Drug Gene Type Source RALOXIFENE HYDROCHLORIDE ESR1 IC50=0.00037(uM) D1 PubChem RALOXIFENE HYDROCHLORIDE ESR2 IC50=0.00037(uM) D1 PubChem RALOXIFENE HYDROCHLORIDE ESR1 IC50=0.00072(uM) D1 PubChem RALOXIFENE HYDROCHLORIDE ESR1 Potency=0.0013(uM) D1 PubChem RALOXIFENE HYDROCHLORIDE ESR1 Ratio Potency (uM)=0.00182629(uM) D1 PubChem RALOXIFENE HYDROCHLORIDE ESR1 IC50=0.002(uM) D1 PubChem RALOXIFENE HYDROCHLORIDE ESR1 Potency=0.0039(uM) D1 PubChem RALOXIFENE HYDROCHLORIDE CYP19A1 Potency=0.0043(uM) D1 PubChem RALOXIFENE HYDROCHLORIDE ESR1 IC50=0.00432(uM) D1 PubChem RALOXIFENE HYDROCHLORIDE ESR2 IC50=0.00432(uM) D1 PubChem RALOXIFENE HYDROCHLORIDE ESR1 ER Potency (uM)=0.00467296(uM) D1 PubChem RALOXIFENE HYDROCHLORIDE CYP19A1 Potency=0.0119(uM) D1 PubChem RALOXIFENE HYDROCHLORIDE ESR1 Potency=0.0188(uM) D1 PubChem RALOXIFENE HYDROCHLORIDE ESR1 Ratio Potency (uM)=0.0194938(uM) D1 PubChem RALOXIFENE HYDROCHLORIDE ESR1 ER Potency (uM)=0.0203361(uM) D1 PubChem RALOXIFENE HYDROCHLORIDE ESR2 IC50=0.043(uM) D1 PubChem RALOXIFENE HYDROCHLORIDE ESR1 Ratio Potency (uM)=0.278822(uM) D1 PubChem RALOXIFENE HYDROCHLORIDE CYP3A4 Potency=2.5119(uM) D1 PubChem RALOXIFENE HYDROCHLORIDE ALDH1A1 Potency=2.8184(uM) D1 PubChem RALOXIFENE HYDROCHLORIDE ALDH1A1 Potency=3.5481(uM) D1 PubChem RALOXIFENE HYDROCHLORIDE ESR1 Potency=4.8966(uM) D1 PubChem RALOXIFENE HYDROCHLORIDE GBA Potency=10.0(uM) D1 PubChem RALOXIFENE HYDROCHLORIDE GMNN Potency=11.2202(uM) D1 PubChem RALOXIFENE HYDROCHLORIDE KCNH2 Potency=12.5893(uM) D1 PubChem RALOXIFENE HYDROCHLORIDE PPARG Potency=15.4845(uM) D1 PubChem RALOXIFENE HYDROCHLORIDE TDP1 Potency=16.7889(uM) D1 PubChem RALOXIFENE HYDROCHLORIDE IDH1 Potency=18.3564(uM) D1 PubChem RALOXIFENE HYDROCHLORIDE MPHOSPH8 Potency=19.9526(uM) D1 PubChem RALOXIFENE HYDROCHLORIDE ESR1 Potency=21.3138(uM) D1 PubChem RALOXIFENE HYDROCHLORIDE AR Potency=21.8724(uM) D1 PubChem RALOXIFENE HYDROCHLORIDE RXRA Potency=25.1189(uM) D1 PubChem RALOXIFENE HYDROCHLORIDE NR1I2 Potency=28.1838(uM) D1 PubChem RALOXIFENE HYDROCHLORIDE PPARG Potency=29.847(uM) D1 PubChem RALOXIFENE HYDROCHLORIDE TP53 Potency=29.8493(uM) D1 PubChem RALOXIFENE HYDROCHLORIDE TP53 Ratio Potency (uM)=31.618(uM) D1 PubChem RALOXIFENE HYDROCHLORIDE PPARD Potency=33.4889(uM) D1 PubChem RALOXIFENE HYDROCHLORIDE PPARG Potency=39.8107(uM) D1 PubChem RALOXIFENE