2D CAMK2A CAMK2B CSNK1G2 CSNK1G3 RIOK1 PIK3C2G STK17B CSNK2A2 CSNK2A1 STK17A MYLK BMPR2 DCLK3 MAPKAPK5 NEK10 JAK3 PHKG2 BUB1 RPS6KA2 RPS6KA5 RPS6KA6 CAMKK2 CAMKK1 STK33 PIK3CA CLK1 CLK2 CLK3 CLK4 PI4KB BMPR1B MAPK15 DYRK2 BMP2K GSG2 MYLK4 MTOR MERTK TAOK1 TAOK3 RIOK3 DYRK1B EIF2AK4 CDK7 CDK8 MAP4K2 CIT MAP2K2 MAP2K1 MAP2K4 CDK19 MELK CDK15 GAK DAPK3 DAPK2 DAPK1 PIM2 PIM3 PIM1 AAK1 SLK PIK3C2B MAP3K19 AG1478 http://dsigdb.tanlab.org/DSigDBv1.0/displayDrug.py?db=d2_lincs&id=210 MKNK2 EPHA6 STK10 CIT EGFR RET MAPK10 MAP2K5 HIPK4 ABL1 MAPKAPK5 FLT3 MAP3K3 GAK LYN IRAK1 CHEK2 IRAK4 ERBB2 SRC MKNK1 BUB1 ERBB4 PIK3C2B BLK SLK HCK PIP5K1C DDR1 MAP3K19 LCK HG-5-113-01 http://dsigdb.tanlab.org/DSigDBv1.0/displayDrug.py?db=d2_lincs&id=77 MUSK STK10 STK16 PLK4 PTK2B INSRR TYK2 ROS1 AXL MAP3K9 MAP3K3 NTRK1 FGR NTRK3 DMPK IRAK3 DYRK1B PIP4K2B IGF1R CSNK1G2 STK3 STK4 CSNK2A1 FGFR1 SYK KIT BMPR2 STK38L PAK3 NUAK1 NUAK2 DCLK3 TTK JAK2 JAK3 JAK1 BMX PRKACB BLK SBK3 TNK2 TNK1 RPS6KA4 STK33 STK35 PIK3CA CLK1 CLK2 CLK3 CLK4 LCK BTK PDGFRB EPHA7 RET MAP3K7 MAPK15 PTK2 NTRK2 HCK ABL1 ABL2 FLT3 TEK SIK1 SIK2 TEC BMP2K MARK4 MARK3 MAPK8 SRC RPS6KA1 RPS6KA2 FER FES MERTK LTK SRPK1 TAOK1 SRPK3 TAOK3 RIOK2 RIOK3 RIOK1 ITK PIP5K1A INSR MET CDK7 MAP4K1 MAP4K3 MAP4K2 MAP4K5 PRKAA2 PRKAA1 MAP2K3 MAP2K2 MAP2K1 YES1 ALK FYN GAK AURKA AURKB AURKC ULK2 ULK3 ULK1 PKN1 PKN2 PRKCD AAK1 SLK TIE1 ROCK2 MAP3K11 MAP3K12 NPK76-II-72-1 http://dsigdb.tanlab.org/DSigDBv1.0/displayDrug.py?db=d2_lincs&id=195 RPS6KA2 PTK2 ALK RPS6KA6 PLK3 DCLK1 MYLK TTK PTK2B STK33 GAK SLK CLK2 PLX4032 http://dsigdb.tanlab.org/DSigDBv1.0/displayDrug.py?db=d2_lincs&id=154 PDGFRB PDGFRA MAP4K5 PI4KB PTK6 CSF1R TNIK MAP2K2 MAP2K1 RIPK2 MAP2K5 MAP2K4 ABL1 RAF1 FLT3 AXL CDK19 SIK1 FYN FGR SRMS TGFBR2 EPHB6 CSK MYLK4 SRC STK3 STK4 BLK SLK HCK TNK2 ZAK DDR1 EIF2AK4 KIT HUNK BRAF STK36 CDK8 PRKD1 LCK HG-9-91-01 http://dsigdb.tanlab.org/DSigDBv1.0/displayDrug.py?db=d2_lincs&id=566 STK10 STK16 PTK2B MAP3K2 MAP3K3 MAP3K7 FGR TESK1 STK24 DMPK LYN IRAK1 JAK3 ERBB2 ERBB3 ERBB4 PIK3C2B RET FGFR4 FGFR2 FGFR3 FGFR1 ZAK KIT HUNK PAK6 PAK7 PAK1 MYO3A MYO3B ACVR1B DSTYK NUAK2 DCLK3 DCLK2 ACVRL1 NEK10 EPHB4 LRRK2 TTK STK26 STK25 CDC42BPG CDC42BPA CDC42BPB PRKACA BMX CHEK2 EPHB2 EPHB3 EPHB1 EPHB6 CSK SRMS BLK HCK SBK1 TNK2 TNK1 RPS6KA3 RPS6KA6 DDR2 DDR1 STK35 STK36 LCK BTK PDGFRB PDGFRA EPHA8 EPHA7 EPHA6 EPHA5 EPHA4 EPHA3 EPHA2 EPHA1 MAPK14 TNIK MAPK10 MAPK11 ABL1 ACVR1 ABL2 FLT1 TEK SIK1 SIK3 PTK6 CSF1R BMP2K CSNK1E MAPK7 MARK2 MARK3 MAPK8 MAPK9 KDR MARK1 TGFBR2 ACVR2B RPS6KA1 FRK RPS6KA2 FES LTK TAOK1 TAOK2 TAOK3 ALK BMPR1A MET CDK4 PRKACB STK32B PRKD1 PRKD2 PRKD3 MAP4K1 MAP4K3 MAP4K2 MAP4K5 MAP4K4 ACVR2A LIMK2 LIMK1 EGFR TGFBR1 MAP2K3 MAP2K2 BMPR1B RIPK2 MAP2K5 CIT STK32A YES1 MINK1 MAP2K4 ADCK4 FYN GAK AURKA ULK2 ULK3 ULK1 PRKCE SRC SLK TXK TNNI3K MAP3K10 BRAF MAP3K19 Dinaciclib http://dsigdb.tanlab.org/DSigDBv1.0/displayDrug.py?db=d2_lincs&id=1155 CDK16 NUAK2 HIPK3 MAPK15 HIPK1 CDKL3 CDKL2 CDK18 CDKL5 CDK13 CDKL1 CDK17 CDK14 CDK15 STK25 CSNK1E MAPK7 DYRK1A DYRK1B ICK CLK2 CDK9 TAOK1 TAOK2 TAOK3 MAPK9 TLK1 HIPK2 TLK2 GSK3A CDK2 CDK3 CDK4 CDK5 STK36 CDK7 CLK1 MAK CLK4 PAK3 HG-5-88-01 http://dsigdb.tanlab.org/DSigDBv1.0/displayDrug.py?db=d2_lincs&id=953 MYO3A PTK2 PTK6 EPHA7 EGFR PLK4 EPHA1 INSR INSRR ABL1 FLT3 AXL ADCK4 ADCK3 ROS1 TTK MKNK2 SLC12A7 SRMS GAK MAPK8 CHEK2 PHKG2 PHKG1 IGF1R ERBB4 TNK2 FRK FER FES SLK LTK STK32B TNK1 ALK RPS6KA6 MYLK PTK2B CAMKK2 STK33 CLK1 CLK2 CLK3 CLK4 LCK GSK2126458 http://dsigdb.tanlab.org/DSigDBv1.0/displayDrug.py?db=d2_lincs&id=250 CDK19 PI4KB PIK3CA PIK3CB JAK1 STK16 PIK3CD TTK PIK3C2B AAK1 GAK IRAK3 MAP2K4 MTOR PIK3C2G MAPKAPK5 PIK3CG PIP4K2C BX-912 http://dsigdb.tanlab.org/DSigDBv1.0/displayDrug.py?db=d2_lincs&id=433 MUSK STK10 STK11 PRPF4B PLK4 HIPK3 HIPK2 HIPK1 INSRR IKBKE TYK2 AXL NIM1K MAP3K9 CAMK1 STK17B GRK4 MAP3K7 FGR CSNK2A2 SRPK2 TAOK2 DMPK DYRK1A IRAK3 STK17A IRAK4 PIP4K2B PLK2 RPS6KB1 STK16 JAK1 STK3 STK4 ANKK1 FGFR4 FGFR2 FGFR3 CSNK2A1 FGFR1 IKBKB BRSK2 BRSK1 SYK DAPK3 PTK2B KIT BMPR2 PAK4 PAK6 PAK7 PAK3 ICK NUAK1 NUAK2 HIPK4 MYLK NEK6 NEK7 NEK4 ABL2 NEK2 NEK3 LRRK2 NEK9 TTK STK26 STK24 JAK2 JAK3 PRKG2 PRKACA BMX PHKG2 PHKG1 CHEK1 EPHB6 CAMK1D CDK7 CHUK BLK SBK3 SBK1 RPS6KA1 RPS6KA2 RPS6KA3 RPS6KA4 SIK3 RPS6KA6 MAP3K2 CAMKK1 STK33 MAP3K3 CLK1 CLK2 TIE1 LCK BTK PDGFRB PDGFRA MKNK2 CDKL1 RET NTRK1 MAPK15 TNIK DYRK2 MAPK10 NTRK2 MAPK13 ABL1 FLT4 NTRK3 FLT3 FLT1 TEK SIK1 TBK1 SIK2 CDKL5 CSF1R BMP2K CDKL2 MARK4 MAPK6 MARK1 MAPK4 MARK3 MAPK8 MAPK9 KDR ACVR2A ACVR2B MARK2 MYLK4 MYLK2 TNK1 