Drug Gene Type Source amitriptyline HRH1 Ki=0.00112(uM) D1 PubChem amitriptyline SLC6A4 IC50=0.00166(uM) D1 PubChem amitriptyline HRH1 IC50=0.00478(uM) D1 PubChem amitriptyline CHRM4 IC50=0.0053(uM) D1 PubChem amitriptyline HTR2C IC50=0.00605(uM) D1 PubChem amitriptyline CHRM5 IC50=0.00802(uM) D1 PubChem amitriptyline ADRA2B IC50=0.00808(uM) D1 PubChem amitriptyline SLC6A4 Ki=0.00955(uM) D1 PubChem amitriptyline CHRM1 IC50=0.011(uM) D1 PubChem amitriptyline HTR2A IC50=0.015(uM) D1 PubChem amitriptyline SLC6A2 IC50=0.023(uM) D1 PubChem amitriptyline CHRM3 IC50=0.026(uM) D1 PubChem amitriptyline ADRA2C IC50=0.059(uM) D1 PubChem amitriptyline HTR2B IC50=0.07(uM) D1 PubChem amitriptyline CHRM2 IC50=0.081(uM) D1 PubChem amitriptyline DRD1 Ki=0.089(uM) D1 PubChem amitriptyline ADRA1D IC50=0.105(uM) D1 PubChem amitriptyline HTR6 IC50=0.14(uM) D1 PubChem amitriptyline DRD5 Ki=0.17(uM) D1 PubChem amitriptyline DRD3 IC50=0.182(uM) D1 PubChem amitriptyline DRD2 Ki=0.196(uM) D1 PubChem amitriptyline DRD3 Ki=0.206(uM) D1 PubChem amitriptyline ADRA2A IC50=0.351(uM) D1 PubChem amitriptyline DRD1 IC50=0.355(uM) D1 PubChem amitriptyline SLC6A4 IC50=0.54954(uM) D1 PubChem amitriptyline HRH2 IC50=0.73(uM) D1 PubChem amitriptyline SCN9A IC50=1.0(uM) D1 PubChem amitriptyline DRD2 IC50=1.009(uM) D1 PubChem amitriptyline SIGMAR1 IC50=1.031(uM) D1 PubChem amitriptyline DRD1 Potency=1.122(uM) D1 PubChem amitriptyline SCN5A IC50=1.6(uM) D1 PubChem amitriptyline SLC6A2 IC50=2.04174(uM) D1 PubChem amitriptyline SCN2A IC50=3.1(uM) D1 PubChem amitriptyline SCN9A IC50=7.0(uM) D1 PubChem amitriptyline CYP2D6 Potency=7.9433(uM) D1 PubChem amitriptyline KCNH2 IC50=10.0(uM) D1 PubChem amitriptyline SLC6A3 IC50=12.5893(uM) D1 PubChem amitriptyline SLC22A1 IC50=16.9(uM) D1 PubChem amitriptyline KCNH2 IC50=17.5894(uM) D1 PubChem amitriptyline CYP1A2 - D1 PubChem amitriptyline CYP2C9 - D1 PubChem amitriptyline HTR6 - D1 PubChem amitriptyline CYP2D6 - D1 PubChem amitriptyline CYP3A4 - D1 PubChem amitriptyline CYP2D6 Inhibition=None(Unspecified) D1 ChEMBL amitriptyline CYP2C9 Inhibition=None(Unspecified) D1 ChEMBL amitriptyline CYP3A4 Inhibition=None(Unspecified) D1 ChEMBL amitriptyline CYP1A2 Inhibition=None(Unspecified) D1 ChEMBL amitriptyline DRD1 Potency=1122.0(nM) D1 ChEMBL amitriptyline CYP2D6 Potency=7943.3(nM) D1 ChEMBL amitriptyline CYP2D6 AC50=7943.28(nM) D1 ChEMBL