Drug Gene Type Source chlorhexidine SLC22A1 IC50=0.21(uM) D1 PubChem chlorhexidine SLC22A2 IC50=0.4(uM) D1 PubChem chlorhexidine SLC22A3 IC50=0.41(uM) D1 PubChem chlorhexidine SLC47A2 IC50=0.5(uM) D1 PubChem chlorhexidine SLC47A1 IC50=0.7(uM) D1 PubChem chlorhexidine PLIN5 IC50=1.655(uM) D1 PubChem chlorhexidine ABHD5 IC50=1.655(uM) D1 PubChem chlorhexidine RAD52 AC50_uM=1.7(uM) D1 PubChem chlorhexidine MC4R IC50=1.997(uM) D1 PubChem chlorhexidine ABHD5 IC50=2.138(uM) D1 PubChem chlorhexidine PLIN1 IC50=2.138(uM) D1 PubChem chlorhexidine PLIN1 IC50=2.175(uM) D1 PubChem chlorhexidine ABHD5 IC50=2.175(uM) D1 PubChem chlorhexidine UBE2N IC50=2.197(uM) D1 PubChem chlorhexidine NFE2L2 Ratio Potency (uM)=2.2835(uM) D1 PubChem chlorhexidine PLIN1 IC50=2.312(uM) D1 PubChem chlorhexidine PLIN5 IC50=2.635(uM) D1 PubChem chlorhexidine ABHD5 IC50=2.635(uM) D1 PubChem chlorhexidine ABHD5 IC50=2.642(uM) D1 PubChem chlorhexidine PLIN5 IC50=2.642(uM) D1 PubChem chlorhexidine UBE2N IC50=3.012(uM) D1 PubChem chlorhexidine AR Ratio Potency (uM)=3.30503(uM) D1 PubChem chlorhexidine AR Ratio Potency (uM)=3.72066(uM) D1 PubChem chlorhexidine PLIN5 IC50=4.022(uM) D1 PubChem chlorhexidine ABHD5 IC50=4.022(uM) D1 PubChem chlorhexidine MLLT3 AC50_uM=5.27(uM) D1 PubChem chlorhexidine PAX8 AC50_uM=5.69(uM) D1 PubChem chlorhexidine PLIN5 IC50=6.217(uM) D1 PubChem chlorhexidine ABHD5 IC50=6.217(uM) D1 PubChem chlorhexidine GBA Potency=6.3096(uM) D1 PubChem chlorhexidine ESR1 Ratio Potency (uM)=6.61637(uM) D1 PubChem chlorhexidine PLIN5 IC50=6.856(uM) D1 PubChem chlorhexidine ABHD5 IC50=6.856(uM) D1 PubChem chlorhexidine MMP2 IC50=7.63(uM) D1 PubChem chlorhexidine MMP9 IC50=7.63(uM) D1 PubChem chlorhexidine CYP2D6 Potency=7.9433(uM) D1 PubChem chlorhexidine HKDC1 IC50_Mean=8.99(uM) D1 PubChem chlorhexidine ESR1 Ratio Potency (uM)=9.31485(uM) D1 PubChem chlorhexidine ESR1 Potency=12.2261(uM) D1 PubChem chlorhexidine PAX8 AC50_uM=12.25(uM) D1 PubChem chlorhexidine TDP1 Potency=12.9953(uM) D1 PubChem chlorhexidine HTT Potency=14.1254(uM) D1 PubChem chlorhexidine IDH1 Potency=14.581(uM) D1 PubChem chlorhexidine GBA Potency=16.3433(uM) D1 PubChem chlorhexidine TDP1 Potency=16.3601(uM) D1 PubChem chlorhexidine AR Ratio Potency (uM)=16.9301(uM) D1 PubChem chlorhexidine AR Potency=16.9301(uM) D1 PubChem chlorhexidine TDP1 Potency=18.8375(uM) D1 PubChem chlorhexidine ESR1 Potency=19.3127(uM) D1 PubChem chlorhexidine PAX8 AC50_uM=20.02(uM) D1 PubChem