MERTK SRPK1 TAOK1 SRPK3 TAOK3 RIOK3 RIOK1 ITK LATS2 PIP5K1A EIF2AK4 MET CDK4 PIP4K2C PRKACB PRKD1 PRKD2 PRKD3 MAP4K1 MAP4K3 MAP4K2 MAP4K5 MAP4K4 SRC CIT EGFR PRKAA2 PRKAA1 MAP2K2 MAP2K1 RIPK4 MAP2K5 MAP2K4 PRKX MINK1 ALK CAMKK2 CDK13 VRK2 FYN IRAK1 PDPK1 GAK ZAP70 AURKB AURKC PTK2 DAPK1 ULK2 ULK3 ULK1 BMPR1B PKN1 PKN2 PRKCE PRKCD AAK1 NEK5 SLK PRKCQ AURKA ZAK MELK ROCK1 ROCK2 MAP3K10 MAP3K11 MAP3K13 MAP3K19 AZD7762 http://dsigdb.tanlab.org/DSigDBv1.0/displayDrug.py?db=d2_lincs&id=471 TSSK1B STK10 STK11 PRPF4B PLK4 HIPK3 AKT1 HIPK1 IKBKE TYK2 ROS1 AXL MAP3K9 CAMK1 FGFR2 GRK4 MAP3K7 FGR GRK1 EPHA7 SLC12A7 CSNK1E PTK6 MAP3K3 DMPK DYRK1A IRAK3 LYN DYRK1B IRAK4 PIP4K2B ERBB2 EPHA4 ERBB4 CSF1R CAMK2D JAK1 CAMK2A CSNK1G2 CSNK1G3 CSNK1G1 STK4 EPHA1 ANKK1 FGFR4 STK17B CSNK2A2 CSNK2A1 STK17A PTK2B IKBKB JAK2 BRSK2 BRSK1 HIPK2 SYK MST1R MYLK KIT BMPR2 DAPK1 PAK4 PAK6 PAK7 STK38L PAK3 MYO3A PRKCI MYO3B PRKCH DSTYK NUAK1 FGFR1 DCLK1 DCLK2 MAPKAPK5 MAPKAPK2 ABL2 CSK LRRK2 TTK STK26 STK25 STK24 PRKG1 JAK3 PRKG2 BMX PDPK1 CHEK2 PHKG2 PHKG1 CHEK1 EPHB2 EPHB1 EPHB4 CAMK1D CDK7 CHUK SRMS BLK HCK SBK1 TYRO3 RPS6KA1 RPS6KA2 RPS6KA3 RPS6KA4 CSNK1A1 RPS6KA6 TLK2 DDR2 DDR1 PAK1 CAMKK2 CAMKK1 STK33 STK35 GRK7 STK38 CLK1 CLK2 TIE1 CLK4 LCK BTK PDGFRB PDGFRA EPHA8 MKNK2 EPHA6 EPHA5 MKNK1 EPHA3 EPHA2 RET NTRK1 TNIK PTK2 NTRK2 OXSR1 SBK3 ABL1 ACVR1 FLT4 NTRK3 FLT3 FLT1 SIK1 SIK3 SIK2 TEC RPS6KB1 CSNK1D MAP3K2 MARK4 TBK1 BMP2K MARK2 MARK3 NUAK2 KDR MARK1 ACVR2A ACVR2B TNK2 FRK STK39 TNK1 MAST1 FER FES MERTK LTK TLK1 SRPK1 TAOK1 SRPK3 TAOK3 RIOK3 CSNK1A1L RIOK1 ITK LATS2 MAP2K6 SNRK EIF2AK2 EIF2AK4 MET SRPK2 PRKACA PRKACB STK32B PRKD1 PRKD2 PRKD3 MAP4K1 MAP4K3 MAP4K2 MAP4K5 MAP4K4 CAMK1G TGFBR2 CIT EGFR PRKAA2 PRKAA1 MAP2K3 MAP2K2 MAP2K1 RIPK4 MAP2K5 MAP2K4 STK32A PRKX YES1 MINK1 TXK ALK FYN IRAK1 MAP3K13 GAK ZAP70 AURKB AURKC DAPK3 DAPK2 PIP5K1A ULK2 ULK3 ULK1 PIM3 BMPR1B PKN1 PRKCE PRKCD SRC AAK1 SLK PRKCQ NIM1K LATS1 RPS6KA5 TESK1 TNNI3K MELK ROCK1 ROCK2 MAP3K10 MAP3K11 MAP3K12 STK3 MAP3K19 XMD8-85 http://dsigdb.tanlab.org/DSigDBv1.0/displayDrug.py?db=d2_lincs&id=826 PTK6 PLK1 NUAK1 NUAK2 DCLK1 PLK4 DCLK2 ABL1 ROS1 MKNK2 GAK MAPK7 ULK2 ULK1 FRK TNK1 FGFR4 SBK1 TAOK1 TAOK3 TNK2 RPS6KA2 RPS6KA6 MYLK CAMKK2 STK33 PRKD1 PRKD2 PRKD3 GW-5074 http://dsigdb.tanlab.org/DSigDBv1.0/displayDrug.py?db=d2_lincs&id=649 MYO3A PDGFRB MYO3B MAP4K4 TNIK MAP2K4 HIPK3 HIPK2 BMPR1B CIT TYK2 RAF1 FLT3 PI4KB JAK3 MINK1 HIPK1 LRRK2 BMP2K GAK MAPK7 AURKB JAK1 DAPK3 DAPK2 DAPK1 PIP4K2B ULK3 TGFBR1 PIM2 PIM3 PIM1 MYLK4 PIK3C2B AAK1 STK3 ANKK1 CSNK2A2 SRPK3 STK17A RPS6KA1 RIOK1 RPS6KA6 CHEK2 MYLK KIT CAMKK2 CAMKK1 HUNK BRAF STK36 MAP3K19 CLK2 CSNK2A1 Crizotinib http://dsigdb.tanlab.org/DSigDBv1.0/displayDrug.py?db=d2_lincs&id=219 MUSK STK10 PLK4 IKBKB PTK2B INSRR HIPK4 TYK2 ROS1 AXL MAP3K2 MAP3K3 GRK4 MAP3K1 MAP3K7 FGR NTRK3 EPHA7 TAOK2 DMPK IRAK3 LYN IRAK1 PIP4K2B IGF1R RPS6KB1 STK3 STK4 ANKK1 TESK1 SYK MST1R KIT PAK3 ACVR1B DSTYK NUAK1 NUAK2 DCLK1 DCLK2 NEK7 NEK9 STK26 JAK2 JAK3 JAK1 EPHB1 EPHB6 EPHB4 CDK11A CDK11B BLK SBK3 SBK1 TYRO3 TNK2 TNK1 DDR2 DDR1 CAMKK2 STK35 TIE1 LCK EPHA8 MKNK2 EPHA6 EPHA5 EPHA4 EPHA3 EPHA2 EPHA1 NTRK1 DYRK2 NTRK2 ABL1 ACVR1 ABL2 FLT3 TEK TBK1 SIK2 CSF1R BMP2K CASK CDKL2 MAPK7 MARK3 SRC TGFBR1 TAOK1 FRK FER FES MERTK LTK TNNI3K SRPK3 TAOK3 RIOK3 RIOK1 ALK PIP5K1A BMPR1B MET CDK7 PRKD1 PRKD2 PRKD3 MAP4K1 MAP4K3 MAP4K2 MAP4K5 LIMK2 LIMK1 PRKAA1 RIPK1 INSR RIPK2 RIPK4 TXK ADCK4 FYN AURKA AURKB AURKC PTK2 ULK2 ULK3 ULK1 SLK NIM1K ROCK1 ROCK2 MAP3K12 MAP3K13 MAP3K19 WH-4-023 http://dsigdb.tanlab.org/DSigDBv1.0/displayDrug.py?db=d2_lincs&id=83 STK10 STK16 PTK2B HIPK4 ROS1 MAP3K9 MAP3K2 MAP3K3 GRK4 FGR FGFR3 SRMS TAOK2 DMPK LYN PIP4K2B ERBB2 ERBB3 ERBB4 PIK3C2B RET FGFR4 FGFR2 TESK1 FGFR1 SYK KIT HUNK PAK1 PAK3 ACVR1B NUAK2 ACVRL1 EPHB4 CDC42BPG JAK3 CDC42BPB PRKACA BMX PHKG1 EPHB2 EPHB3 EPHB1 EPHB6 CSK BLK HCK TNK2 TNK1 DDR2 DDR1 STK36 TIE1 LCK BTK PDGFRB PDGFRA EPHA8 EPHA6 EPHA5 EPHA4 EPHA3 EPHA2 EPHA1 MAPK11 ABL1 ACVR1 ABL2 FLT3 FLT1 TEK SIK1 SIK2 TEC CSF1R BMP2K CDKL3 CDKL2 MARK3 MAPK9 KDR ACVR2A TGFBR1 STK32B FRK MYLK2 STK32A PRKAA2 FER FES LTK TAOK1 SRPK3 TAOK3 RIOK3 RIOK1 ALK PIP5K1A MET CDK4 PRKACB PRKD1 PRKD2 PRKD3 MAP4K1 MAP4K3 MAP4K2 MAP4K5 MAP4K4 PTK6 LIMK2 LIMK1 EGFR ACVR2B BMPR1A BMPR1B RIPK2 MAP2K5 CIT YES1 MINK1 TXK FYN GAK AURKA AURKC PKN1 PRKCD SRC AAK1 SLK TNNI3K NLK MAP3K11 MAP3K19 GW843682 http://dsigdb.tanlab.org/DSigDBv1.0/displayDrug.py?db=d2_lincs&id=1185 PDGFRB MAP4K5 PLK1 PLK3 PLK2 RET MAP2K5 HIPK4 FLT4 FLT3 NEK2 MAP3K1 BMP2K GAK STK10 DAPK1 PIP4K2B EPHB6 STK3 