HYDROCHLORIDE NR3C1 Potency=39.8107(uM) D1 PubChem RALOXIFENE HYDROCHLORIDE NR1H4 Potency=44.6684(uM) D1 PubChem RALOXIFENE HYDROCHLORIDE P4HB AC50_uM=45.26(uM) D1 PubChem RALOXIFENE HYDROCHLORIDE HSPB1 Ratio Potency (uM)=51.8676(uM) D1 PubChem RALOXIFENE HYDROCHLORIDE TP53 Potency=61.1306(uM) D1 PubChem RALOXIFENE HYDROCHLORIDE TP53 Ratio Potency (uM)=63.5221(uM) D1 PubChem RALOXIFENE HYDROCHLORIDE APAF1 - D1 PubChem RALOXIFENE HYDROCHLORIDE GFER - D1 PubChem RALOXIFENE HYDROCHLORIDE DRD3 - D1 PubChem RALOXIFENE HYDROCHLORIDE MDM4 - D1 PubChem RALOXIFENE HYDROCHLORIDE MDM2 - D1 PubChem RALOXIFENE HYDROCHLORIDE CYP19A1 - D1 PubChem RALOXIFENE HYDROCHLORIDE ESR1 - D1 PubChem RALOXIFENE HYDROCHLORIDE UBE2N - D1 PubChem RALOXIFENE HYDROCHLORIDE ESR2 - D1 PubChem RALOXIFENE HYDROCHLORIDE KCNQ1 - D1 PubChem RALOXIFENE HYDROCHLORIDE ABCB1 - D1 PubChem RALOXIFENE HYDROCHLORIDE PIP4K2A Potency=None(uM) D1 PubChem RALOXIFENE HYDROCHLORIDE MAP4K2 - D1 PubChem RALOXIFENE HYDROCHLORIDE ALDH1A1 Potency=2818.4(nM) D1 ChEMBL RALOXIFENE HYDROCHLORIDE NR3C1 Potency=39810.7(nM) D1 ChEMBL RALOXIFENE HYDROCHLORIDE NR1H4 Potency=44668.4(nM) D1 ChEMBL RALOXIFENE HYDROCHLORIDE BAZ2B Potency=44668.4(nM) D1 ChEMBL RALOXIFENE HYDROCHLORIDE MAPT Potency=12589.3(nM) D1 ChEMBL RALOXIFENE HYDROCHLORIDE ALDH1A1 Potency=3548.1(nM) D1 ChEMBL RALOXIFENE HYDROCHLORIDE KDM4A Potency=56234.1(nM) D1 ChEMBL RALOXIFENE HYDROCHLORIDE KDM4A Potency=39810.7(nM) D1 ChEMBL RALOXIFENE HYDROCHLORIDE MPHOSPH8 Potency=19952.6(nM) D1 ChEMBL RALOXIFENE HYDROCHLORIDE CYP3A4 Potency=2511.9(nM) D1 ChEMBL RALOXIFENE HYDROCHLORIDE GMNN Potency=11220.2(nM) D1 ChEMBL RALOXIFENE HYDROCHLORIDE P4HB AC50=45260.0(nM) D1 ChEMBL RALOXIFENE HYDROCHLORIDE MAPT Potency=14125.4(nM) D1 ChEMBL RALOXIFENE HYDROCHLORIDE UBE2N IC50=14164.0(nM) D1 ChEMBL RALOXIFENE HYDROCHLORIDE GBA Potency=10000.0(nM) D1 ChEMBL RALOXIFENE HYDROCHLORIDE KCNH2 Potency=12589.3(nM) D1 ChEMBL RALOXIFENE HYDROCHLORIDE PPARG Potency=39810.7(nM) D1 ChEMBL RALOXIFENE HYDROCHLORIDE EHMT2 Potency=22387.2(nM) D1 ChEMBL RALOXIFENE HYDROCHLORIDE HSD17B10 Potency=10000.0(nM) D1 ChEMBL RALOXIFENE HYDROCHLORIDE UBE2N IC50=17531.0(nM) D1 ChEMBL RALOXIFENE HYDROCHLORIDE RXRA Potency=25118.9(nM) D1 ChEMBL RALOXIFENE HYDROCHLORIDE IDH1 Potency=18356.4(nM) D1 ChEMBL RALOXIFENE HYDROCHLORIDE IDH1 Potency=20596.2(nM) D1 ChEMBL