chlorhexidine PAX8 AC50_uM=21.59(uM) D1 PubChem chlorhexidine CYP19A1 Potency=24.1139(uM) D1 PubChem chlorhexidine CYP19A1 Potency=24.1881(uM) D1 PubChem chlorhexidine TARDBP Potency=25.1189(uM) D1 PubChem chlorhexidine RORC Potency=26.6032(uM) D1 PubChem chlorhexidine ATXN2 Potency=31.6228(uM) D1 PubChem chlorhexidine PAX8 AC50_uM=33.88(uM) D1 PubChem chlorhexidine PPARD Potency=38.6622(uM) D1 PubChem chlorhexidine NR1H4 Potency=48.6728(uM) D1 PubChem chlorhexidine SNUPN Potency=51.7352(uM) D1 PubChem chlorhexidine KPNB1 Potency=51.7352(uM) D1 PubChem chlorhexidine AR Potency=54.1504(uM) D1 PubChem chlorhexidine USP1 Potency=56.2341(uM) D1 PubChem chlorhexidine AR Potency=60.5715(uM) D1 PubChem chlorhexidine GSK3A AC50_uM=162.8(uM) D1 PubChem chlorhexidine DRD1 - D1 PubChem chlorhexidine CYP2D6 - D1 PubChem chlorhexidine ABCB1 - D1 PubChem chlorhexidine BARD1 - D1 PubChem chlorhexidine NLRP3 - D1 PubChem chlorhexidine MAPT - D1 PubChem chlorhexidine APAF1 - D1 PubChem chlorhexidine AR Potency=None(uM) D1 PubChem chlorhexidine UBE2N - D1 PubChem chlorhexidine RAD52 - D1 PubChem chlorhexidine CYP1A2 - D1 PubChem chlorhexidine MC4R - D1 PubChem chlorhexidine MDM4 - D1 PubChem chlorhexidine PLIN5 - D1 PubChem chlorhexidine MDM2 - D1 PubChem chlorhexidine RAD54L - D1 PubChem chlorhexidine HKDC1 - D1 PubChem chlorhexidine IL1B - D1 PubChem chlorhexidine KCNQ1 - D1 PubChem chlorhexidine PAX8 - D1 PubChem chlorhexidine MLLT3 - D1 PubChem chlorhexidine MRGPRX1 - D1 PubChem chlorhexidine BRCA1 - D1 PubChem chlorhexidine ABHD5 - D1 PubChem chlorhexidine PPP1CA - D1 PubChem chlorhexidine CYP2D6 AC50=7943.28(nM) D1 ChEMBL chlorhexidine CYP2D6 Potency=7943.3(nM) D1 ChEMBL chlorhexidine USP1 Potency=56234.1(nM) D1 ChEMBL chlorhexidine GBA Potency=16343.3(nM) D1 ChEMBL chlorhexidine UBE2N IC50=3012.0(nM) D1 ChEMBL chlorhexidine RORC Potency=26603.2(nM) D1 ChEMBL chlorhexidine ATXN2 Potency=31622.8(nM) D1 ChEMBL chlorhexidine PLIN1 IC50=2312.0(nM) D1 ChEMBL chlorhexidine MC4R IC50=1997.0(nM) D1 ChEMBL chlorhexidine GBA Potency=6309.6(nM) D1 ChEMBL chlorhexidine EHMT2 Potency=14125.4(nM) D1 ChEMBL chlorhexidine TARDBP Potency=25118.9(nM) D1 ChEMBL chlorhexidine IDH1 Potency=14581.0(nM) D1 ChEMBL chlorhexidine HTT Potency=14125.4(nM) D1 ChEMBL chlorhexidine HKDC1 IC50=8990.0(nM) D1 ChEMBL chlorhexidine UBE2N IC50=2197.0(nM) D1 ChEMBL chlorhexidine PAX8 AC50=5690.0(nM) D1 ChEMBL chlorhexidine RAD52 AC50=1700.0(nM) D1 ChEMBL