MERTK SLK SRPK1 RIOK3 RIOK1 PIP5K1C PIP5K1A ROCK1 KIT MET NUAK2 Bosutinib http://dsigdb.tanlab.org/DSigDBv1.0/displayDrug.py?db=d2_lincs&id=540 MAP4K3 MAP4K2 MAP4K5 MAP4K4 MAP2K1 EPHA8 STK10 CIT EGFR EPHA2 RET BMP2K MAP2K2 TNIK MAP3K11 FGR MAP2K5 MAPK6 ABL1 ABL2 AXL CAMK1D MINK1 MAP3K9 NEK2 CSK SIK3 SIK2 MAP3K2 MAP3K3 GRK4 CSF1R MAP3K7 MAP3K4 STK26 CSNK1D CSNK1E JAK2 YES1 DMPK STK25 WEE2 LYN NUAK2 PIP4K2B ERBB2 ERBB3 MAPK4 ERBB4 VRK2 FRK EPHA3 MYLK2 PRKCD SRC AAK1 STK3 STK24 BLK SLK HCK GAK WEE1 SRPK3 RIOK3 STK32A RIOK1 CSNK1A1 SYK EIF2AK4 LCK EIF2AK1 BMPR2 STK35 MAP3K19 PAK1 BTK FES BMS-536924_KIN001-126 http://dsigdb.tanlab.org/DSigDBv1.0/displayDrug.py?db=d2_lincs&id=808 STK11 STK16 PLK4 PTK2B INSRR IKBKE TYK2 ROS1 AXL MAP3K9 CAMK1 MAP3K3 NTRK1 FGR NTRK3 FGFR2 SLC12A7 CDC42BPG JAK2 LYN STK17A PIP4K2B IGF1R PRKG2 STK3 STK4 ANKK1 FGFR4 STK17B FGFR3 CSNK2A1 FGFR1 SYK MYLK KIT BMPR2 PAK4 PAK6 PAK7 PAK3 JAK3 NUAK1 NUAK2 DCLK3 NEK6 NEK7 NEK9 STK26 SRMS PRKG1 CDC42BPA CDC42BPB JAK1 PHKG2 PHKG1 ACVRL1 CSK STK24 BLK HCK TNK2 TNK1 RPS6KA6 DDR1 MELK STK33 STK35 CLK1 CLK2 TIE1 CLK4 LCK BTK PDGFRB EPHA8 EPHA7 EPHA5 EPHA3 RET MAP3K7 TNIK PTK2 NTRK2 SBK3 ABL1 ACVR1 FLT4 ABL2 FLT3 FLT1 TEC CSF1R BMP2K MARK1 MARK2 MARK3 SRC RPS6KA1 FRK FER MERTK IRAK3 LTK SRPK1 SRPK3 RIOK3 RIOK1 ITK PIP5K1A EIF2AK4 MET MAP4K1 MAP4K3 MAP4K2 MAP4K5 MAP4K4 EGFR PRKAA2 PRKAA1 MAP2K3 MAP2K2 MAP2K1 YES1 MINK1 TXK ALK FYN GAK AURKB AURKC DAPK3 DAPK2 DAPK1 ULK2 ULK3 PKN1 AAK1 SLK INSR MAP3K10 MAP3K11 MAP3K12 A443654 http://dsigdb.tanlab.org/DSigDBv1.0/displayDrug.py?db=d2_lincs&id=1183 AKT1 AKT2 AKT3 AXL MAP3K7 SLC12A7 CSNK1E DMPK DYRK1B PIP4K2B CAMK2D CAMK2G CAMK2A CAMK2B CSNK1G2 CSNK1G3 STK3 CSNK2A2 STK17A GSK3A HIPK1 KIT PAK4 PAK1 PAK2 NUAK2 DCLK3 MYLK GSK3B CDC42BPG PRKG1 CDC42BPA CDC42BPB PRKG2 PHKG1 CDK7 CHUK CSNK1D RPS6KA4 RPS6KA5 CAMKK2 CAMKK1 STK33 CLK1 CLK2 CLK3 CLK4 MKNK2 RET MAPK15 TNIK MAPK12 MAPK13 FLT3 CAMK1D BMP2K CDKL2 MARK2 MARK3 MYLK4 TAOK1 SRPK3 TAOK3 RIOK2 RIOK3 CSNK1A1L RIOK1 PIP5K1A PRKACA PRKACB CDK8 CDK9 PRKD1 PRKD2 PRKD3 MAP4K3 MAP4K2 MAP4K4 MAP2K3 LATS2 LATS1 CIT PRKX MINK1 CDK19 MELK CDK14 GAK DAPK3 DAPK2 DAPK1 ULK2 PRKCH PIM2 PIM3 PIM1 PKN1 PKN2 PRKCE PRKCD AAK1 PRKCQ ROCK2 CSNK1G1 BEZ235 http://dsigdb.tanlab.org/DSigDBv1.0/displayDrug.py?db=d2_lincs&id=1055 MAP4K2 PIK3CA PIK3CD PIK3C2B PIK3C2G FLT3 NVP-TAE684 http://dsigdb.tanlab.org/DSigDBv1.0/displayDrug.py?db=d2_lincs&id=589 MUSK TSSK1B PLK1 FYN STK10 STK16 PLK4 ADCK3 PTK2B INSRR TYK2 ROS1 AXL MAP3K9 CAMK1 MAP3K3 MAP3K7 FGR TAOK1 EPHA7 SLC12A7 PTK6 DMPK IRAK3 LYN FGFR1 PLK3 PIP4K2B ERBB2 IGF1R ERBB4 CAMK2D CAMK2G CAMK2A CAMK2B STK3 STK4 EPHA1 FGFR4 FGFR2 FGFR3 STK17A JAK2 BRSK2 BRSK1 SYK MST1R MYLK KIT PAK4 PAK6 PAK7 STK38L PAK3 MYO3A MYO3B ACVR1B MAP4K4 NUAK1 NUAK2 DCLK1 PRKG2 DCLK3 DCLK2 ACVRL1 NEK6 NEK7 NEK2 NEK9 TTK SRMS PRKG1 JAK3 JAK1 BMX CHEK2 PHKG2 PHKG1 CHEK1 EPHB1 CSK CDK7 BLK HCK STK32C RPS6KA1 RPS6KA2 RPS6KA3 RPS6KA4 RPS6KA6 DDR2 DDR1 PAK1 CAMKK2 CAMKK1 STK33 STK36 CLK1 CLK2 CLK3 CLK4 LCK BTK PDGFRB PDGFRA MKNK2 EPHA6 RET NTRK1 MAPK15 TNIK PTK2 MAPK10 MAP3K4 SBK3 ABL1 ACVR1 FLT4 ABL2 FLT3 FLT1 TEK SIK1 SIK2 TEC CSF1R BMP2K MARK4 MAPK3 MAPK1 MAPK7 MARK2 MARK3 MAPK8 MAPK9 KDR MARK1 ACVR2A TGFBR1 TNK2 FRK TNK1 FER PRKAA1 MERTK LTK SRPK1 TNNI3K SRPK3 TAOK3 RIOK2 RIOK3 RIOK1 ITK BMPR1A PIP5K1A EIF2AK4 MET SRPK2 PRKACA CDK5 PRKACB STK32B PRKD1 PRKD2 PRKD3 MAP4K1 MAP4K3 MAP4K2 MAP4K5 CAMK1D TGFBR2 LIMK2 LIMK1 EGFR PRKAA2 INSR MAP2K3 MAP2K2 MAP2K1 MAP2K4 NTRK2 YES1 TXK ALK ADCK4 CDK16 CDK17 GAK ZAP70 AURKB AURKC DAPK3 DAPK2 DAPK1 ULK2 ULK3 ULK1 BMPR1B PKN1 PKN2 SRC AAK1 SLK PRKCQ AURKA TIE1 MELK ROCK2 MAP3K10 MAP3K12 FES XMD14-99 http://dsigdb.tanlab.org/DSigDBv1.0/displayDrug.py?db=d2_lincs&id=335 DCLK1 DCLK3 DCLK2 ROS1 CAMK1 MAPK7 TRPM6 ICK EPHB3 CDK11A CDK11B SLK LTK TAOK2 TAOK3 RPS6KA2 ALK CAMKK2 CAMKK1 CDK4 CDK7 CLK2 CLK3 PLX-4720 http://dsigdb.tanlab.org/DSigDBv1.0/displayDrug.py?db=d2_lincs&id=1146 PDGFRB PDGFRA PTK6 FYN MAP2K1 MAP2K2 BMPR1B RIPK2 MAP2K5 MAP2K4 ABL1 RAF1 NEK11 CDK19 SIK1 CAMK1 CSF1R FGR FLT3 SRMS TGFBR2 SRC EPHB6 CSK MYLK4 BLK SLK TESK1 CSNK2A2 ALK RIOK2 TNK2 ZAK DDR2 DDR1 EIF2AK4 KIT BRAF CDK8 CLK2 PAK1 LCK PD0332991 http://dsigdb.tanlab.org/DSigDBv1.0/displayDrug.py?db=d2_lincs&id=617 TSSK1B MAP3K19 CAMK1D DAPK1 PLK1 NUAK2 PLK2 STK16 PLK4 DCLK3 DCLK2 HIPK3 HIPK2 HIPK1 DYRK2 MAPK10 CDK14 SLK HIPK4 ABL1 CDK17 MAPK7 CDKL2 FLT3 MINK1 DSTYK CDKL5 GRK7 PIK3CB CDK16 MAP3K7 NTRK2 PIK3CG IRAK1 JAK2 EIF2AK4 MARK3 DYRK1A GAK MAPK8 DYRK1B DAPK3 PHKG2 PIP4K2C JAK3 ULK2 ULK1 MAP3K3 TAOK1 