Drug Gene Type Source pergolide DRD2 Ki=0.004(uM) D1 PubChem pergolide HTR1A Ki=0.004(uM) D1 PubChem pergolide DRD3 Ki=0.004(uM) D1 PubChem pergolide DRD3 IC50=0.00539(uM) D1 PubChem pergolide HTR2A IC50=0.014(uM) D1 PubChem pergolide DRD1 Potency=0.0184(uM) D1 PubChem pergolide HTR6 IC50=0.039(uM) D1 PubChem pergolide ADRA2B IC50=0.064(uM) D1 PubChem pergolide HTR2B IC50=0.076(uM) D1 PubChem pergolide DRD2 IC50=0.111(uM) D1 PubChem pergolide KCNH2 IC50=0.12023(uM) D1 PubChem pergolide CYP2D6 IC50=0.2(uM) D1 PubChem pergolide ADRA2A IC50=0.264(uM) D1 PubChem pergolide HTR2C IC50=0.379(uM) D1 PubChem pergolide DRD1 Potency=0.5623(uM) D1 PubChem pergolide DRD1 IC50=0.679(uM) D1 PubChem pergolide ADRA2C IC50=1.41(uM) D1 PubChem pergolide ADRA1D IC50=1.513(uM) D1 PubChem pergolide CYP3A4 Potency=12.5893(uM) D1 PubChem pergolide HTR1A - D1 PubChem pergolide HTR1B - D1 PubChem pergolide HTR1D - D1 PubChem pergolide HTR2C - D1 PubChem pergolide HTR2A - D1 PubChem pergolide HTR2B - D1 PubChem pergolide CYP3A4 Potency=12589.3(nM) D1 ChEMBL pergolide DRD1 Potency=562.3(nM) D1 ChEMBL pergolide DRD1 Potency=18.4(nM) D1 ChEMBL