Drug Gene Type Source oxymetazoline ADRA2A Ki=0.00229(uM) D1 PubChem oxymetazoline ADRA2C Ki=0.00501(uM) D1 PubChem oxymetazoline NISCH Ki=0.00619(uM) D1 PubChem oxymetazoline ADRA2A IC50=0.023(uM) D1 PubChem oxymetazoline CYP2D6 Potency=0.0398(uM) D1 PubChem oxymetazoline CYP2D6 IC50=0.2(uM) D1 PubChem oxymetazoline HTR2C IC50=0.578(uM) D1 PubChem oxymetazoline ADRA2B IC50=1.273(uM) D1 PubChem oxymetazoline HTR2A IC50=1.285(uM) D1 PubChem oxymetazoline CHRM5 IC50=1.332(uM) D1 PubChem oxymetazoline HTR6 IC50=1.67(uM) D1 PubChem oxymetazoline ADRA2C IC50=2.633(uM) D1 PubChem oxymetazoline ADRA1D IC50=2.844(uM) D1 PubChem oxymetazoline HTR2B IC50=3.056(uM) D1 PubChem oxymetazoline CHRM4 IC50=3.261(uM) D1 PubChem oxymetazoline CYP2D6 Potency=3.9811(uM) D1 PubChem oxymetazoline TDP1 Potency=10.5931(uM) D1 PubChem oxymetazoline CYP2D6 Potency=12.5893(uM) D1 PubChem oxymetazoline CYP3A4 Potency=15.8489(uM) D1 PubChem oxymetazoline CYP3A4 - D1 PubChem oxymetazoline CYP2D6 - D1 PubChem oxymetazoline HTR2C - D1 PubChem oxymetazoline HTR1B - D1 PubChem oxymetazoline HTR1D - D1 PubChem oxymetazoline CYP2D6 Potency=39.8(nM) D1 ChEMBL oxymetazoline CYP3A4 Potency=15848.9(nM) D1 ChEMBL oxymetazoline CYP2D6 Potency=12589.3(nM) D1 ChEMBL oxymetazoline CYP2D6 AC50=39.81(nM) D1 ChEMBL oxymetazoline CYP2D6 AC50=3981.07(nM) D1 ChEMBL oxymetazoline CYP2D6 Potency=3981.1(nM) D1 ChEMBL oxymetazoline ADRA2A Activity=None(Unspecified) D1 ChEMBL oxymetazoline CYP2D6 AC50=12589.2(nM) D1 ChEMBL oxymetazoline CYP3A4 AC50=15848.9(nM) D1 ChEMBL