CAMK2D DCLK1 MAP3K15 CAMK2G CIT CAMK2A CAMK2B MAST1 AAK1 CDK7 RET STK39 CSNK2A2 CSNK2A1 TAOK3 RPS6KA1 RPS6KA2 MAPK9 RPS6KA4 RPS6KA5 MAPK15 DAPK2 MYLK PRKD1 MAP2K2 CDK4 PRKD2 PIK3CA CLK1 CLK2 CLK4 NTRK1 BTK PRKD3 Canertinib http://dsigdb.tanlab.org/DSigDBv1.0/displayDrug.py?db=d2_lincs&id=49 ERBB2 GAK EGFR BLK ERBB4 KU63794 http://dsigdb.tanlab.org/DSigDBv1.0/displayDrug.py?db=d2_lincs&id=768 MTOR PIK3CA PIK3CD AZD4547 http://dsigdb.tanlab.org/DSigDBv1.0/displayDrug.py?db=d2_lincs&id=349 MUSK TSSK1B FYN STK10 STK16 PLK4 INSRR TYK2 AXL MAP3K9 MAP3K2 MAP3K3 MAP3K7 NTRK2 NTRK3 STK17A AURKA IGF1R WNK3 WNK1 CAMK2A CAMK2B STK3 STK4 FGFR4 FGFR2 FGFR3 FGFR1 ZAK MYLK KIT PAK7 NUAK1 NUAK2 DCLK1 DCLK3 DCLK2 NEK2 STK26 STK25 STK24 JAK2 JAK3 PHKG2 PHKG1 CHEK1 EPHB6 CAMK1D BLK HCK TNK2 TNK1 RPS6KA3 DDR2 DDR1 CAMKK2 CAMKK1 STK33 STK35 CLK1 CLK2 TIE1 CLK4 LCK PDGFRB PDGFRA RET NTRK1 TNIK FGR ABL1 FLT4 ABL2 FLT3 FLT1 TEK SIK1 TBK1 SIK2 CSF1R BMP2K CDKL2 MARK4 MARK1 MARK2 MARK3 KDR SRC FRK MYLK2 FES MERTK SRPK1 TAOK1 TAOK3 RIOK1 ALK EIF2AK1 EIF2AK4 CDK4 CDK7 MAP4K3 MAP4K2 MAP4K5 MAP4K4 TGFBR2 PRKAA2 RIPK1 MAP2K2 INSR RIPK2 MAP2K5 MINK1 CDK18 MELK CDK16 ZAP70 AURKB AURKC DAPK3 ULK2 ULK1 BMPR1B AAK1 SLK MAP3K10 MAP3K11 MAP3K19 Lapatinib http://dsigdb.tanlab.org/DSigDBv1.0/displayDrug.py?db=d2_lincs&id=643 ERBB2 ERBB4 STK10 EGFR RIPK2 MAP2K5 RAF1 WZ4002 http://dsigdb.tanlab.org/DSigDBv1.0/displayDrug.py?db=d2_lincs&id=144 PDGFRB PTK2 MKNK2 NUAK1 NUAK2 DCLK1 PLK4 DCLK3 DCLK2 RIPK1 MAPK10 INSRR FLT3 JAK3 NEK7 ALK TEC CSF1R ROS1 TTK GAK MARK1 AURKC BMX STK17A CHEK2 PHKG2 PHKG1 MAPK7 ERBB2 ULK3 IGF1R ULK1 ULK2 ERBB4 EGFR MARK3 AAK1 FER FES BLK LTK NEK6 SRPK3 FGFR1 RIOK2 RPS6KA1 TNK1 ITK DAPK3 PIP5K1A CAMKK2 EIF2AK4 KIT MELK STK33 BTK CLK1 CHEK1 CLK4 PRKD1 PRKD2 PRKD3 KIN001-111_A770041 http://dsigdb.tanlab.org/DSigDBv1.0/displayDrug.py?db=d2_lincs&id=538 FYN STK10 TYK2 AXL FGR SLC12A7 STK24 LYN ERBB2 ERBB4 STK4 TESK1 ZAK BMX KIT MAPK1 PAK7 STK38L PAK3 MYO3A MYO3B DCLK3 NEK2 CDC42BPG CIT CDC42BPA CDC42BPB NLK CHEK2 CSK SRMS BLK HCK TNK2 TNK1 STK35 STK36 TIE1 LCK BTK PDGFRB PDGFRA EPHA8 EPHA1 TNIK MAP3K4 ABL1 ABL2 RAF1 TEK SIK1 TEC CSF1R CSNK1D CSNK1E MAPK7 SRC RPS6KA1 FRK RPS6KA2 FER FES MERTK TNNI3K LATS2 MET CDK8 MAP4K1 MAP4K3 MAP4K5 PTK6 LIMK2 LIMK1 EGFR PRKAA2 PRKAA1 MAP2K2 MAP2K1 RIPK2 MAP2K4 YES1 CDK19 TXK CDK16 AURKA AURKB AURKC ULK2 ULK1 SLK ROCK2 MAP3K12 BRAF Torin2 http://dsigdb.tanlab.org/DSigDBv1.0/displayDrug.py?db=d2_lincs&id=662 PI4KB CLK2 CSF1R MKNK2 PIK3CA PIK3CB PIK3CD PIK3CG CSNK1E PIK3C2G JAK1 MTOR CLK1 TYK2 FLT3 QL-X-138 http://dsigdb.tanlab.org/DSigDBv1.0/displayDrug.py?db=d2_lincs&id=1152 PDGFRB MAP4K2 PI4KB MKNK2 NUAK1 CLK1 EGFR PIK3C2G MAP2K3 BMPR1B DYRK2 MAPK10 MAP2K5 MAP2K4 FLT3 TXK LRRK2 CDKL5 PIK3CA TEC MAP3K7 PIK3CG CSNK2A1 DYRK1A IRAK3 BMX DYRK1B PIP4K2C JAK3 MTOR BLK MAP3K19 MAPK8 CSNK2A2 RIOK2 MAPK9 ZAK GSK3A KIT CDK7 MAP2K7 CLK2 CLK4 BTK SigmaA6730 http://dsigdb.tanlab.org/DSigDBv1.0/displayDrug.py?db=d2_lincs&id=137 PIK3CB CSNK1E NU7441 http://dsigdb.tanlab.org/DSigDBv1.0/displayDrug.py?db=d2_lincs&id=445 PIK3CA PIK3CB PIK3CD PIK3CG Torin1 http://dsigdb.tanlab.org/DSigDBv1.0/displayDrug.py?db=d2_lincs&id=59 MAP4K3 PTK2 MAP4K5 MAP4K4 LIMK2 LIMK1 RIPK1 INSR HIPK4 FLT3 NEK5 PIK3CA ADCK4 PIK3CG TTK CSNK1D CDC42BPG MAPK6 CDC42BPA CDC42BPB MTOR CDK19 STK4 CSNK2A2 TNK1 KIT CDK2 CDK8 PIK3C2G SB590885 http://dsigdb.tanlab.org/DSigDBv1.0/displayDrug.py?db=d2_lincs&id=999 RIOK2 MINK1 ERBB3 CSNK1D STK10 SLK ADCK3 PRKD1 CSNK1E HIPK1 RIPK2 MAPK10 BRAF CIT ABL1 TNIK MAPK9 RAF1 JAK1 WYE-125132 http://dsigdb.tanlab.org/DSigDBv1.0/displayDrug.py?db=d2_lincs&id=517 MTOR PIK3CA PIK3CD DAPK1 PD0325901 http://dsigdb.tanlab.org/DSigDBv1.0/displayDrug.py?db=d2_lincs&id=690 MAP2K2 MAP2K1 MAPK13 PHA-793887 http://dsigdb.tanlab.org/DSigDBv1.0/displayDrug.py?db=d2_lincs&id=25 ICK CDK16 DCLK1 DCLK3 DCLK2 MAP2K3 MAPK15 CDK14 GRK1 CDK18 STK26 CDKL5 GRK7 CDKL1 CDK17 CDKL3 CDKL2 MAPK3 STK25 CDK3 MAPK7 DYRK1A DYRK1B PHKG2 PHKG1 PAK1 ULK2 ULK1 CLK2 CLK3 PRKCE CDK15 CDK9 PRKCQ TAOK1 TAOK3 STK32B RPS6KA3 PAK6 RPS6KA6 GSK3A GSK3B CDK2 STK33 CDK4 CDK5 CDK7 PAK4 CLK1 MAK PAK7 CLK4 PRKD1 PRKD2 PRKD3 Dabrafenib http://dsigdb.tanlab.org/DSigDBv1.0/displayDrug.py?db=d2_lincs&id=667 FYN STK10 STK16 PLK4 ADCK3 HIPK3 HIPK2 HIPK1 HIPK4 TYK2 AXL MAP3K9 CAMK1 NTRK2 SLC12A7 LYN DYRK1B ERBB2 ERBB3 PIK3C2B TESK1 ZAK BRSK2 BRSK1 KIT BMPR2 PAK4 PAK7 PAK3 ACVR1B DCLK1 DCLK3 DCLK2 EPHB6 NEK11 NEK6 NEK7 NEK2 NEK1 NEK9 STK25 SRMS JAK2 JAK3 JAK1 NLK BUB1 CSK BLK HCK RPS6KA1 TNK1 DDR1 MELK STK36 CLK3 LCK BTK PDGFRB PI4KB MKNK2 CSF1R EPHA3 EPHA1 TNIK MAPK10 FGR ABL1 ABL2 RAF1 TEK SIK1 CDKL5 PTK6 RPS6KB1 CDKL2 MAPK8 TGFBR2 TGFBR1 FRK TAOK2 ITK EIF2AK1 EIF2AK4 MET CDK2 CDK3 CDK4 CDK5 CDK7 CDK8 PRKD1 PRKD2 PRKD3 ACVR1 CAMK1D SRC LIMK2 LIMK1 EGFR PRKAA2 PRKAA1 BMPR1B RIPK2 MAP2K5 CIT YES1 CDK18 CDK19 MAP2K4 CDK13 ADCK4 CDK16 CDK17 CDK14 CDK15 GAK AURKB ULK2 ULK3 ULK1 TIE1 MAP3K10 MAP3K11 BRAF Momelotinib http://dsigdb.tanlab.org/DSigDBv1.0/displayDrug.py?db=d2_lincs&id=348 MAP4K1 PDGFRB ACVR1 TYK2 MKNK2 PLK3 IKBKE PRPF4B PLK4 DCLK3 EIF2AK4 IKBKB MAPK15 BMPR1B MAPK10 HIPK4 ABL1 MAPKAPK5 NEK9 FLT3 NEK6 NEK7 HIPK1 NEK5 NEK3 TBK1 SIK2 STK17B GRK4 BMP2K PIK3CG CIT AURKA JAK1 GAK MAPK8 IRAK1 DAPK3 NUAK2 DAPK1 JAK3 ULK3 BUB1 STK16 MYLK4 CHUK CAMK2B AAK1 RIOK1 CLK1 SRPK1 CSNK2A2 STK17A RIOK3 JAK2 RPS6KA5 SGK1 HIPK2 ROCK1 ROCK2 CDK4 CDK7 MAP3K19 CLK2 CLK4 JNK-IN-5A http://dsigdb.tanlab.org/DSigDBv1.0/displayDrug.py?db=d2_lincs&id=464 MAPK9 MAPK10 XMD13-2 http://dsigdb.tanlab.org/DSigDBv1.0/displayDrug.py?db=d2_lincs&id=908 STK16 PLK4 RIPK1 MAPK15 MAPK11 MAP2K5 MAPK13 ABL1 FLT3 GRK4 CDK16 BMP2K CDKL2 AURKC PIP4K2B ICK ULK3 EPHB6 RIOK3 MYLK2 AAK1 ANKK1 TAOK1 SRPK3 MAPK14 RIOK1 PIP5K1C KIT CDK2 CDK3 MAP3K19 MLN8054 http://dsigdb.tanlab.org/DSigDBv1.0/displayDrug.py?db=d2_lincs&id=775 BLK EPHA7 EPHA6 STK10 EPHA4 EPHA3 EPHA2 EPHA1 HIPK1 ABL1 AXL FLT1 STK17B TEK SIK1 EPHB4 PIK3CA TEC FGR CSNK2A2 AURKA AURKB IRAK3 STK17A EPHA5 SRC EPHB1 CSK PLK4 MERTK HCK FGFR2 FGFR3 FGFR1 CLK3 DDR2 DDR1 YES1 CLK2 TIE1 LCK AZD5438 http://dsigdb.tanlab.org/DSigDBv1.0/displayDrug.py?db=d2_lincs&id=248 STK16 PLK4 HIPK3 HIPK2 HIPK1 HIPK4 TYK2 AXL MAP3K9 MAP3K2 PIK3CA GRK4 MAP3K7 NTRK2 PIK3CG CSNK1D CSNK1E TAOK2 DYRK1A IRAK3 DYRK1B PIP4K2C PIP4K2B CSNK1G2 CSNK1G3 STK3 ANKK1 STK17B CSNK2A2 CSNK2A1 STK17A IKBKB SYK GSK3A MYLK KIT BMPR2 MAK PAK3 DSTYK NUAK1 NUAK2 DCLK3 EPHB6 GSK3B NEK10 NEK7 LRRK2 TTK STK26 STK25 STK24 JAK2 JAK3 JAK1 BUB1 CDK11A CDK11B CHUK TLK1 CSNK1A1 TLK2 DDR2 DDR1 CAMKK2 STK35 STK36 MAP3K3 CLK1 CLK2 CLK3 CLK4 PDGFRB PI4KB CSF1R EPHA3 BMPR1B MAPK15 TNIK DYRK2 MAPK10 MAPK13 ABL1 FLT3 TBK1 CDKL5 CDKL1 BMP2K CDKL3 CDKL2 MAPK7 MARK2 MAPK8 MAPK9 TGFBR2 GSG2 MYLK4 MTOR MERTK TAOK1 SRPK3 TAOK3 RIOK2 RIOK3 CSNK1A1L RIOK1 SGK1 MAP2K6 PIP5K1A EIF2AK2 INSR MET CDK2 CDK3 CDK4 CDK5 CDK7 CDK9 PRKD1 PRKD2 PRKD3 MAP4K3 MAP4K2 ACVR1 MAP4K4 CIT MAP2K3 MAP2K2 MAP2K1 RIPK4 MAP2K5 MAP2K4 MINK1 CDK18 CDK13 CDK16 CDK17 CDK14 CDK15 RIPK1 IRAK1 GAK AURKA AURKB AURKC ICK ULK3 PKN2 PRKCD AAK1 SLK ROCK1 ROCK2 MAP3K11 MAP3K14 MAP3K19 ALW-II-49-7 http://dsigdb.tanlab.org/DSigDBv1.0/displayDrug.py?db=d2_lincs&id=107 PDGFRB PDGFRA EPHA8 EPHA5 EPHA4 EPHA3 EPHA2 MAPK14 ABL1 RAF1 CSF1R NTRK3 LYN EPHB2 EPHB3 EPHB1 EPHB4 FRK TNNI3K ZAK DDR2 DDR1 KIT BRAF LCK OTSSP167 http://dsigdb.tanlab.org/DSigDBv1.0/displayDrug.py?db=d2_lincs&id=265 MUSK PLK1 FYN STK10 PLK2 PLK4 CDK17 HIPK3 AKT1 AKT2 HIPK4 TYK2 ROS1 MAP3K9 MAP3K2 GRK7 MAP3K6 MAP3K7 FGR MAP3K5 EPHA7 SLC12A7 CSNK1E MAP3K3 DMPK DYRK1A JAK2 LYN DYRK1B IRAK4 ERBB3 ULK2 VRK2 CAMK2D PRKG2 CSNK1G2 CSNK1G3 STK4 EPHA1 ANKK1 FGFR2 CSNK2A2 CSNK2A1 ITK PTK2B IKBKB ZAK HIPK2 SYK MYLK GSK3B BMPR2 CAMK2G PAK7 STK38L ICK PRKCH DSTYK NUAK1 NUAK2 DCLK1 DCLK3 BUB1 MAPKAPK5 KIT NEK10 MAPKAPK2 HIPK1 STK26 STK25 CDC42BPG PRKG1 JAK3 CDC42BPB JAK1 HUNK BMX PHKG1 EPHB2 EPHB3 EPHB1 EPHB6 EPHB4 SGK2 CDK7 CDK11A CDK11B CHUK STK24 BLK HCK RPS6KA1 RPS6KA2 RPS6KA3 RPS6KA4 CSNK1A1 RPS6KA6 TLK2 DDR1 CAMKK2 CAMKK1 STK33 STK35 STK36 PIK3CA STK38 CLK1 STK17A CLK4 LCK BTK PDGFRB PDGFRA PI4KB EPHA8 MKNK2 EPHA6 EPHA5 EPHA4 EPHA2 RET NTRK1 MAPK15 TNIK DYRK2 MAPK10 NTRK2 MAPK13 ABL1 ACVR1 FLT4 ABL2 FLT3 FLT1 TEK SIK1 SIK3 CDKL5 TEC CSF1R CSNK1D CDKL3 CDKL2 TBK1 BMP2K MARK3 GRK1 MAPK8 MAPK9 KDR MAPK7 SRC TNK2 FRK MYLK4 MYLK2 TNK1 FER FES MERTK LTK SRPK1 TAOK1 TAOK2 TAOK3 PIK3C2G CSNK1A1L IRAK1 SGK3 ALK SGK1 LATS2 INSR CDK2 CDK3 CDK4 CDK5 PRKACB CDK8 CDK9 STK32B RPS6KB1 PRKD1 PRKD2 MAP4K1 MAP4K3 MAP4K2 MAP4K5 MAP2K5 TGFBR2 SRMS CIT EGFR PRKAA2 PRKAA1 MAP2K3 MAP2K2 MAP2K1 MAP2K7 RIPK4 PIK3CG MAP2K4 YES1 MINK1 CDK18 CDK19 TXK MELK CDK16 ADCK3 CDK14 CDK15 PDPK1 AURKA AURKB NTRK3 PTK2 PRKCI ULK3 ULK1 PIM2 BMPR1B CDKL1 PRKCE PRKCD FGFR1 AAK1 SLK PRKACA LATS1 RPS6KA5 TNNI3K PIK3C2B MAP3K11 MAP3K14 BRAF MAP3K19 CP466722 http://dsigdb.tanlab.org/DSigDBv1.0/displayDrug.py?db=d2_lincs&id=258 STK10 PLK2 STK16 PLK4 HIPK3 HIPK2 HIPK1 HIPK4 TYK2 AXL GRK7 PIK3CB PIK3CD MAP3K7 PIK3CG CSNK1D CSNK1E DYRK1A IRAK3 IRAK1 IRAK4 ERBB3 VRK2 CSNK1G2 PIK3C2B PIK3C2G RET ANKK1 STK17B CSNK2A2 CSNK2A1 STK17A BRSK2 MYLK KIT BMPR2 PAK3 ACVR1B IKBKE NEK6 NEK7 NEK9 JAK1 NLK ACVRL1 EPHB6 BLK HCK RPS6KA1 TNK1 RPS6KA3 RPS6KA4 CSNK1A1 RPS6KA6 CAMKK2 STK33 STK36 PIK3CA CLK1 CLK2 CLK3 CLK4 LCK PDGFRB PI4KB MKNK2 EPHA3 EPHA1 MAPK15 DYRK2 MAPK10 MAPK11 ABL1 FLT4 FLT3 CDKL5 RPS6KB1 BMP2K CDKL3 CDKL2 MAPK8 MAPK9 SRC TGFBR1 MTOR TAOK1 RIOK2 DYRK1B BMPR1A PIP5K1C PIP5K1A EIF2AK4 PIP4K2C CDK7 ZAK ACVR1 TGFBR2 LATS2 BMPR1B RIPK2 RIPK4 MAP2K5 MAP2K4 MELK ADCK4 ADCK3 GAK AURKA AURKB AURKC DAPK3 DAPK2 DAPK1 ULK2 ULK3 ULK1 PIM3 PIM1 AAK1 MAP3K19 GSK461364 http://dsigdb.tanlab.org/DSigDBv1.0/displayDrug.py?db=d2_lincs&id=220 PDGFRB PLK1 STK10 PLK2 CSNK2A2 NEK9 FLT3 JAK3 NEK2 PIK3CB MAP3K1 PIK3CD BMP2K PIK3CG PLK3 SRPK3 DAPK3 DAPK2 DAPK1 PIP4K2B ULK2 CAMK2G PIM3 PIM1 CAMK2D STK39 PKN2 PRKCE CAMK2A PIK3C2B RIOK1 SLK TAOK1 CSNK2A1 RIOK3 RPS6KA2 RPS6KA3 RPS6KA4 RPS6KA6 MAST1 PIP5K1A ROCK1 NUAK2 MAP3K19 PRKD3 (R)-Roscovitine http://dsigdb.tanlab.org/DSigDBv1.0/displayDrug.py?db=d2_lincs&id=939 CSNK1A1L CSNK1A1 CDK7 HIPK1 TTK CSNK1D CSNK1E HIPK4 DYRK1A CLK1 CLK2 DYRK1B CLK4 CGP60474 http://dsigdb.tanlab.org/DSigDBv1.0/displayDrug.py?db=d2_lincs&id=930 ICK MAPK15 CDKL5 CDK16 CDKL3 CDKL2 HIPK2 HIPK1 CDK9 HIPK4 DYRK1A CLK1 CLK2 DYRK1B CLK4 MAK XMD11-50 http://dsigdb.tanlab.org/DSigDBv1.0/displayDrug.py?db=d2_lincs&id=719 RPS6KA1 TNK1 ALK LRRK2 MKNK2 RPS6KA2 DCLK1 MYLK RPS6KA6 DCLK2 PLK1 STK33 AURKA ABL1 PIK3CG PLK4 ROS1 MAPK7 R406 http://dsigdb.tanlab.org/DSigDBv1.0/displayDrug.py?db=d2_lincs&id=822 MUSK TSSK1B PLK1 STK10 STK16 PLK4 CDK17 IKBKB HIPK1 INSRR IKBKE TYK2 ROS1 AXL MAP3K9 CAMK1 STK17B MAP3K7 FGR FGFR3 EPHA7 PTK6 DMPK WEE2 WEE1 DYRK1B PLK3 PIP4K2B IGF1R EPHA4 ERBB4 JAK1 EPHA1 ANKK1 FGFR4 FGFR2 CSNK2A2 CSNK2A1 FGFR1 SYK GSK3A PTK2B KIT PAK4 PAK6 PAK7 PAK1 PAK3 NUAK1 NUAK2 DCLK1 DCLK3 NEK6 NEK7 NEK5 NEK2 NEK1 NEK9 STK25 JAK2 JAK3 PRKG2 BMX PHKG2 CHEK1 EPHB1 CSK CHUK BLK HCK TNK2 TNK1 TLK1 RPS6KA5 TLK2 DDR2 DDR1 MELK STK33 STK35 STK36 MAP3K3 CLK1 STK17A CLK3 CLK4 LCK BTK PDGFRB PDGFRA EPHA8 MKNK2 EPHA6 EPHA5 MKNK1 EPHA3 EPHA2 RET NTRK1 MAPK15 MAPK10 MAP3K4 MAPK12 MAPK13 ABL1 FLT4 ABL2 FLT3 FLT1 MST1R TEK SIK1 SIK2 TEC CSF1R BMP2K MARK4 MARK1 MARK2 MARK3 MAPK8 MAPK9 KDR TGFBR2 TAOK1 RPS6KA1 FRK MYLK4 FER FES MERTK IRAK3 LTK RPS6KA4 SRPK1 LYN SRPK3 RIOK3 RIOK1 ITK PIP5K1A EIF2AK2 EIF2AK4 MET PRKACA PRKACB MAP4K1 MAP4K3 PTK2 CAMK1D SRC LIMK2 LIMK1 EGFR PRKAA2 PRKAA1 MAP2K3 MAP2K1 RIPK2 MAP2K6 CIT NTRK2 YES1 MINK1 MAP2K4 ALK ADCK4 FYN ADCK3 GAK ZAP70 AURKB AURKC NTRK3 DAPK3 DAPK2 DAPK1 ULK2 ULK3 ULK1 PKN1 PKN2 AAK1 SLK AURKA CLK2 TIE1 TNNI3K SBK3 ROCK2 MAP3K10 MAP3K11 PDPK1 TXK XMD8-92 http://dsigdb.tanlab.org/DSigDBv1.0/displayDrug.py?db=d2_lincs&id=661 TNK1 DCLK1 PLK4 DCLK2 MAPK7 ROS1 QL-XI-92 http://dsigdb.tanlab.org/DSigDBv1.0/displayDrug.py?db=d2_lincs&id=201 PDGFRB ZAK EPHA8 FRK DDR1 EPHA3 KIT MAPK14 MAPK11 ABL1 GDC-0941 http://dsigdb.tanlab.org/DSigDBv1.0/displayDrug.py?db=d2_lincs&id=438 PIK3CA PDGFRA PIK3CD PIK3CB PIK3CG HG-14-10-04 http://dsigdb.tanlab.org/DSigDBv1.0/displayDrug.py?db=d2_lincs&id=575 MUSK TSSK1B PLK1 STK10 STK16 PLK4 HIPK3 HIPK2 HIPK1 INSRR SLK HIPK4 TYK2 ROS1 AXL MAP3K9 CAMK1 FGFR2 MYLK MAP3K7 NTRK2 FGFR3 EPHA7 SLC12A7 MAP3K3 DMPK DYRK1A IRAK3 LYN DYRK1B PLK3 IRAK4 PIP4K2B ERBB2 IGF1R ERBB4 CAMK2D CAMK2G CAMK2A CAMK2B EPHA1 FGFR4 STK17B CSNK2A2 CSNK2A1 STK17A SYK PTK2B KIT HUNK PAK4 PAK7 PAK2 PAK3 MYO3A MYO3B DSTYK NUAK1 FGFR1 IKBKE DCLK1 DCLK3 DCLK2 EPHB6 NEK10 NEK6 NEK7 LRRK2 NEK9 TTK SRMS JAK2 JAK3 JAK1 CHEK2 PHKG2 PHKG1 CHEK1 BUB1 CAMK1D BLK HCK SBK1 TNK2 TNK1 RPS6KA3 RPS6KA4 RPS6KA6 DDR1 CAMKK2 CAMKK1 STK33 GRK7 CLK1 CLK2 CLK3 CLK4 LCK PDGFRB PDGFRA MKNK2 MKNK1 RET NTRK1 MAPK15 TNIK DYRK2 MAPK10 OXSR1 NIM1K ABL1 FLT4 ABL2 FLT3 FLT1 TEK SIK1 TBK1 SIK2 PTK6 CSF1R BMP2K MARK4 MAPK7 MARK2 MARK3 MAPK8 MAPK9 NUAK2 KDR MARK1 SRC RPS6KA1 FRK MYLK4 RPS6KA2 MAST1 FER FES MERTK WEE2 LTK SRPK1 SRPK2 RIOK2 RIOK3 CSNK1A1L RIOK1 ITK PIP5K1A EIF2AK4 MET PRKACA STK32B PRKD1 PRKD2 PRKD3 MAP4K3 PTK2 MAP4K4 CAMK1G TGFBR2 CIT EGFR PRKAA2 PRKAA1 MAP2K3 MAP2K2 MAP2K1 MAP2K6 MAP2K5 MAP2K4 STK32A YES1 MINK1 ALK ADCK4 IRAK1 GAK ZAP70 AURKC DAPK3 DAPK2 DAPK1 ULK2 ULK3 ULK1 PIM3 PIM1 AAK1 STK39 AURKA LATS1 TIE1 INSR MELK ROCK1 ROCK2 MAP3K10 MAP3K11 MAP3K12 MAP3K13 MAP3K14 MAP3K19 Sorafenib http://dsigdb.tanlab.org/DSigDBv1.0/displayDrug.py?db=d2_lincs&id=169 MUSK PDGFRB PDGFRA MAP4K5 EPHA8 MKNK2 EPHA6 STK10 MKNK1 EPHA3 RET HIPK3 MAPK15 HIPK1 CDKL3 MAP2K5 HIPK4 ABL1 FLT4 NTRK3 RAF1 FLT3 AXL FLT1 CDK19 CSF1R MAP3K7 NTRK2 CDKL2 TTK AURKB CDK14 FGFR1 KDR EPHB6 FRK TEK MERTK SLK FGFR2 TAOK2 TAOK3 MAPK14 ZAK HIPK2 DDR2 DDR1 KIT MAPK13 BRAF CDK7 CDK8 MAP3K19 TIE1 LCK MAPK11 KIN001-127 http://dsigdb.tanlab.org/DSigDBv1.0/displayDrug.py?db=d2_lincs&id=502 MUSK EPHA6 STK10 DCLK3 INSR INSRR FLT3 YES1 NEK7 MAP3K4 AXL WEE2 TAOK3 PHKG2 SRC IGF1R FER MERTK ITK ALK STK38L STK33 CDK7 CLK1 CLK2 TIE1 LCK BTK BMS345541 http://dsigdb.tanlab.org/DSigDBv1.0/displayDrug.py?db=d2_lincs&id=717 RPS6KA4 CDK13 MYLK4 CDK11A CDK11B IKBKB DYRK2 MAPK7 CDK7 TYK2 BI-2536 http://dsigdb.tanlab.org/DSigDBv1.0/displayDrug.py?db=d2_lincs&id=1004 PTK2 PLK3 STK16 DCLK2 TTK GAK DAPK3 DAPK1 EGFR DCLK1 SLK ALK RPS6KA2 RPS6KA4 RPS6KA5 RPS6KA6 MYLK CAMKK2 CAMKK1 STK33 CLK2 PRKD1 PRKD3 WZ-7043 http://dsigdb.tanlab.org/DSigDBv1.0/displayDrug.py?db=d2_lincs&id=383 TAOK3 TIE1 EPHB6 TAOK1 MAP3K2 MAP3K3 DDR1 CSF1R EIF2AK4 MAP3K4 KIT STK26 STK24 MAPK7 LCK FGFR4 FGFR1 FGFR2 FGFR3 FLT1 KIN001-220 http://dsigdb.tanlab.org/DSigDBv1.0/displayDrug.py?db=d2_lincs&id=780 MUSK PDGFRB SLK ACVR1 CAMK1D ULK3 MKNK2 STK10 STK11 STK16 PLK4 RET BMP2K HIPK3 HIPK2 HIPK1 MAPK10 MAP2K5 HIPK4 ABL1 TYK2 FLT3 AXL FLT1 NEK6 NEK7 NEK5 TXK TBK1 MAP3K11 CAMK1 SRPK1 GRK4 CSF1R MAP3K7 SRPK2 GAK JAK3 AURKB JAK1 IRAK3 MAPK8 STK17A DAPK3 DAPK2 PIP5K1A PIP4K2B ACVR2A LIMK1 EPHB6 BMPR1B RIOK3 EGFR MYLK4 AURKC ADCK4 AAK1 RIOK1 MERTK WEE2 AURKA STK17B CSNK2A2 SRPK3 FGFR1 TNK2 TNK1 MAPK9 ZAK FLT4 EIF2AK2 EIF2AK4 KIT MAP3K10 MET DAPK1 STK36 MAP3K19 CLK2 TIE1 LCK PAK3 AZD-9291 http://dsigdb.tanlab.org/DSigDBv1.0/displayDrug.py?db=d2_lincs&id=674 PDGFRB PTK2 MAP4K4 PTK6 MKNK2 MKNK1 EGFR PLK4 INSR HIPK2 TNIK MYO3B INSRR MAP2K5 HIPK4 ROS1 MINK1 HIPK1 TXK LRRK2 TEC FLT3 PLK1 GAK JAK3 DAPK3 DAPK2 DAPK1 ERBB2 IGF1R EPHB6 ERBB4 CAMK2B AAK1 BLK LTK CSNK2A2 CSNK2A1 TNK2 TNK1 RPS6KA4 ALK MYLK STK33 HUNK PIP4K2C MAP3K19 BTK ZM-447439 http://dsigdb.tanlab.org/DSigDBv1.0/displayDrug.py?db=d2_lincs&id=375 PDGFRB PDGFRA MAP4K5 BLK PTK6 MKNK2 STK10 EGFR PLK4 RET MAP2K2 HIPK1 RIPK2 MAP2K5 HIPK4 ABL1 FLT3 AXL CSK RPS6KB1 CDKL2 SRMS AURKA AURKB LYN ERBB2 ERBB3 EPHB6 ERBB4 CDK11A PIK3C2G MERTK SLK LTK HCK TNK2 ULK3 MST1R MAP2K1 KIT MET CDK7 LCK BTK RO-3306 http://dsigdb.tanlab.org/DSigDBv1.0/displayDrug.py?db=d2_lincs&id=46 MAP4K2 MAP4K4 HIPK4 MYLK HIPK3 MAPK15 DYRK2 CIT PRKX MAPKAPK2 BMP2K PIK3CG IRAK1 GAK CSNK2A1 CDC42BPB DYRK1A DYRK1B DAPK3 PHKG2 FLT3 DMPK PIM1 GSG2 PKN2 PRKCD CSNK1G2 CSNK1G3 AAK1 CLK1 STK17B TAOK1 CSNK2A2 STK17A RIOK1 RPS6KA4 RPS6KA5 SGK1 ROCK1 ROCK2 MELK STK33 BMPR2 CDK7 MAP3K19 CLK2 CLK3 CLK4 JW-7-24-1 http://dsigdb.tanlab.org/DSigDBv1.0/displayDrug.py?db=d2_lincs&id=76 PDGFRB PDGFRA MAP4K4 STK10 LATS2 ABL1 TYK2 FLT3 PIK3CA PIK3CD MAP3K7 PIK3CG CSNK1E GAK NUAK2 SRC PRKCE PRKCD PIK3C2B SLK TAOK1 TAOK3 MAPK15 GSK3A KIT BMPR1A BRAF STK36 CDK7 CLK1 CLK3 LCK JWE-035 http://dsigdb.tanlab.org/DSigDBv1.0/displayDrug.py?db=d2_lincs&id=932 MAP4K3 ULK3 MKNK2 NUAK1 NUAK2 DCLK1 PLK4 RET DCLK2 BMPR1B RIPK2 RIPK4 ABL1 TYK2 ABL2 ROS1 AXL LRRK2 MAP3K2 PIK3CA PIK3CD BMP2K CASK PIK3CG STK26 JAK2 JAK3 YES1 JAK1 GAK PIP4K2C MAPK7 ULK2 SRC ULK1 FLT3 AURKB CDK7 CSF1R STK16 MARK3 PRKAA2 CSNK1G2 CSNK1G3 CSNK1G1 PRKAA1 BLK SLK SBK3 SBK1 TAOK1 TAOK2 TAOK3 TNK1 AURKA AURKC PIP5K1A DDR1 STK3 MAP3K3 DSTYK PRKD3 LCK PAK3 ALW-II-38-3 http://dsigdb.tanlab.org/DSigDBv1.0/displayDrug.py?db=d2_lincs&id=440 PDGFRB PDGFRA EPHA8 CSF1R EPHA4 EPHA3 EPHA2 MAPK14 MAPK11 ABL1 ABL2 RAF1 YES1 TXK FYN LYN EPHB2 SRC EPHB4 FRK BLK HCK ZAK DDR2 DDR1 KIT BRAF LCK AZD-6482 http://dsigdb.tanlab.org/DSigDBv1.0/displayDrug.py?db=d2_lincs&id=773 PIK3CA PIK3CB PIK3CD PIK3CG PIK3C2B PIK3C2G MTOR FLT3 SP600125 http://dsigdb.tanlab.org/DSigDBv1.0/displayDrug.py?db=d2_lincs&id=846 CAMK1D MKNK2 NUAK2 MAP2K4 STK16 PLK4 BMPR1B IKBKB MAP2K2 MAP2K1 MAPK10 MAP2K6 IKBKE MINK1 NEK1 CAMK1 CDK16 BMP2K TTK STK26 CSNK1D STK24 GAK MAPK8 MAPK9 DAPK3 DAPK2 DAPK1 ULK2 ULK3 ULK1 PIM3 RPS6KA1 TNK1 MYLK4 CHUK AAK1 ANKK1 MAP2K3 TAOK1 RIOK3 RPS6KA2 RIOK1 RPS6KA4 RPS6KA5 RPS6KA6 MYLK PHKG2 CAMKK2 BMPR2 CLK2 RIPK4 HG-6-64-01 http://dsigdb.tanlab.org/DSigDBv1.0/displayDrug.py?db=d2_lincs&id=510 MUSK STK10 STK11 PRPF4B IKBKB PTK2B HIPK4 TYK2 AXL MAP3K9 MAP3K2 STK17B GRK4 NTRK1 FGR TESK1 PTK6 TAOK2 WEE2 LYN STK17A PIP4K2B ERBB2 ERBB4 CSF1R STK3 EPHA1 ANKK1 FGFR4 FGFR2 FGFR3 FGFR1 ZAK SYK KIT BMPR2 PAK3 DCLK3 NEK5 CSK LRRK2 NEK9 TTK SRMS JAK2 JAK3 BMX EPHB2 EPHB3 EPHB1 EPHB6 EPHB4 CDK11A CDK11B CHUK BLK HCK TNK2 TNK1 RPS6KA3 RPS6KA6 DDR2 DDR1 STK36 MAP3K3 CLK1 TIE1 LCK BTK PDGFRB PDGFRA EPHA8 MKNK2 EPHA6 EPHA5 EPHA4 EPHA3 EPHA2 RET MAP3K7 MAPK14 TNIK MAPK10 MAPK11 ABL1 FLT4 ABL2 RAF1 FLT3 FLT1 TEK SIK1 TEC RPS6KB1 BMP2K CDKL3 CDKL2 MAPK9 KDR TGFBR2 FRK MYLK2 RPS6KA2 FES MERTK SRPK1 TAOK1 SRPK3 TAOK3 RIOK3 RIOK1 PIP5K1A EIF2AK4 PRKD1 MAP4K1 MAP4K3 MAP4K2 MAP4K5 MAP4K4 SRC LIMK2 LIMK1 EGFR RIPK1 RIPK2 MAP2K7 MAP2K5 CIT NTRK2 YES1 MINK1 CDK19 TXK FYN GAK AURKC NTRK3 ULK3 ULK1 CDC42BPA SLK TNNI3K MAP3K11 BRAF MAP3K19 CG-930 http://dsigdb.tanlab.org/DSigDBv1.0/displayDrug.py?db=d2_lincs&id=764 ERBB3 EPHB6 RPS6KA6 CLK2 EGFR MAPK14 MAPK1 CSNK1E GAK STK36 ABL1 MAPK10 MAPK8 MAPK9 NLK PD173074 http://dsigdb.tanlab.org/DSigDBv1.0/displayDrug.py?db=d2_lincs&id=498 FGFR1 DDR1 CSF1R STK25 STK24 FLT4 TIE1 FGFR2 FGFR3 FLT1 XMD-12 http://dsigdb.tanlab.org/DSigDBv1.0/displayDrug.py?db=d2_lincs&id=1013 MKNK2 DCLK1 PLK4 RET DCLK2 BMPR1B ABL1 TYK2 LRRK2 MAP3K2 MAP3K3 CSF1R FGR PIK3CG JAK2 AURKA AURKB JAK1 MAPK7 ULK2 BLK SBK3 TAOK1 TAOK2 TAOK3 TNK1 WZ3105 http://dsigdb.tanlab.org/DSigDBv1.0/displayDrug.py?db=d2_lincs&id=521 PDGFRB FGR FLT3 MAP3K2 GRK7 NTRK1 NTRK2 CSNK1D CSNK1E JAK2 DMPK IRAK1 IRAK4 ULK2 SRC ULK1 VRK2 CDK7 CSNK1A1L CSNK1G2 CSNK1G3 CLK1 PRKCQ RPS6KA1 RPS6KA2 RPS6KA3 CSNK1A1 RPS6KA6 ROCK2 KIT STK33 MAP3K3 MAP3K19 CLK2 CLK3 CLK4 PHA-767491 http://dsigdb.tanlab.org/DSigDBv1.0/displayDrug.py?db=d2_lincs&id=513 MUSK PLK1 PLK3 HIPK3 HIPK2 HIPK1 HIPK4 TYK2 MAP3K5 CSNK1D CSNK1E DYRK1A JAK2 DYRK1B CAMK2B CSNK1G2 CSNK1G3 CSNK1G1 CSNK2A2 CSNK2A1 STK17A IKBKB GSK3A MYLK GSK3B BMPR2 NUAK2 DCLK3 MAPKAPK5 MAPKAPK2 PRKG1 JAK3 PRKG2 CDK4 CHEK2 PHKG2 BUB1 CHUK RPS6KA2 RPS6KA4 CSNK1A1 CAMKK2 STK33 STK35 STK38 CLK1 CLK2 CLK3 CLK4 MKNK2 MAPK15 TNIK DYRK2 ABL1 FLT3 CDKL5 BMP2K TGFBR2 ACVR2B GSG2 TAOK1 TAOK2 TAOK3 CSNK1A1L IRAK1 SGK1 MET PRKACA CDK7 CDK8 CDK9 PRKD1 PRKD2 PRKD3 MAP4K2 ACVR2A LATS2 BMPR1B RIPK4 CIT PRKX MINK1 CDK19 CDK13 DAPK3 DAPK2 DAPK1 ULK2 PRKCH PIM2 PIM3 PKN1 PKN2 PRKCE PRKCD AAK1 PRKCQ RPS6KA5 ROCK1 ROCK2 MAP3K19 CP724714 http://dsigdb.tanlab.org/DSigDBv1.0/displayDrug.py?db=d2_lincs&id=386 ERBB2 CDK19 ERBB4 MKNK2 STK10 EGFR MAP2K2 MAP2K1 MAP2K5 CDK8 TAK-715 http://dsigdb.tanlab.org/DSigDBv1.0/displayDrug.py?db=d2_lincs&id=352 ACVR1 MAP4K4 ACVR1B EGFR MAPK14 BMPR1B RIPK2 MAPK10 CDC42BPG MAP2K5 CIT ABL1 YES1 MINK1 ADCK4 ADCK3 CSNK1D CSNK1E GAK MAPK8 MAPK9 SRC TGFBR1 ERBB4 CSNK1A1L NLK CSNK1A1 STK32B STK32A ZAK RPS6KA6 DDR1 TNIK KIT HUNK STK36 MAPK11 JNK-9L http://dsigdb.tanlab.org/DSigDBv1.0/displayDrug.py?db=d2_lincs&id=648 PDGFRB MAP4K3 MAP4K2 CSF1R JAK2 HIPK4 STK16 PDGFRA BMP2K RIPK1 MAPK15 HIPK1 MAPK10 MAP2K5 CIT TYK2 PIK3CG FLT3 NEK5 MAP2K4 NEK3 CDKL5 ADCK4 CDK16 MAP3K7 CDKL2 IRAK1 MAPK6 JAK3 MAPK4 JAK1 DYRK1A IRAK3 MAPK8 DYRK1B PIP4K2C PIP4K2B ICK ULK3 STK11 EPHB6 RIOK3 AAK1 GSK3B CLK1 CSNK2A2 CSNK2A1 RIOK2 HIPK3 RIOK1 HIPK2 MAPK9 GSK3A EIF2AK4 KIT MET CDK4 SLK STK36 CDK7 MAP3K19 CLK2 CLK4 CDK9 Neratinib http://dsigdb.tanlab.org/DSigDBv1.0/displayDrug.py?db=d2_lincs&id=1127 MAP4K3 MAP4K2 MAP4K5 MAP4K4 STK10 EGFR MAP2K2 MAP2K1 MAP2K5 AXL MINK1 NEK2 ERBB4 MAP3K3 TNIK MAP3K4 STK26 STK25 STK24 GAK NUAK2 ERBB2 ERBB3 CSK STK3 BLK SLK MERTK EIF2AK4 MAP3K19 LCK BTK CGP74514A http://dsigdb.tanlab.org/DSigDBv1.0/displayDrug.py?db=d2_lincs&id=1116 PLK1 FYN STK10 HIPK3 HIPK2 HIPK1 HIPK4 TYK2 AXL MAP3K9 MAP3K2 GRK7 NTRK1 FGR GRK1 CSNK1D CSNK1E DYRK1A DYRK1B IRAK4 WNK3 CSNK1G2 CSNK1G3 CSNK1G1 RET STK17B CSNK2A2 CSNK2A1 STK17A KIT PAK4 PAK6 PAK7 PAK2 PAK3 ICK PRKCH NUAK1 NUAK2 DCLK1 STK26 JAK2 PHKG1 EPHB1 BLK HCK SBK1 STK32B STK32A RPS6KA3 CSNK1A1 RPS6KA6 MELK STK33 MAP3K3 STK38 CLK1 CLK2 CLK4 LCK PDGFRB EPHA3 EPHA1 MAP3K7 MAPK15 NTRK2 ABL1 NTRK3 FLT3 SIK1 SLC12A7 MAPK3 MAPK1 MAPK6 MAPK7 MAPK4 MARK3 SRC RPS6KA1 GSG2 RPS6KA2 MERTK TAOK1 TAOK2 TAOK3 CSNK1A1L IRAK1 ALK SGK1 PIP5K1C CDK2 CDK3 CDK4 CDK5 CDK7 CDK9 MAP4K1 MAP4K2 EGFR LATS2 MAP2K5 YES1 MINK1 CDK18 TXK CDK13 CDK16 CDK17 CDK14 CDK15 AURKC DAPK3 DAPK1 ULK2 ULK3 ULK1 PIM2 PIM3 PKN1 PRKCD SLK ROCK1 ROCK2 MATK MAP3K11 XMD11-85h http://dsigdb.tanlab.org/DSigDBv1.0/displayDrug.py?db=d2_lincs&id=197 BRSK2 PIP5K1A PRKCD RET MARK4 FLT4 SRPK1 AZ-628 http://dsigdb.tanlab.org/DSigDBv1.0/displayDrug.py?db=d2_lincs&id=859 PDGFRB PDGFRA MAP4K4 EPHA8 EPHA6 EPHA5 EPHA4 EGFR EPHA2 EPHA1 MAPK14 TNIK RIPK2 MAPK11 MAP2K5 CIT ABL1 FLT4 ABL2 RAF1 YES1 FLT1 MINK1 TXK EPHB4 CSF1R FGR SRMS LYN MAPK9 STK10 KDR EPHB2 EPHB3 EPHB1 EPHB6 CSK FRK EPHA3 FYN CDK11A CDK11B RET BLK HCK TNNI3K ZAK RPS6KA6 SRC DDR1 KIT MAPK13 BRAF MAP3K19 TIE1 LCK KIN001-123_WZ-1-84 http://dsigdb.tanlab.org/DSigDBv1.0/displayDrug.py?db=d2_lincs&id=414 STK10 EGFR PLK4 RET MAPK10 MAP2K4 ABL1 FLT4 FLT3 TXK TEC CSF1R TTK SRMS JAK2 JAK3 MAPK8 NUAK2 SRC ERBB4 BLK SLK BMX ITK KIT BTK